BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

89 related articles for article (PubMed ID: 30973227)

  • 1. Development of a NanoBRET-Based Sensitive Screening Method for CXCR4 Ligands.
    Sakyiamah MM; Nomura W; Kobayakawa T; Tamamura H
    Bioconjug Chem; 2019 May; 30(5):1442-1450. PubMed ID: 30973227
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis and biological evaluation of low molecular weight CXCR4 ligands.
    Sakyiamah MM; Kobayakawa T; Fujino M; Konno M; Narumi T; Tanaka T; Nomura W; Yamamoto N; Murakami T; Tamamura H
    Bioorg Med Chem; 2019 Mar; 27(6):1130-1138. PubMed ID: 30772128
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Fluorophore labeling enables imaging and evaluation of specific CXCR4-ligand interaction at the cell membrane for fluorescence-based screening.
    Nomura W; Tanabe Y; Tsutsumi H; Tanaka T; Ohba K; Yamamoto N; Tamamura H
    Bioconjug Chem; 2008 Sep; 19(9):1917-20. PubMed ID: 18707146
    [TBL] [Abstract][Full Text] [Related]  

  • 4. A radiogallium-DOTA-based bivalent peptidic ligand targeting a chemokine receptor, CXCR4, for tumor imaging.
    Sano K; Masuda R; Hisada H; Oishi S; Shimokawa K; Ono M; Fujii N; Saji H; Mukai T
    Bioorg Med Chem Lett; 2014 Mar; 24(5):1386-8. PubMed ID: 24491461
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Discovery of Environment-Sensitive Fluorescent Ligands of β-Adrenergic Receptors for Cell Imaging and NanoBRET Assay.
    Li W; Ma Z; Chen J; Dong G; Du L; Li M
    Anal Chem; 2022 May; 94(19):7021-7028. PubMed ID: 35504022
    [TBL] [Abstract][Full Text] [Related]  

  • 6. New Horizons on Molecular Pharmacology Applied to Drug Discovery: When Resonance Overcomes Radioligand Binding.
    Pernomian L; Gomes MS; Moreira JD; da Silva CHTP; Rosa JMC; Cardoso CRB
    Curr Radiopharm; 2017; 10(1):16-20. PubMed ID: 28183248
    [TBL] [Abstract][Full Text] [Related]  

  • 7. The CXCR4 agonist ligand stromal derived factor-1 maintains high affinity for receptors in both Galpha(i)-coupled and uncoupled states.
    Di Salvo J; Koch GE; Johnson KE; Blake AD; Daugherty BL; DeMartino JA; Sirotina-Meisher A; Liu Y; Springer MS; Cascieri MA; Sullivan KA
    Eur J Pharmacol; 2000 Dec; 409(2):143-54. PubMed ID: 11104827
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A novel CXCR4-selective high-affinity fluorescent probe and its application in competitive binding assays.
    Yang Y; Zhang Q; Gao M; Yang X; Huang Z; An J
    Biochemistry; 2014 Aug; 53(30):4881-3. PubMed ID: 25058910
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Development and application of fluorescent SDF-1 derivatives.
    Masuda R; Oishi S; Tanahara N; Ohno H; Hirasawa A; Tsujimoto G; Kodama E; Matsuoka M; Fujii N
    Future Med Chem; 2012 May; 4(7):837-44. PubMed ID: 22571609
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Microtiter plate-based antibody-competition assay to determine binding affinities and plasma/blood stability of CXCR4 ligands.
    Harms M; Gilg A; Ständker L; Beer AJ; Mayer B; Rasche V; Gruber CW; Münch J
    Sci Rep; 2020 Sep; 10(1):16036. PubMed ID: 32994431
    [TBL] [Abstract][Full Text] [Related]  

  • 11. CXCR4 Antagonists: A Screening Strategy for Identification of Functionally Selective Ligands.
    Castaldo C; Benicchi T; Otrocka M; Mori E; Pilli E; Ferruzzi P; Valensin S; Diamanti D; Fecke W; Varrone M; Porcari V
    J Biomol Screen; 2014 Jul; 19(6):859-69. PubMed ID: 24632660
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Peptide-functionalized luminescent iridium complexes for lifetime imaging of CXCR4 expression.
    Kuil J; Steunenberg P; Chin PT; Oldenburg J; Jalink K; Velders AH; van Leeuwen FW
    Chembiochem; 2011 Aug; 12(12):1897-903. PubMed ID: 21739561
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Regulation of CXCR4 receptor dimerization by the chemokine SDF-1alpha and the HIV-1 coat protein gp120: a fluorescence resonance energy transfer (FRET) study.
    Toth PT; Ren D; Miller RJ
    J Pharmacol Exp Ther; 2004 Jul; 310(1):8-17. PubMed ID: 15014135
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids.
    Tanaka T; Nomura W; Narumi T; Esaka A; Oishi S; Ohashi N; Itotani K; Evans BJ; Wang ZX; Peiper SC; Fujii N; Tamamura H
    Org Biomol Chem; 2009 Sep; 7(18):3805-9. PubMed ID: 19707686
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Bivalent 14-mer peptide ligands of CXCR4 with polyproline linkers with anti-chemotactic activity against Jurkat cells.
    Tanaka T; Aoki T; Nomura W; Tamamura H
    J Pept Sci; 2017 Jul; 23(7-8):574-580. PubMed ID: 28078743
    [TBL] [Abstract][Full Text] [Related]  

  • 16. NanoBRET ligand binding at a GPCR under endogenous promotion facilitated by CRISPR/Cas9 genome editing.
    White CW; Johnstone EKM; See HB; Pfleger KDG
    Cell Signal; 2019 Feb; 54():27-34. PubMed ID: 30471466
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Measuring Protein-Protein Interactions in Cells using Nanoluciferase Bioluminescence Resonance Energy Transfer (NanoBRET) Assay.
    Szewczyk MM; Owens DDG; Barsyte-Lovejoy D
    Methods Mol Biol; 2023; 2706():137-148. PubMed ID: 37558946
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Development of a receptor-targeted gene delivery system using CXCR4 ligand-conjugated cross-linking peptides.
    Egorova A; Bogacheva M; Shubina A; Baranov V; Kiselev A
    J Gene Med; 2014; 16(11-12):336-51. PubMed ID: 25382058
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Fluorescent CXCR4 targeting peptide as alternative for antibody staining in Ewing sarcoma.
    Sand LGL; Buckle T; van Leeuwen FWB; Corver WE; Kruisselbrink AB; Jochemsen AG; Hogendoorn PCW; Szuhai K
    BMC Cancer; 2017 May; 17(1):383. PubMed ID: 28549419
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Use of a new proximity assay (NanoBRET) to investigate the ligand-binding characteristics of three fluorescent ligands to the human
    Soave M; Stoddart LA; Brown A; Woolard J; Hill SJ
    Pharmacol Res Perspect; 2016 Oct; 4(5):e00250. PubMed ID: 27588207
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.