These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

294 related articles for article (PubMed ID: 31124602)

  • 1. Investigation of Dipicolinic Acid Isosteres for the Inhibition of Metallo-β-Lactamases.
    Chen AY; Thomas PW; Cheng Z; Xu NY; Tierney DL; Crowder MW; Fast W; Cohen SM
    ChemMedChem; 2019 Jul; 14(13):1271-1282. PubMed ID: 31124602
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Probing the mechanisms of inhibition for various inhibitors of metallo-β-lactamases VIM-2 and NDM-1.
    Thomas CA; Cheng Z; Yang K; Hellwarth E; Yurkiewicz CJ; Baxter FM; Fullington SA; Klinsky SA; Otto JL; Chen AY; Cohen SM; Crowder MW
    J Inorg Biochem; 2020 Sep; 210():111123. PubMed ID: 32622213
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Dipicolinic Acid Derivatives as Inhibitors of New Delhi Metallo-β-lactamase-1.
    Chen AY; Thomas PW; Stewart AC; Bergstrom A; Cheng Z; Miller C; Bethel CR; Marshall SH; Credille CV; Riley CL; Page RC; Bonomo RA; Crowder MW; Tierney DL; Fast W; Cohen SM
    J Med Chem; 2017 Sep; 60(17):7267-7283. PubMed ID: 28809565
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Recent research and development of NDM-1 inhibitors.
    Wang T; Xu K; Zhao L; Tong R; Xiong L; Shi J
    Eur J Med Chem; 2021 Nov; 223():113667. PubMed ID: 34225181
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Probing the Interaction of Aspergillomarasmine A with Metallo-β-lactamases NDM-1, VIM-2, and IMP-7.
    Bergstrom A; Katko A; Adkins Z; Hill J; Cheng Z; Burnett M; Yang H; Aitha M; Mehaffey MR; Brodbelt JS; Tehrani KHME; Martin NI; Bonomo RA; Page RC; Tierney DL; Fast W; Wright GD; Crowder MW
    ACS Infect Dis; 2018 Feb; 4(2):135-145. PubMed ID: 29091730
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design of dipicolinic acid derivatives as New Delhi metallo-β-lactamase-1 inhibitors using a combined computational approach.
    Wang X; Gao Y; Yu Y; Yang Y; Wang G; Sun L; Niu X
    J Biomol Struct Dyn; 2020 Jul; 38(11):3384-3395. PubMed ID: 31549586
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and Preclinical Evaluation of TPA-Based Zinc Chelators as Metallo-β-lactamase Inhibitors.
    Schnaars C; Kildahl-Andersen G; Prandina A; Popal R; Radix S; Le Borgne M; Gjøen T; Andresen AMS; Heikal A; Økstad OA; Fröhlich C; Samuelsen Ø; Lauksund S; Jordheim LP; Rongved P; Åstrand OAH
    ACS Infect Dis; 2018 Sep; 4(9):1407-1422. PubMed ID: 30022668
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Kinetics, Thermodynamics, and Structural Effects of Quinoline-2-Carboxylates, Zinc-Binding Inhibitors of New Delhi Metallo-β-lactamase-1 Re-sensitizing Multidrug-Resistant Bacteria for Carbapenems.
    Jia Y; Schroeder B; Pfeifer Y; Fröhlich C; Deng L; Arkona C; Kuropka B; Sticht J; Ataka K; Bergemann S; Wolber G; Nitsche C; Mielke M; Leiros HS; Werner G; Rademann J
    J Med Chem; 2023 Sep; 66(17):11761-11791. PubMed ID: 37585683
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Metallo-β-lactamase inhibitors by bioisosteric replacement: Preparation, activity and binding.
    Skagseth S; Akhter S; Paulsen MH; Muhammad Z; Lauksund S; Samuelsen Ø; Leiros HS; Bayer A
    Eur J Med Chem; 2017 Jul; 135():159-173. PubMed ID: 28445786
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Iminodiacetic Acid as a Novel Metal-Binding Pharmacophore for New Delhi Metallo-β-lactamase Inhibitor Development.
    Chen AY; Thomas CA; Thomas PW; Yang K; Cheng Z; Fast W; Crowder MW; Cohen SM
    ChemMedChem; 2020 Jul; 15(14):1272-1282. PubMed ID: 32315115
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Stereochemically altered cephalosporins as potent inhibitors of New Delhi metallo-β-lactamases.
    Hu L; Yang H; Yu T; Chen F; Liu R; Xue S; Zhang S; Mao W; Ji C; Wang H; Xie H
    Eur J Med Chem; 2022 Mar; 232():114174. PubMed ID: 35152091
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors.
    Gavara L; Sevaille L; De Luca F; Mercuri P; Bebrone C; Feller G; Legru A; Cerboni G; Tanfoni S; Baud D; Cutolo G; Bestgen B; Chelini G; Verdirosa F; Sannio F; Pozzi C; Benvenuti M; Kwapien K; Fischer M; Becker K; Frère JM; Mangani S; Gresh N; Berthomieu D; Galleni M; Docquier JD; Hernandez JF
    Eur J Med Chem; 2020 Dec; 208():112720. PubMed ID: 32937203
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Aspergillomarasmine A inhibits metallo-β-lactamases by selectively sequestering Zn
    Sychantha D; Rotondo CM; Tehrani KHME; Martin NI; Wright GD
    J Biol Chem; 2021 Aug; 297(2):100918. PubMed ID: 34181945
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Fragment-based discovery of inhibitor scaffolds targeting the metallo-β-lactamases NDM-1 and VIM-2.
    Christopeit T; Leiros HK
    Bioorg Med Chem Lett; 2016 Apr; 26(8):1973-7. PubMed ID: 26976213
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Efforts towards the inhibitor design for New Delhi metallo-beta-lactamase (NDM-1).
    Nagulapalli Venkata KC; Ellebrecht M; Tripathi SK
    Eur J Med Chem; 2021 Dec; 225():113747. PubMed ID: 34391033
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Discovery of a novel covalent non-β-lactam inhibitor of the metallo-β-lactamase NDM-1.
    Christopeit T; Albert A; Leiros HS
    Bioorg Med Chem; 2016 Jul; 24(13):2947-2953. PubMed ID: 27184103
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Structural and biochemical analysis of the metallo-β-lactamase L1 from emerging pathogen Stenotrophomonas maltophilia revealed the subtle but distinct di-metal scaffold for catalytic activity.
    Kim Y; Maltseva N; Wilamowski M; Tesar C; Endres M; Joachimiak A
    Protein Sci; 2020 Mar; 29(3):723-743. PubMed ID: 31846104
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Structure-guided optimization of D-captopril for discovery of potent NDM-1 inhibitors.
    Ma G; Wang S; Wu K; Zhang W; Ahmad A; Hao Q; Lei X; Zhang H
    Bioorg Med Chem; 2021 Jan; 29():115902. PubMed ID: 33302045
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of Aspergillomarasmine A derivatives as novel NDM-1 inhibitor to overcome antibiotics resistance.
    Zhang J; Wang S; Wei Q; Guo Q; Bai Y; Yang S; Song F; Zhang L; Lei X
    Bioorg Med Chem; 2017 Oct; 25(19):5133-5141. PubMed ID: 28784300
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Thermokinetic profile of NDM-1 and its inhibition by small carboxylic acids.
    Wang Q; He Y; Lu R; Wang WM; Yang KW; Fan HM; Jin Y; Blackburn GM
    Biosci Rep; 2018 Apr; 38(2):. PubMed ID: 29507059
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 15.