155 related articles for article (PubMed ID: 31569409)
1. Synthesis and Biological Evaluation of New Glycoconjugated LDH Inhibitors as Anticancer Agents.
D'Andrea F; Vagelli G; Granchi C; Guazzelli L; Tuccinardi T; Poli G; Iacopini D; Minutolo F; Di Bussolo V
Molecules; 2019 Sep; 24(19):. PubMed ID: 31569409
[TBL] [Abstract][Full Text] [Related]
2. Assessing the differential action on cancer cells of LDH-A inhibitors based on the N-hydroxyindole-2-carboxylate (NHI) and malonic (Mal) scaffolds.
Granchi C; Calvaresi EC; Tuccinardi T; Paterni I; Macchia M; Martinelli A; Hergenrother PJ; Minutolo F
Org Biomol Chem; 2013 Oct; 11(38):6588-96. PubMed ID: 23986182
[TBL] [Abstract][Full Text] [Related]
3. Dual targeting of the Warburg effect with a glucose-conjugated lactate dehydrogenase inhibitor.
Calvaresi EC; Granchi C; Tuccinardi T; Di Bussolo V; Huigens RW; Lee HY; Palchaudhuri R; Macchia M; Martinelli A; Minutolo F; Hergenrother PJ
Chembiochem; 2013 Nov; 14(17):2263-7. PubMed ID: 24174263
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis and biological evaluation of colchicine glycoconjugates as tubulin polymerization inhibitors.
Wang Z; Liu R; Zhang X; Chang X; Gao M; Zhang S; Guan Q; Sun J; Zuo D; Zhang W
Bioorg Med Chem; 2022 Mar; 58():116671. PubMed ID: 35193066
[TBL] [Abstract][Full Text] [Related]
5. Glycoconjugation of Betulin Derivatives Using Copper-Catalyzed 1,3-Dipolar Azido-Alkyne Cycloaddition Reaction and a Preliminary Assay of Cytotoxicity of the Obtained Compounds.
Grymel M; Pastuch-Gawołek G; Lalik A; Zawojak M; Boczek S; Krawczyk M; Erfurt K
Molecules; 2020 Dec; 25(24):. PubMed ID: 33353244
[TBL] [Abstract][Full Text] [Related]
6. First Examples of H
Fortunato S; Lenzi C; Granchi C; Citi V; Martelli A; Calderone V; Di Pietro S; Signore G; Di Bussolo V; Minutolo F
Bioconjug Chem; 2019 Mar; 30(3):614-620. PubMed ID: 30609890
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and Preliminary Evaluation of the Cytotoxicity of Potential Metabolites of Quinoline Glycoconjugates.
Domińska M; Pastuch-Gawołek G; Domiński A; Kurcok P; Erfurt K
Molecules; 2022 Feb; 27(3):. PubMed ID: 35164304
[TBL] [Abstract][Full Text] [Related]
8. Evaluation on the inhibition of pyrrol-2-yl ethanone derivatives to lactate dehydrogenase and anticancer activities.
Lu NN; Weng ZY; Chen QY; Boison D; Xiao XX; Gao J
Spectrochim Acta A Mol Biomol Spectrosc; 2016 Aug; 165():21-25. PubMed ID: 27104676
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of 1,2,3-triazole glycoconjugates as inhibitors of α-glucosidases.
da Rocha DR; Santos WC; Lima ES; Ferreira VF
Carbohydr Res; 2012 Mar; 350():14-9. PubMed ID: 22269981
[TBL] [Abstract][Full Text] [Related]
10. N-Hydroxyindole-based inhibitors of lactate dehydrogenase against cancer cell proliferation.
Granchi C; Roy S; De Simone A; Salvetti I; Tuccinardi T; Martinelli A; Macchia M; Lanza M; Betti L; Giannaccini G; Lucacchini A; Giovannetti E; Sciarrillo R; Peters GJ; Minutolo F
Eur J Med Chem; 2011 Nov; 46(11):5398-407. PubMed ID: 21944286
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and Preliminary Evaluation of Biological Activity of Glycoconjugates Analogues of Acyclic Uridine Derivatives.
Komor R; Pastuch-Gawolek G; Krol E; Szeja W
Molecules; 2018 Aug; 23(8):. PubMed ID: 30104510
[TBL] [Abstract][Full Text] [Related]
12. Amphiphilic glycoconjugates as potential anti-cancer chemotherapeutics.
Govindarajan M
Eur J Med Chem; 2018 Jan; 143():1208-1253. PubMed ID: 29126728
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and biological evaluation of a new class of glycoconjugated disulfides that exhibit potential anticancer properties.
Bonaccorsi P; Marino-Merlo F; Barattucci A; Battaglia G; Papaianni E; Papalia T; Aversa MC; Mastino A
Bioorg Med Chem; 2012 May; 20(10):3186-95. PubMed ID: 22537679
[TBL] [Abstract][Full Text] [Related]
14. Design, synthesis and anti-tumor evaluation of novel steroidal glycoconjugate with furoxan derivatives.
Li H; Wang K; Wan Q; Chen Y
Steroids; 2019 Jan; 141():81-95. PubMed ID: 30521816
[TBL] [Abstract][Full Text] [Related]
15. Design, Synthesis, biological investigations and molecular interactions of triazole linked tacrine glycoconjugates as Acetylcholinesterase inhibitors with reduced hepatotoxicity.
Kaur Gulati H; Choudhary S; Kumar N; Ahmed A; Bhagat K; Vir Singh J; Singh A; Kumar A; Singh Bedi PM; Singh H; Mukherjee D
Bioorg Chem; 2022 Jan; 118():105479. PubMed ID: 34801945
[TBL] [Abstract][Full Text] [Related]
16. Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors.
Rupiani S; Buonfiglio R; Manerba M; Di Ianni L; Vettraino M; Giacomini E; Masetti M; Falchi F; Di Stefano G; Roberti M; Recanatini M
Eur J Med Chem; 2015 Aug; 101():63-70. PubMed ID: 26114812
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and antiproliferative activity of a natural like glycoconjugate polycyclic compound.
Maggio B; Raimondi MV; Raffa D; Plescia F; Scherrmann MC; Prosa N; Lauricella M; D'Anneo A; Daidone G
Eur J Med Chem; 2016 Oct; 122():247-256. PubMed ID: 27372287
[TBL] [Abstract][Full Text] [Related]
18. New insights into structure-activity relationship of ipomoeassin F from its bioisosteric 5-oxa/aza analogues.
Zong G; Sun X; Bhakta R; Whisenhunt L; Hu Z; Wang F; Shi WQ
Eur J Med Chem; 2018 Jan; 144():751-757. PubMed ID: 29291442
[TBL] [Abstract][Full Text] [Related]
19. Synthesis of artemisinic acid derived glycoconjugates and their anticancer studies.
Kotammagari TK; Paul S; Barik GK; Santra MK; Bhattacharya AK
Org Biomol Chem; 2020 Mar; 18(12):2252-2263. PubMed ID: 32149317
[TBL] [Abstract][Full Text] [Related]
20. Discovery of N-hydroxyindole-based inhibitors of human lactate dehydrogenase isoform A (LDH-A) as starvation agents against cancer cells.
Granchi C; Roy S; Giacomelli C; Macchia M; Tuccinardi T; Martinelli A; Lanza M; Betti L; Giannaccini G; Lucacchini A; Funel N; León LG; Giovannetti E; Peters GJ; Palchaudhuri R; Calvaresi EC; Hergenrother PJ; Minutolo F
J Med Chem; 2011 Mar; 54(6):1599-612. PubMed ID: 21332213
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]