These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

170 related articles for article (PubMed ID: 31082763)

  • 1. Discovery of tropinone-thiazole derivatives as potent caspase 3/7 activators, and noncompetitive tyrosinase inhibitors with high antiproliferative activity: Rational design, one-pot tricomponent synthesis, and lipophilicity determination.
    Piechowska K; Świtalska M; Cytarska J; Jaroch K; Łuczykowski K; Chałupka J; Wietrzyk J; Misiura K; Bojko B; Kruszewski S; Łączkowski KZ
    Eur J Med Chem; 2019 Aug; 175():162-171. PubMed ID: 31082763
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Tropinone-Derived Alkaloids as Potent Anticancer Agents: Synthesis, Tyrosinase Inhibition, Mechanism of Action, DFT Calculation, and Molecular Docking Studies.
    Piechowska K; Mizerska-Kowalska M; Zdzisińska B; Cytarska J; Baranowska-Łączkowska A; Jaroch K; Łuczykowski K; Płaziński W; Bojko B; Kruszewski S; Misiura K; Łączkowski KZ
    Int J Mol Sci; 2020 Nov; 21(23):. PubMed ID: 33260768
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Effect of the dichloro-substitution on antiproliferative activity of phthalimide-thiazole derivatives. Rational design, synthesis, elastase, caspase 3/7, and EGFR tyrosine kinase activity and molecular modeling study.
    Donarska B; Świtalska M; Płaziński W; Wietrzyk J; Łączkowski KZ
    Bioorg Chem; 2021 May; 110():104819. PubMed ID: 33752144
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and evaluation of 2(3H)-thiazole thiones as tyrosinase inhibitors.
    Emami S; Hosseinimehr SJ; Shahrbandi K; Enayati AA; Esmaeeli Z
    Arch Pharm (Weinheim); 2012 Aug; 345(8):629-37. PubMed ID: 22532401
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Benzo[b]thiophene-thiazoles as potent anti-Toxoplasma gondii agents: Design, synthesis, tyrosinase/tyrosine hydroxylase inhibitors, molecular docking study, and antioxidant activity.
    Rosada B; Bekier A; Cytarska J; Płaziński W; Zavyalova O; Sikora A; Dzitko K; Łączkowski KZ
    Eur J Med Chem; 2019 Dec; 184():111765. PubMed ID: 31629163
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Structure-based modification of 3-/4-aminoacetophenones giving a profound change of activity on tyrosinase: from potent activators to highly efficient inhibitors.
    You A; Zhou J; Song S; Zhu G; Song H; Yi W
    Eur J Med Chem; 2015 Mar; 93():255-62. PubMed ID: 25686594
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis, molecular docking studies of coumarinyl-pyrazolinyl substituted thiazoles as non-competitive inhibitors of mushroom tyrosinase.
    Saeed A; Mahesar PA; Channar PA; Abbas Q; Larik FA; Hassan M; Raza H; Seo SY
    Bioorg Chem; 2017 Oct; 74():187-196. PubMed ID: 28837887
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and in vitro antiproliferative activity of thiazole-based nitrogen mustards: the hydrogen bonding interaction between model systems and nucleobases.
    Łączkowski KZ; Misiura K; Świtalska M; Wietrzyk J; Łączkowska AB; Fernandez B; Paneth A; Plech T
    Anticancer Agents Med Chem; 2014; 14(9):1271-81. PubMed ID: 25060901
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel synthetic kojic acid-methimazole derivatives inhibit mushroom tyrosinase and melanogenesis.
    Chen MJ; Hung CC; Chen YR; Lai ST; Chan CF
    J Biosci Bioeng; 2016 Dec; 122(6):666-672. PubMed ID: 27353860
    [TBL] [Abstract][Full Text] [Related]  

  • 10. New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies.
    Pintus F; Matos MJ; Vilar S; Hripcsak G; Varela C; Uriarte E; Santana L; Borges F; Medda R; Di Petrillo A; Era B; Fais A
    Bioorg Med Chem; 2017 Mar; 25(5):1687-1695. PubMed ID: 28189394
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and preliminary in vitro biological evaluation of 5-chloro-2-(substituted phenyl)benzo[d]thiazole derivatives designed as novel antimelanogenesis agents.
    Ha YM; Uehara Y; Park D; Jeong HO; Park JY; Park YJ; Lee JY; Lee HJ; Song YM; Moon HR; Chung HY
    Appl Biochem Biotechnol; 2012 Nov; 168(6):1416-33. PubMed ID: 22968587
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Potent inhibitory effects of N-aryl S-alkylthiocarbamate derivatives on the dopa oxidase activity of mushroom tyrosinase.
    Lee KH; Koketsu M; Choi SY; Lee KJ; Lee P; Ishihara H; Kim SY
    Chem Pharm Bull (Tokyo); 2005 Jul; 53(7):747-9. PubMed ID: 15997128
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Design, synthesis, kinetic mechanism and molecular docking studies of novel 1-pentanoyl-3-arylthioureas as inhibitors of mushroom tyrosinase and free radical scavengers.
    Larik FA; Saeed A; Channar PA; Muqadar U; Abbas Q; Hassan M; Seo SY; Bolte M
    Eur J Med Chem; 2017 Dec; 141():273-281. PubMed ID: 29040952
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis of chiral pyrazolo[4,3-e][1,2,4]triazine sulfonamides with tyrosinase and urease inhibitory activity.
    Mojzych M; Tarasiuk P; Kotwica-Mojzych K; Rafiq M; Seo SY; Nicewicz M; Fornal E
    J Enzyme Inhib Med Chem; 2017 Dec; 32(1):99-105. PubMed ID: 27778522
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Evaluation of thiazolidinone derivatives as a new class of mushroom tyrosinase inhibitors.
    Rezaei M; Mohammadi HT; Mahdavi A; Shourian M; Ghafouri H
    Int J Biol Macromol; 2018 Mar; 108():205-213. PubMed ID: 29180052
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and biological evaluation of novel hydroxybenzaldehyde-based kojic acid analogues as inhibitors of mushroom tyrosinase.
    Xie W; Zhang H; He J; Zhang J; Yu Q; Luo C; Li S
    Bioorg Med Chem Lett; 2017 Feb; 27(3):530-532. PubMed ID: 28011217
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Tyrosinase inhibitory components from Aloe vera and their antiviral activity.
    Kim JH; Yoon JY; Yang SY; Choi SK; Kwon SJ; Cho IS; Jeong MH; Ho Kim Y; Choi GS
    J Enzyme Inhib Med Chem; 2017 Dec; 32(1):78-83. PubMed ID: 27778516
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Inhibitory effects of novel synthetic methimazole derivatives on mushroom tyrosinase and melanogenesis.
    Chan CF; Lai ST; Guo YC; Chen MJ
    Bioorg Med Chem; 2014 May; 22(9):2809-15. PubMed ID: 24703463
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design and synthesis of thiourea derivatives with sulfur-containing heterocyclic scaffolds as potential tyrosinase inhibitors.
    Liu P; Shu C; Liu L; Huang Q; Peng Y
    Bioorg Med Chem; 2016 Apr; 24(8):1866-71. PubMed ID: 26972919
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design and synthesis of novel hydroxypyridinone derivatives as potential tyrosinase inhibitors.
    Zhao DY; Zhang MX; Dong XW; Hu YZ; Dai XY; Wei X; Hider RC; Zhang JC; Zhou T
    Bioorg Med Chem Lett; 2016 Jul; 26(13):3103-3108. PubMed ID: 27185329
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.