BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

191 related articles for article (PubMed ID: 31525527)

  • 1. Design, synthesis and biological evaluation of theophylline containing variant acetylene derivatives as α-amylase inhibitors.
    Ruddarraju RR; Kiran G; Murugulla AC; Maroju R; Prasad DK; Kumar BH; Bakshi V; Reddy NS
    Bioorg Chem; 2019 Nov; 92():103120. PubMed ID: 31525527
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis, antidiabetic activity and molecular docking study of rhodanine-substitued spirooxindole pyrrolidine derivatives as novel α-amylase inhibitors.
    Toumi A; Boudriga S; Hamden K; Sobeh M; Cheurfa M; Askri M; Knorr M; Strohmann C; Brieger L
    Bioorg Chem; 2021 Jan; 106():104507. PubMed ID: 33288322
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Discovery of novel 6-(piperidin-1-ylsulfonyl)-2H-chromenes targeting α-glucosidase, α-amylase, and PPAR-γ: Design, synthesis, virtual screening, and anti-diabetic activity for type 2 diabetes mellitus.
    Thabet HK; Abusaif MS; Imran M; Helal MH; Alaqel SI; Alshehri A; Mohd AA; Ammar YA; Ragab A
    Comput Biol Chem; 2024 Aug; 111():108097. PubMed ID: 38772048
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 2-Aryl benzimidazoles: Synthesis, In vitro α-amylase inhibitory activity, and molecular docking study.
    Adegboye AA; Khan KM; Salar U; Aboaba SA; Kanwal ; Chigurupati S; Fatima I; Taha M; Wadood A; Mohammad JI; Khan H; Perveen S
    Eur J Med Chem; 2018 Apr; 150():248-260. PubMed ID: 29533872
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and in vitro evaluation of chlorogenic acid amides as potential hypoglycemic agents and their synergistic effect with acarbose.
    Cardullo N; Floresta G; Rescifina A; Muccilli V; Tringali C
    Bioorg Chem; 2021 Dec; 117():105458. PubMed ID: 34736132
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of alpha amylase inhibitors based on privileged indole scaffold.
    Noreen T; Taha M; Imran S; Chigurupati S; Rahim F; Selvaraj M; Ismail NH; Mohammad JI; Ullah H; Javid MT; Nawaz F; Irshad M; Ali M
    Bioorg Chem; 2017 Jun; 72():248-255. PubMed ID: 28482265
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Fluorinated indeno-quinoxaline bearing thiazole moieties as hypoglycaemic agents targeting
    Gohar NA; Fayed EA; A Ammar Y; A Abu Ali O; Ragab A; Mahfoz AM; Abusaif MS
    J Enzyme Inhib Med Chem; 2024 Dec; 39(1):2367128. PubMed ID: 38913598
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, α-amylase inhibitory potential and molecular docking study of indole derivatives.
    Taha M; Baharudin MS; Ismail NH; Imran S; Khan MN; Rahim F; Selvaraj M; Chigurupati S; Nawaz M; Qureshi F; Vijayabalan S
    Bioorg Chem; 2018 Oct; 80():36-42. PubMed ID: 29864686
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Exploring the Dual Inhibitory Activity of Novel Anthranilic Acid Derivatives towards α-Glucosidase and Glycogen Phosphorylase Antidiabetic Targets: Design, In Vitro Enzyme Assay, and Docking Studies.
    Ihmaid S
    Molecules; 2018 May; 23(6):. PubMed ID: 29844263
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis of novel 5-(2,5-bis(2,2,2-trifluoroethoxy)phenyl)-1,3,4-oxadiazole-2-thiol derivatives as potential glucosidase inhibitors.
    Gani RS; Kudva AK; Timanagouda K; Raghuveer ; Mujawar SBH; Joshi SD; Raghu SV
    Bioorg Chem; 2021 Sep; 114():105046. PubMed ID: 34126575
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Evaluation and docking of indole sulfonamide as a potent inhibitor of α-glucosidase enzyme in streptozotocin -induced diabetic albino wistar rats.
    Taha M; Imran S; Salahuddin M; Iqbal N; Rahim F; Uddin N; Shehzad A; Khalid Farooq R; Alomari M; Mohammed Khan K
    Bioorg Chem; 2021 May; 110():104808. PubMed ID: 33756236
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Taxifolin prevents postprandial hyperglycemia by regulating the activity of α-amylase: Evidence from an in vivo and in silico studies.
    Rehman K; Chohan TA; Waheed I; Gilani Z; Akash MSH
    J Cell Biochem; 2019 Jan; 120(1):425-438. PubMed ID: 30191607
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of piperazine sulfonamide analogs as diabetic-II inhibitors and their molecular docking study.
    Taha M; Irshad M; Imran S; Chigurupati S; Selvaraj M; Rahim F; Ismail NH; Nawaz F; Khan KM
    Eur J Med Chem; 2017 Dec; 141():530-537. PubMed ID: 29102178
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Novel enantiopure isoxazolidine and C-alkyl imine oxide derivatives as potential hypoglycemic agents: Design, synthesis, dual inhibitors of α-amylase and α-glucosidase, ADMET and molecular docking study.
    Ghannay S; Snoussi M; Messaoudi S; Kadri A; Aouadi K
    Bioorg Chem; 2020 Nov; 104():104270. PubMed ID: 32947132
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and biological evaluation of 3-arylcoumarin derivatives as potential anti-diabetic agents.
    Hu Y; Wang B; Yang J; Liu T; Sun J; Wang X
    J Enzyme Inhib Med Chem; 2019 Dec; 34(1):15-30. PubMed ID: 30362362
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Spiroindolone Analogues as Potential Hypoglycemic with Dual Inhibitory Activity on α-Amylase and α-Glucosidase.
    Altowyan MS; Barakat A; Al-Majid AM; Al-Ghulikah HA
    Molecules; 2019 Jun; 24(12):. PubMed ID: 31242688
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Dihydropyridines as potential α-amylase and α-glucosidase inhibitors: Synthesis, in vitro and in silico studies.
    Yousuf H; Shamim S; Khan KM; Chigurupati S; Kanwal ; Hameed S; Khan MN; Taha M; Arfeen M
    Bioorg Chem; 2020 Mar; 96():103581. PubMed ID: 31978686
    [TBL] [Abstract][Full Text] [Related]  

  • 18. In vitro and in vivo α-amylase and α-glucosidase inhibiting activities of the protein extracts from two varieties of bitter gourd (Momordica charantia L.).
    Poovitha S; Parani M
    BMC Complement Altern Med; 2016 Jul; 16 Suppl 1(Suppl 1):185. PubMed ID: 27454418
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis of new indazole based dual inhibitors of α-glucosidase and α-amylase enzymes, their in vitro, in silico and kinetics studies.
    Rafique R; Khan KM; Arshia ; Kanwal ; Chigurupati S; Wadood A; Rehman AU; Karunanidhi A; Hameed S; Taha M; Al-Rashida M
    Bioorg Chem; 2020 Jan; 94():103195. PubMed ID: 31451297
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design and synthesis of epigallocatechin (EGC) analogs selective to inhibit α-amylase over α-glucosidases via the incorporation of caffeine acid and its derivatives.
    Chen W; Zhou C; Chen J; Wang M; Zhou F; Wang C; Zhang X; Zhou W
    Bioorg Chem; 2022 Feb; 119():105515. PubMed ID: 34896919
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.