133 related articles for article (PubMed ID: 31186146)
1. Defined concatenated α6α1β3γ2 GABA
Simeone X; Iorio MT; Siebert DCB; Rehman S; Schnürch M; Mihovilovic MD; Ernst M
Bioorg Med Chem; 2019 Jul; 27(14):3167-3178. PubMed ID: 31186146
[TBL] [Abstract][Full Text] [Related]
2. Behavioural interaction of pyrazoloquinolinone positive allosteric modulators at α6GABA
Divović Matović B; Knutson D; Mitrović J; Stevanović V; Stanojević B; Savić S; Cook JM; Savić MM
Basic Clin Pharmacol Toxicol; 2022 Dec; 131(6):514-524. PubMed ID: 36180380
[TBL] [Abstract][Full Text] [Related]
3. Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABA
Siebert DCB; Bampali K; Puthenkalam R; Varagic Z; Sarto-Jackson I; Scholze P; Sieghart W; Mihovilovic MD; Schnürch M; Ernst M
ACS Chem Biol; 2018 Aug; 13(8):2040-2047. PubMed ID: 29989390
[TBL] [Abstract][Full Text] [Related]
4. Structure-Guided Computational Methods Predict Multiple Distinct Binding Modes for Pyrazoloquinolinones in GABA
Fabjan J; Koniuszewski F; Schaar B; Ernst M
Front Neurosci; 2020; 14():611953. PubMed ID: 33519364
[TBL] [Abstract][Full Text] [Related]
5. Towards functional selectivity for α6β3γ2 GABA
Treven M; Siebert DCB; Holzinger R; Bampali K; Fabjan J; Varagic Z; Wimmer L; Steudle F; Scholze P; Schnürch M; Mihovilovic MD; Ernst M
Br J Pharmacol; 2018 Feb; 175(3):419-428. PubMed ID: 29127702
[TBL] [Abstract][Full Text] [Related]
6. Cerebellar α
Chiou LC; Lee HJ; Ernst M; Huang WJ; Chou JF; Chen HL; Mouri A; Chen LC; Treven M; Mamiya T; Fan PC; Knutson DE; Witzigmann C; Cook J; Sieghart W; Nabeshima T
Br J Pharmacol; 2018 Jun; 175(12):2414-2427. PubMed ID: 29518821
[TBL] [Abstract][Full Text] [Related]
7. GABA
Iorio MT; Vogel FD; Koniuszewski F; Scholze P; Rehman S; Simeone X; Schnürch M; Mihovilovic MD; Ernst M
Int J Mol Sci; 2020 Jan; 21(1):. PubMed ID: 31947863
[TBL] [Abstract][Full Text] [Related]
8. Variations on a scaffold - Novel GABA
Iorio MT; Rehman S; Bampali K; Stoeger B; Schnürch M; Ernst M; Mihovilovic MD
Eur J Med Chem; 2019 Oct; 180():340-349. PubMed ID: 31325782
[TBL] [Abstract][Full Text] [Related]
9. Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface.
Varagic Z; Wimmer L; Schnürch M; Mihovilovic MD; Huang S; Rallapalli S; Cook JM; Mirheydari P; Ecker GF; Sieghart W; Ernst M
Br J Pharmacol; 2013 May; 169(2):371-83. PubMed ID: 23472852
[TBL] [Abstract][Full Text] [Related]
10. Subtype selectivity of α+β- site ligands of GABAA receptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors.
Varagic Z; Ramerstorfer J; Huang S; Rallapalli S; Sarto-Jackson I; Cook J; Sieghart W; Ernst M
Br J Pharmacol; 2013 May; 169(2):384-99. PubMed ID: 23472935
[TBL] [Abstract][Full Text] [Related]
11. Alterations in the expression of GABAA receptor subunits in cerebellar granule cells after the disruption of the alpha6 subunit gene.
Nusser Z; Ahmad Z; Tretter V; Fuchs K; Wisden W; Sieghart W; Somogyi P
Eur J Neurosci; 1999 May; 11(5):1685-97. PubMed ID: 10215922
[TBL] [Abstract][Full Text] [Related]
12. SB-205384 is a positive allosteric modulator of recombinant GABAA receptors containing rat α3, α5, or α6 subunit subtypes coexpressed with β3 and γ2 subunits.
Heidelberg LS; Warren JW; Fisher JL
J Pharmacol Exp Ther; 2013 Oct; 347(1):235-41. PubMed ID: 23902941
[TBL] [Abstract][Full Text] [Related]
13. Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β- Site.
Mirheydari P; Ramerstorfer J; Varagic Z; Scholze P; Wimmer L; Mihovilovic MM; Sieghart W; Ernst M
Neurochem Res; 2014 Jun; 39(6):1057-1067. PubMed ID: 24072672
[TBL] [Abstract][Full Text] [Related]
14. GABA(A) receptor subunit alteration-dependent diazepam insensitivity in the cerebellum of phospholipase C-related inactive protein knockout mice.
Mizokami A; Tanaka H; Ishibashi H; Umebayashi H; Fukami K; Takenawa T; Nakayama KI; Yokoyama T; Nabekura J; Kanematsu T; Hirata M
J Neurochem; 2010 Jul; 114(1):302-10. PubMed ID: 20412381
[TBL] [Abstract][Full Text] [Related]
15. Alcohol selectivity of β3-containing GABAA receptors: evidence for a unique extracellular alcohol/imidazobenzodiazepine Ro15-4513 binding site at the α+β- subunit interface in αβ3δ GABAA receptors.
Wallner M; Hanchar HJ; Olsen RW
Neurochem Res; 2014 Jun; 39(6):1118-26. PubMed ID: 24500446
[TBL] [Abstract][Full Text] [Related]
16. Subunit composition and quantitative importance of hetero-oligomeric receptors: GABAA receptors containing alpha6 subunits.
Jechlinger M; Pelz R; Tretter V; Klausberger T; Sieghart W
J Neurosci; 1998 Apr; 18(7):2449-57. PubMed ID: 9502805
[TBL] [Abstract][Full Text] [Related]
17. The α6 subunit-containing GABA
Fan PC; Lai TH; Hor CC; Lee MT; Huang P; Sieghart W; Ernst M; Knutson DE; Cook J; Chiou LC
Neuropharmacology; 2018 Sep; 140():1-13. PubMed ID: 30016665
[TBL] [Abstract][Full Text] [Related]
18. Actions of two GABAA receptor benzodiazepine-site ligands that are mediated via non-γ2-dependent modulation.
Leppä E; Linden AM; Rabe H; Vekovischeva OY; Wulff P; Lüddens H; Wisden W; Korpi ER
Eur J Pharmacol; 2011 Sep; 666(1-3):111-21. PubMed ID: 21616065
[TBL] [Abstract][Full Text] [Related]
19. GABA
Belelli D; Hales TG; Lambert JJ; Luscher B; Olsen R; Peters JA; Rudolph U; Sieghart W
IUPHAR BPS Guide Pharm CITE; 2021 Sep; 2021(3):. PubMed ID: 35005623
[TBL] [Abstract][Full Text] [Related]
20. Probing the molecular basis for affinity/potency- and efficacy-based subtype-selectivity exhibited by benzodiazepine-site modulators at GABA
Söderhielm PC; Balle T; Bak-Nyhus S; Zhang M; Hansen KM; Ahring PK; Jensen AA
Biochem Pharmacol; 2018 Dec; 158():339-358. PubMed ID: 30121248
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]