161 related articles for article (PubMed ID: 31757526)
1. Synthesis of novel 3-halo-3-nitroflavanones and their activities as DNA methyltransferase inhibitors in cancer cells.
Pechalrieu D; Dauzonne D; Arimondo PB; Lopez M
Eur J Med Chem; 2020 Jan; 186():111829. PubMed ID: 31757526
[TBL] [Abstract][Full Text] [Related]
2. Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A.
Erdmann A; Menon Y; Gros C; Masson V; Aussagues Y; Ausseil F; Novosad N; Schambel P; Baltas M; Arimondo PB
Future Med Chem; 2016; 8(4):373-80. PubMed ID: 26976348
[TBL] [Abstract][Full Text] [Related]
3. Rapid synthesis of new DNMT inhibitors derivatives of procainamide.
Halby L; Champion C; Sénamaud-Beaufort C; Ajjan S; Drujon T; Rajavelu A; Ceccaldi A; Jurkowska R; Lequin O; Nelson WG; Guy A; Jeltsch A; Guianvarc'h D; Ferroud C; Arimondo PB
Chembiochem; 2012 Jan; 13(1):157-65. PubMed ID: 22170584
[TBL] [Abstract][Full Text] [Related]
4. Novel anticancer drug curaxin CBL0137 impairs DNA methylation by eukaryotic DNA methyltransferase Dnmt3a.
Sergeev A; Vorobyov A; Yakubovskaya M; Kirsanova O; Gromova E
Bioorg Med Chem Lett; 2020 Aug; 30(16):127296. PubMed ID: 32631516
[TBL] [Abstract][Full Text] [Related]
5. Development of a versatile DNMT and HDAC inhibitor C02S modulating multiple cancer hallmarks for breast cancer therapy.
Yuan Z; Chen S; Gao C; Dai Q; Zhang C; Sun Q; Lin JS; Guo C; Chen Y; Jiang Y
Bioorg Chem; 2019 Jun; 87():200-208. PubMed ID: 30901675
[TBL] [Abstract][Full Text] [Related]
6. Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation.
Rilova E; Erdmann A; Gros C; Masson V; Aussagues Y; Poughon-Cassabois V; Rajavelu A; Jeltsch A; Menon Y; Novosad N; Gregoire JM; Vispé S; Schambel P; Ausseil F; Sautel F; Arimondo PB; Cantagrel F
ChemMedChem; 2014 Mar; 9(3):590-601. PubMed ID: 24678024
[TBL] [Abstract][Full Text] [Related]
7. Effect of Withaferin-A, Withanone, and Caffeic Acid Phenethyl Ester on DNA Methyltransferases: Potential in Epigenetic Cancer Therapy.
Kumar V; Dhanjal JK; Sari AN; Khurana M; Kaul SC; Wadhwa R; Sundar D
Curr Top Med Chem; 2024; 24(4):379-391. PubMed ID: 37496252
[TBL] [Abstract][Full Text] [Related]
8. Design and synthesis of N-benzoyl amino acid derivatives as DNA methylation inhibitors.
Garella D; Atlante S; Borretto E; Cocco M; Giorgis M; Costale A; Stevanato L; Miglio G; Cencioni C; Fernández-de Gortari E; Medina-Franco JL; Spallotta F; Gaetano C; Bertinaria M
Chem Biol Drug Des; 2016 Nov; 88(5):664-676. PubMed ID: 27225604
[TBL] [Abstract][Full Text] [Related]
9. 5-Nitro-Thiophene-Thiosemicarbazone Derivatives Present Antitumor Activity Mediated by Apoptosis and DNA Intercalation.
Roque Marques KM; do Desterro MR; de Arruda SM; de Araújo Neto LN; do Carmo Alves de Lima M; de Almeida SMV; da Silva ECD; de Aquino TM; da Silva-Júnior EF; de Araújo-Júnior JX; de M Silva M; de A Dantas MD; Santos JCC; Figueiredo IM; Bazin MA; Marchand P; da Silva TG; Mendonça Junior FJB
Curr Top Med Chem; 2019; 19(13):1075-1091. PubMed ID: 31223089
[TBL] [Abstract][Full Text] [Related]
10. Identification of novel inhibitors of DNA methylation by screening of a chemical library.
Ceccaldi A; Rajavelu A; Ragozin S; Sénamaud-Beaufort C; Bashtrykov P; Testa N; Dali-Ali H; Maulay-Bailly C; Amand S; Guianvarc'h D; Jeltsch A; Arimondo PB
ACS Chem Biol; 2013 Mar; 8(3):543-8. PubMed ID: 23294304
[TBL] [Abstract][Full Text] [Related]
11. Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells.
Zwergel C; Schnekenburger M; Sarno F; Battistelli C; Manara MC; Stazi G; Mazzone R; Fioravanti R; Gros C; Ausseil F; Florean C; Nebbioso A; Strippoli R; Ushijima T; Scotlandi K; Tripodi M; Arimondo PB; Altucci L; Diederich M; Mai A; Valente S
Clin Epigenetics; 2019 May; 11(1):68. PubMed ID: 31060628
[TBL] [Abstract][Full Text] [Related]
12. Anticancer drug discovery targeting DNA hypermethylation.
Yu N; Wang M
Curr Med Chem; 2008; 15(14):1350-75. PubMed ID: 18537614
[TBL] [Abstract][Full Text] [Related]
13. Molecular modeling and virtual screening of DNA methyltransferase inhibitors.
Medina-Franco JL; Yoo J
Curr Pharm Des; 2013; 19(12):2138-47. PubMed ID: 23016844
[TBL] [Abstract][Full Text] [Related]
14. Development of DNA methyltransferase inhibitors for the treatment of neoplastic diseases.
Fandy TE
Curr Med Chem; 2009; 16(17):2075-85. PubMed ID: 19519382
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis and anticancer potential of NSC-319745 hydroxamic acid derivatives as DNMT and HDAC inhibitors.
Yuan Z; Sun Q; Li D; Miao S; Chen S; Song L; Gao C; Chen Y; Tan C; Jiang Y
Eur J Med Chem; 2017 Jul; 134():281-292. PubMed ID: 28419930
[TBL] [Abstract][Full Text] [Related]
16. DNA Methyltransferase 3A: A Significant Target for the Discovery of Inhibitors as Potent Anticancer Drugs.
Feng Q; Duan H; Zhou X; Wang Y; Zhang J; Zhang H; Chen G; Bao X
Mini Rev Med Chem; 2024; 24(5):507-520. PubMed ID: 37642180
[TBL] [Abstract][Full Text] [Related]
17. Identifying novel selective non-nucleoside DNA methyltransferase 1 inhibitors through docking-based virtual screening.
Chen S; Wang Y; Zhou W; Li S; Peng J; Shi Z; Hu J; Liu YC; Ding H; Lin Y; Li L; Cheng S; Liu J; Lu T; Jiang H; Liu B; Zheng M; Luo C
J Med Chem; 2014 Nov; 57(21):9028-41. PubMed ID: 25333769
[TBL] [Abstract][Full Text] [Related]
18. Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1.
Castellano S; Kuck D; Sala M; Novellino E; Lyko F; Sbardella G
J Med Chem; 2008 Apr; 51(7):2321-5. PubMed ID: 18345608
[TBL] [Abstract][Full Text] [Related]
19. Discovery of novel DNA methyltransferase 3A inhibitors via structure-based virtual screening and biological assays.
Shao Z; Xu P; Xu W; Li L; Liu S; Zhang R; Liu YC; Zhang C; Chen S; Luo C
Bioorg Med Chem Lett; 2017 Jan; 27(2):342-346. PubMed ID: 27899265
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and biological activity of selenopsammaplin A and its analogues as antitumor agents with DOT1L inhibitory activity.
Ju Han H; Sub Byun W; Ho Lee G; Kyung Kim W; Jang K; Yang S; Yang J; Woo Ha M; Hong S; Lee J; Shin J; Bong Oh K; Kook Lee S; Park HG
Bioorg Med Chem; 2021 Apr; 35():116072. PubMed ID: 33636429
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
