These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
3. Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers. Dal Corso A; Caruso M; Belvisi L; Arosio D; Piarulli U; Albanese C; Gasparri F; Marsiglio A; Sola F; Troiani S; Valsasina B; Pignataro L; Donati D; Gennari C Chemistry; 2015 Apr; 21(18):6921-9. PubMed ID: 25784522 [TBL] [Abstract][Full Text] [Related]
4. Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α Raposo Moreira Dias A; Pina A; Dal Corso A; Arosio D; Belvisi L; Pignataro L; Caruso M; Gennari C Chemistry; 2017 Oct; 23(58):14410-14415. PubMed ID: 28816404 [TBL] [Abstract][Full Text] [Related]
5. Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting. Bodero L; López Rivas P; Korsak B; Hechler T; Pahl A; Müller C; Arosio D; Pignataro L; Gennari C; Piarulli U Beilstein J Org Chem; 2018; 14():407-415. PubMed ID: 29520305 [TBL] [Abstract][Full Text] [Related]
6. Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonists. Panzeri S; Zanella S; Arosio D; Vahdati L; Dal Corso A; Pignataro L; Paolillo M; Schinelli S; Belvisi L; Gennari C; Piarulli U Chemistry; 2015 Apr; 21(16):6265-71. PubMed ID: 25761230 [TBL] [Abstract][Full Text] [Related]
7. RGD Peptidomimetic MMAE-Conjugate Addressing Integrin αVβ3-Expressing Cells with High Targeting Index. Paulus J; Nachtigall B; Meyer P; Sewald N Chemistry; 2023 Feb; 29(12):e202203476. PubMed ID: 36454662 [TBL] [Abstract][Full Text] [Related]
8. Conjugates of Cryptophycin and RGD or Borbély A; Figueras E; Martins A; Bodero L; Raposo Moreira Dias A; López Rivas P; Pina A; Arosio D; Gallinari P; Frese M; Steinkühler C; Gennari C; Piarulli U; Sewald N ChemistryOpen; 2019 Jun; 8(6):737-742. PubMed ID: 31275795 [TBL] [Abstract][Full Text] [Related]
9. Cyclic RGD and Panzeri S; Arosio D; Gazzola S; Belvisi L; Civera M; Potenza D; Vasile F; Kemker I; Ertl T; Sewald N; Reiser O; Piarulli U Molecules; 2020 Dec; 25(24):. PubMed ID: 33339382 [TBL] [Abstract][Full Text] [Related]
10. Synthesis and Biological Characterization of Monomeric and Tetrameric RGD-Cryptophycin Conjugates. Borbély A; Thoreau F; Figueras E; Kadri M; Coll JL; Boturyn D; Sewald N Chemistry; 2020 Feb; 26(12):2602-2605. PubMed ID: 31943410 [TBL] [Abstract][Full Text] [Related]
11. Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake. Pina A; Kadri M; Arosio D; Dal Corso A; Coll JL; Gennari C; Boturyn D Chemistry; 2020 Jun; 26(33):7492-7496. PubMed ID: 32227540 [TBL] [Abstract][Full Text] [Related]
12. Synthesis and biological evaluation (in vitro and in vivo) of cyclic arginine-glycine-aspartate (RGD) peptidomimetic-paclitaxel conjugates targeting integrin αVβ3. Colombo R; Mingozzi M; Belvisi L; Arosio D; Piarulli U; Carenini N; Perego P; Zaffaroni N; De Cesare M; Castiglioni V; Scanziani E; Gennari C J Med Chem; 2012 Dec; 55(23):10460-74. PubMed ID: 23140358 [TBL] [Abstract][Full Text] [Related]
13. Optimizing the enzymatic release of MMAE from Zambra M; Ranđelović I; Talarico F; Borbély A; Svajda L; Tóvári J; Mező G; Bodero L; Colombo S; Arrigoni F; Fasola E; Gazzola S; Piarulli U Front Pharmacol; 2023; 14():1215694. PubMed ID: 37492088 [TBL] [Abstract][Full Text] [Related]
14. Synthesis and Evaluation of a Non-Peptide Small-Molecule Drug Conjugate Targeting Integrin α Paulus J; Sewald N Front Chem; 2022; 10():869639. PubMed ID: 35480387 [TBL] [Abstract][Full Text] [Related]
15. Integrin-targeted delivery into cancer cells of a Pt(IV) pro-drug through conjugation to RGD-containing peptides. Massaguer A; González-Cantó A; Escribano E; Barrabés S; Artigas G; Moreno V; Marchán V Dalton Trans; 2015 Jan; 44(1):202-12. PubMed ID: 25369773 [TBL] [Abstract][Full Text] [Related]
16. High-Affinity "Click" RGD Peptidomimetics as Radiolabeled Probes for Imaging α Piras M; Testa A; Fleming IN; Dall'Angelo S; Andriu A; Menta S; Mori M; Brown GD; Forster D; Williams KJ; Zanda M ChemMedChem; 2017 Jul; 12(14):1142-1151. PubMed ID: 28608961 [TBL] [Abstract][Full Text] [Related]
17. Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate. Raposo Moreira Dias A; Pina A; Dean A; Lerchen HG; Caruso M; Gasparri F; Fraietta I; Troiani S; Arosio D; Belvisi L; Pignataro L; Dal Corso A; Gennari C Chemistry; 2019 Feb; 25(7):1696-1700. PubMed ID: 30452790 [TBL] [Abstract][Full Text] [Related]
18. The Importance of Detail: How Differences in Ligand Structures Determine Distinct Functional Responses in Integrin α Paladino A; Civera M; Curnis F; Paolillo M; Gennari C; Piarulli U; Corti A; Belvisi L; Colombo G Chemistry; 2019 Apr; 25(23):5959-5970. PubMed ID: 30811704 [TBL] [Abstract][Full Text] [Related]