BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

142 related articles for article (PubMed ID: 3172131)

  • 1. Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands.
    Glennon RA; Naiman NA; Lyon RA; Titeler M
    J Med Chem; 1988 Oct; 31(10):1968-71. PubMed ID: 3172131
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Analogues of the 5-HT1A serotonin antagonist 1-(2-methoxyphenyl)-4-[4-(2-phthalimido)butyl]piperazine with reduced alpha 1-adrenergic affinity.
    Raghupathi RK; Rydelek-Fitzgerald L; Teitler M; Glennon RA
    J Med Chem; 1991 Aug; 34(8):2633-8. PubMed ID: 1652026
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New sigma and 5-HT1A receptor ligands: omega-(tetralin-1-yl)-n-alkylamine derivatives.
    Berardi F; Colabufo NA; Giudice G; Perrone R; Tortorella V; Govoni S; Lucchi L
    J Med Chem; 1996 Jan; 39(1):176-82. PubMed ID: 8568804
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 5-HT1A-versus D2-receptor selectivity of flesinoxan and analogous N4-substituted N1-arylpiperazines.
    Kuipers W; Kruse CG; van Wijngaarden I; Standaar PJ; Tulp MT; Veldman N; Spek AL; IJzerman AP
    J Med Chem; 1997 Jan; 40(3):300-12. PubMed ID: 9022796
    [TBL] [Abstract][Full Text] [Related]  

  • 5. N4-unsubstituted N1-arylpiperazines as high-affinity 5-HT1A receptor ligands.
    Kuipers W; van Wijngaarden I; Kruse CG; ter Horst-van Amstel M; Tulp MT; IJzerman AP
    J Med Chem; 1995 May; 38(11):1942-54. PubMed ID: 7783126
    [TBL] [Abstract][Full Text] [Related]  

  • 6. [3H]1-[2-(4-aminophenyl)ethyl]-4-(3-trifluoromethylphenyl)piperazine: a selective radioligand for 5-HT1A receptors in rat brain.
    Ransom RW; Asarch KB; Shih JC
    J Neurochem; 1986 Jan; 46(1):68-75. PubMed ID: 2933490
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Polycyclic aryl- and heteroarylpiperazinyl imides as 5-HT1A receptor ligands and potential anxiolytic agents: synthesis and structure-activity relationship studies.
    Abou-Gharbia M; Patel UR; Webb MB; Moyer JA; Andree TH; Muth EA
    J Med Chem; 1988 Jul; 31(7):1382-92. PubMed ID: 2898533
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Isoindol-1-one analogues of 4-(2'-methoxyphenyl)-1-[2'-[N-(2"-pyridyl)-p-iodobenzamido]ethyl]pipera zine (p-MPPI) as 5-HT1A receptor ligands.
    Zhuang ZP; Kung MP; Mu M; Kung HF
    J Med Chem; 1998 Jan; 41(2):157-66. PubMed ID: 9457239
    [TBL] [Abstract][Full Text] [Related]  

  • 9. High potent and selective arylpiperazine derivatives as ligands for the 5-HT1A receptor.
    Modica M; Santagati M; Santagati A; Russo F; Cagnotto A; Goegan M; Mennini T
    Bioorg Med Chem Lett; 2000 May; 10(10):1089-92. PubMed ID: 10843224
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Structure-affinity relationship studies on 5-HT1A receptor ligands. 1. Heterobicyclic phenylpiperazines with N4-alkyl substituents.
    van Steen BJ; van Wijngaarden I; Tulp MT; Soudijn W
    J Med Chem; 1993 Sep; 36(19):2751-60. PubMed ID: 8410989
    [TBL] [Abstract][Full Text] [Related]  

  • 11. New (2-methoxyphenyl)piperazine derivatives as 5-HT1A receptor ligands with reduced alpha 1-adrenergic activity. Synthesis and structure-affinity relationships.
    Orjales A; Alonso-Cires L; Labeaga L; Corcóstegui R
    J Med Chem; 1995 Apr; 38(8):1273-7. PubMed ID: 7731013
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Structure-activity relationship studies of CNS agents. Part 10(1): 1-Aryl-2-[3-(4-aryl-1-piperazinyl)propyl]-1,4-dihydro-3(2H)-isoquino linones: two modes of the interaction with the 5-HT1A receptor site.
    Mokrosz JL; Bojarski AJ; Maćkowiak M; Bielecka Z; Boksa J
    Pharmazie; 1994 May; 49(5):328-33. PubMed ID: 8016178
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Derivatives of 4-(2'-methoxyphenyl)-1-[2'-(N-2"-pyridinyl-p-iodobenzamido)ethyl]pipera zine (p-MPPI) as 5-HT1A ligands.
    Zhuang ZP; Kung MP; Chumpradit S; Mu M; Kung HF
    J Med Chem; 1994 Dec; 37(26):4572-5. PubMed ID: 7799409
    [TBL] [Abstract][Full Text] [Related]  

  • 14. High affinity and selectivity on 5-HT1A receptor of 1-aryl-4-[1-tetralin)alkyl]piperazines. 2.
    Perrone R; Berardi F; Colabufo NA; Leopoldo M; Tortorella V; Fiorentini F; Olgiati V; Ghiglieri A; Govoni S
    J Med Chem; 1995 Mar; 38(6):942-9. PubMed ID: 7699710
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Binding of arylpiperazines to 5-HT3 serotonin receptors: results of a structure-affinity study.
    Glennon RA; Ismaiel AE; McCarthy BG; Peroutka SJ
    Eur J Pharmacol; 1989 Sep; 168(3):387-92. PubMed ID: 2583244
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Structure-affinity relationship studies on D-2/5-HT1A receptor ligands. 4-(2-Heteroarylethyl)-1-arylpiperazines.
    Dukić S; Vujović M; Soskić V; Joksimović J
    Arzneimittelforschung; 1997 Mar; 47(3):239-43. PubMed ID: 9105540
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 1-Aryl-4-(4-succinimidobutyl)piperazines and their conformationally constrained analogues: synthesis, binding to serotonin (5-HT1A, 5-HT2A, 5-HT7), alpha1-adrenergic, and dopaminergic D2 receptors, and in vivo 5-HT1A functional characteristics.
    Bojarski AJ; Paluchowska MH; Duszyńska B; Kłodzińska A; Tatarczyńska E; Chojnacka-Wójcik E
    Bioorg Med Chem; 2005 Mar; 13(6):2293-303. PubMed ID: 15727878
    [TBL] [Abstract][Full Text] [Related]  

  • 18. [[(Arylpiperazinyl)alkyl]thio]thieno[2,3-d]pyrimidinone derivatives as high-affinity, selective 5-HT1A receptor ligands.
    Modica M; Santagati M; Russo F; Parotti L; De Gioia L; Selvaggini C; Salmona M; Mennini T
    J Med Chem; 1997 Feb; 40(4):574-85. PubMed ID: 9046348
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure-activity relationship studies of CNS agents. Part III. On the bioactive conformations of 1-arylpiperazines at 5-HT1A receptor.
    Mokrosz JL; Duszyńska B; Bojarski A
    Pol J Pharmacol Pharm; 1992; 44(1):87-97. PubMed ID: 1359516
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 1-Substituted-4-[3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl]piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alpha1 receptors. Part 6.
    Perrone R; Berardi F; Colabufo NA; Leopoldo M; Tortorella V
    Bioorg Med Chem; 2000 May; 8(5):873-81. PubMed ID: 10881999
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.