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2. Ligand-induced activation of human TRPM2 requires the terminal ribose of ADPR and involves Arg1433 and Tyr1349. Fliegert R; Watt JM; Schöbel A; Rozewitz MD; Moreau C; Kirchberger T; Thomas MP; Sick W; Araujo AC; Harneit A; Potter BVL; Guse AH Biochem J; 2017 Jun; 474(13):2159-2175. PubMed ID: 28515263 [TBL] [Abstract][Full Text] [Related]
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8. Divalent copper is a potent extracellular blocker for TRPM2 channel. Zeng B; Chen GL; Xu SZ Biochem Biophys Res Commun; 2012 Jul; 424(2):279-84. PubMed ID: 22750002 [TBL] [Abstract][Full Text] [Related]
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11. Design, synthesis and biological activities of 2,3-dihydroquinazolin-4(1H)-one derivatives as TRPM2 inhibitors. Zhang H; Liu H; Luo X; Wang Y; Liu Y; Jin H; Liu Z; Yang W; Yu P; Zhang L; Zhang L Eur J Med Chem; 2018 May; 152():235-252. PubMed ID: 29723786 [TBL] [Abstract][Full Text] [Related]
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13. Regulation of TRPM2 by extra- and intracellular calcium. Starkus J; Beck A; Fleig A; Penner R J Gen Physiol; 2007 Oct; 130(4):427-40. PubMed ID: 17893195 [TBL] [Abstract][Full Text] [Related]
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