These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

100 related articles for article (PubMed ID: 31207161)

  • 1. Fragment Growing to Design Optimized Inhibitors for Human Blood Group B Galactosyltransferase (GTB).
    Strecker C; Peters H; Hackl T; Peters T; Meyer B
    ChemMedChem; 2019 Jul; 14(14):1336-1342. PubMed ID: 31207161
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A new concept for glycosyltransferase inhibitors: nonionic mimics of the nucleotide donor of the human blood group B galactosyltransferase.
    Schaefer K; Albers J; Sindhuwinata N; Peters T; Meyer B
    Chembiochem; 2012 Feb; 13(3):443-50. PubMed ID: 22223604
    [TBL] [Abstract][Full Text] [Related]  

  • 3. A nonionic inhibitor with high specificity for the UDP-Gal donor binding site of human blood group B galactosyltransferase: design, synthesis, and characterization.
    Schaefer K; Sindhuwinata N; Hackl T; Kötzler MP; Niemeyer FC; Palcic MM; Peters T; Meyer B
    J Med Chem; 2013 Mar; 56(5):2150-4. PubMed ID: 23406460
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Optimization of 1,2,5-thiadiazole carbamates as potent and selective ABHD6 inhibitors.
    Patel JZ; Nevalainen TJ; Savinainen JR; Adams Y; Laitinen T; Runyon RS; Vaara M; Ahenkorah S; Kaczor AA; Navia-Paldanius D; Gynther M; Aaltonen N; Joharapurkar AA; Jain MR; Haka AS; Maxfield FR; Laitinen JT; Parkkari T
    ChemMedChem; 2015 Feb; 10(2):253-65. PubMed ID: 25504894
    [TBL] [Abstract][Full Text] [Related]  

  • 5. NMR-based exploration of the acceptor binding site of human blood group B galactosyltransferase with molecular fragments.
    Rademacher C; Landström J; Sindhuwinata N; Palcic MM; Widmalm G; Peters T
    Glycoconj J; 2010 Apr; 27(3):349-58. PubMed ID: 20217221
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Comparative study of substrate and product binding to the human ABO(H) blood group glycosyltransferases.
    Soya N; Shoemaker GK; Palcic MM; Klassen JS
    Glycobiology; 2009 Nov; 19(11):1224-34. PubMed ID: 19648353
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Blood group B galactosyltransferase: insights into substrate binding from NMR experiments.
    Angulo J; Langpap B; Blume A; Biet T; Meyer B; Krishna NR; Peters H; Palcic MM; Peters T
    J Am Chem Soc; 2006 Oct; 128(41):13529-38. PubMed ID: 17031966
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, in vitro urease inhibition and molecular docking studies of some novel quinazolin-4(3H)-one derivatives containing triazole, thiadiazole and thiosemicarbazide functionalities.
    Menteşe E; Akyüz G; Emirik M; Baltaş N
    Bioorg Chem; 2019 Mar; 83():289-296. PubMed ID: 30391701
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Molecular docking studies and biological evaluation of 1,3,4-thiadiazole derivatives bearing Schiff base moieties as tyrosinase inhibitors.
    Tang J; Liu J; Wu F
    Bioorg Chem; 2016 Dec; 69():29-36. PubMed ID: 27669118
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Solution structures of stromelysin complexed to thiadiazole inhibitors.
    Stockman BJ; Waldon DJ; Gates JA; Scahill TA; Kloosterman DA; Mizsak SA; Jacobsen EJ; Belonga KL; Mitchell MA; Mao B; Petke JD; Goodman L; Powers EA; Ledbetter SR; Kaytes PS; Vogeli G; Marshall VP; Petzold GL; Poorman RA
    Protein Sci; 1998 Nov; 7(11):2281-6. PubMed ID: 9827994
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists.
    van Muijlwijk-Koezen JE; Timmerman H; Vollinga RC; Frijtag von Drabbe Künzel J; de Groote M; Visser S; IJzerman AP
    J Med Chem; 2001 Mar; 44(5):749-62. PubMed ID: 11262085
    [TBL] [Abstract][Full Text] [Related]  

  • 12. High-resolution crystal structures and STD NMR mapping of human ABO(H) blood group glycosyltransferases in complex with trisaccharide reaction products suggest a molecular basis for product release.
    Gagnon SML; Legg MSG; Sindhuwinata N; Letts JA; Johal AR; Schuman B; Borisova SN; Palcic MM; Peters T; Evans SV
    Glycobiology; 2017 Oct; 27(10):966-977. PubMed ID: 28575295
    [TBL] [Abstract][Full Text] [Related]  

  • 13. The effect of heavy atoms on the conformation of the active-site polypeptide loop in human ABO(H) blood-group glycosyltransferase B.
    Letts JA; Persson M; Schuman B; Borisova SN; Palcic MM; Evans SV
    Acta Crystallogr D Biol Crystallogr; 2007 Aug; 63(Pt 8):860-5. PubMed ID: 17642512
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Benzo[c][1,2,5]thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors.
    Wang WL; Chen XY; Gao Y; Gao LX; Sheng L; Zhu J; Xu L; Ding ZZ; Zhang C; Li JY; Li J; Zhou YB
    Bioorg Med Chem Lett; 2017 Dec; 27(23):5154-5157. PubMed ID: 29100798
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Amino-acid substitution in the disordered loop of blood group B-glycosyltransferase enzyme causes weak B phenotype.
    Yazer MH; Denomme GA; Rose NL; Palcic MM
    Transfusion; 2005 Jul; 45(7):1178-82. PubMed ID: 15987364
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Thermodynamic signature of substrates and substrate analogs binding to human blood group B galactosyltransferase from isothermal titration calorimetry experiments.
    Sindhuwinata N; Grimm LL; Weißbach S; Zinn S; Munoz E; Palcic MM; Peters T
    Biopolymers; 2013 Oct; 99(10):784-95. PubMed ID: 23754468
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors.
    Talapatra SK; Tham CL; Guglielmi P; Cirilli R; Chandrasekaran B; Karpoormath R; Carradori S; Kozielski F
    Eur J Med Chem; 2018 Aug; 156():641-651. PubMed ID: 30031975
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Substrate Binding Drives Active-Site Closing of Human Blood Group B Galactosyltransferase as Revealed by Hot-Spot Labeling and NMR Spectroscopy Experiments.
    Weissbach S; Flügge F; Peters T
    Chembiochem; 2018 May; 19(9):970-978. PubMed ID: 29457687
    [TBL] [Abstract][Full Text] [Related]  

  • 19. [Synthesis and antibacterial activity of 3-(4-piperazin-1-yl-phenyl)-s-triazolo [3,4-b] [1,3,4] thiadiazole hydrochlorides].
    Hu GQ; Sun MF; Xie SQ; Huang WL; Zhang HB
    Yao Xue Xue Bao; 2007 Jan; 42(1):54-7. PubMed ID: 17520807
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, synthesis and antimicrobial activities of thiouracil derivatives containing triazolo-thiadiazole as SecA inhibitors.
    Cui P; Li X; Zhu M; Wang B; Liu J; Chen H
    Eur J Med Chem; 2017 Feb; 127():159-165. PubMed ID: 28039774
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.