BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

128 related articles for article (PubMed ID: 31918397)

  • 21. Synthesis and Biological Evaluation of N-Aryl-5-aryloxazol-2-amine Derivatives as 5-Lipoxygenase Inhibitors.
    Suh JH; Yum EK; Cho YS
    Chem Pharm Bull (Tokyo); 2015; 63(8):573-8. PubMed ID: 26040270
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Design, synthesis and identification of novel substituted 2-amino thiazole analogues as potential anti-inflammatory agents targeting 5-lipoxygenase.
    Sinha S; Doble M; Manju SL
    Eur J Med Chem; 2018 Oct; 158():34-50. PubMed ID: 30199704
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Synthesis and evaluation of a new series of 3,5-bis((5-bromo-6-methyl-2-t-aminopyrimidin-4-yl)thio)-4H-1,2,4-triazol-4-amines and their cyclized products 'pyrimidinylthio pyrimidotriazolothiadiazines' as 15- lipo-oxygenase inhibitors.
    Asghari T; Bakavoli M; Rahimizadeh M; Eshghi H; Saberi S; Karimian A; Hadizadeh F; Ghandadi M
    Chem Biol Drug Des; 2015 Feb; 85(2):216-24. PubMed ID: 24925519
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Design and synthesis of pyrimido[4,5-b][1,4]benzothiazine derivatives, as potent 15-lipoxygenase inhibitors.
    Bakavoli M; Nikpour M; Rahimizadeh M; Saberi MR; Sadeghian H
    Bioorg Med Chem; 2007 Mar; 15(5):2120-6. PubMed ID: 17210254
    [TBL] [Abstract][Full Text] [Related]  

  • 25. A class of 5-benzylidene-2-phenylthiazolinones with high potency as direct 5-lipoxygenase inhibitors.
    Hofmann B; Barzen S; Rödl CB; Kiehl A; Borig J; Zivković A; Stark H; Schneider G; Steinhilber D
    J Med Chem; 2011 Mar; 54(6):1943-7. PubMed ID: 21341744
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Synthesis and biological evaluation of isoxazolo[4,5-d]pyridazin-4-(5H)-one analogues as potent anti-inflammatory agents.
    Özadalı K; Özkanlı F; Jain S; Rao PP; Velázquez-Martínez CA
    Bioorg Med Chem; 2012 May; 20(9):2912-22. PubMed ID: 22475926
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Discovery of a benzenesulfonamide-based dual inhibitor of microsomal prostaglandin E
    Cheung SY; Werner M; Esposito L; Troisi F; Cantone V; Liening S; König S; Gerstmeier J; Koeberle A; Bilancia R; Rizza R; Rossi A; Roviezzo F; Temml V; Schuster D; Stuppner H; Schubert-Zsilavecz M; Werz O; Hanke T; Pace S
    Eur J Med Chem; 2018 Aug; 156():815-830. PubMed ID: 30053720
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Chloro-substituted pyridine squaramates as new DNase I inhibitors: Synthesis, structural characterization, in vitro evaluation and molecular docking studies.
    Ruseva N; Atanasova M; Sbirkova-Dimitrova H; Marković A; Šmelcerović Ž; Šmelcerović A; Cherneva E; Bakalova A
    Chem Biol Interact; 2023 Dec; 386():110772. PubMed ID: 37898285
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Coumarin-thiazole and -oxadiazole derivatives: Synthesis, bioactivity and docking studies for aldose/aldehyde reductase inhibitors.
    Ibrar A; Tehseen Y; Khan I; Hameed A; Saeed A; Furtmann N; Bajorath J; Iqbal J
    Bioorg Chem; 2016 Oct; 68():177-86. PubMed ID: 27544072
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Further insight into the dual COX-2 and 15-LOX anti-inflammatory activity of 1,3,4-thiadiazole-thiazolidinone hybrids: The contribution of the substituents at 5th positions is size dependent.
    Omar YM; Abdel-Moty SG; Abdu-Allah HHM
    Bioorg Chem; 2020 Apr; 97():103657. PubMed ID: 32086052
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Rutin as Deoxyribonuclease I Inhibitor.
    Kolarevic A; Pavlovic A; Djordjevic A; Lazarevic J; Savic S; Kocic G; Anderluh M; Smelcerovic A
    Chem Biodivers; 2019 May; 16(5):e1900069. PubMed ID: 30883015
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase.
    Filosa R; Peduto A; Aparoy P; Schaible AM; Luderer S; Krauth V; Petronzi C; Massa A; de Rosa M; Reddanna P; Werz O
    Eur J Med Chem; 2013 Sep; 67():269-79. PubMed ID: 23871907
    [TBL] [Abstract][Full Text] [Related]  

  • 33. Imidazo[2,1-b]thiazole derivatives as new inhibitors of 15-lipoxygenase.
    Tehrani MB; Emami S; Asadi M; Saeedi M; Mirzahekmati M; Ebrahimi SM; Mahdavi M; Nadri H; Moradi A; Moghadam FH; Farzipour S; Vosooghi M; Foroumadi A; Shafiee A
    Eur J Med Chem; 2014 Nov; 87():759-64. PubMed ID: 25310714
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Syntheses and evaluation of novel isoliquiritigenin derivatives as potential dual inhibitors for amyloid-beta aggregation and 5-lipoxygenase.
    Chen YP; Zhang ZY; Li YP; Li D; Huang SL; Gu LQ; Xu J; Huang ZS
    Eur J Med Chem; 2013 Aug; 66():22-31. PubMed ID: 23786711
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Xanthine oxidase inhibitory properties and anti-inflammatory activity of 2-amino-5-alkylidene-thiazol-4-ones.
    Smelcerovic Z; Veljkovic A; Kocic G; Yancheva D; Petronijevic Z; Anderluh M; Smelcerovic A
    Chem Biol Interact; 2015 Mar; 229():73-81. PubMed ID: 25619642
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Novel N-substituted 5-aminosalicylamides as dual inhibitors of cyclooxygenase and 5-lipoxygenase enzymes: Synthesis, biological evaluation and docking study.
    El-Nagar MKS; Abdu-Allah HHM; Salem OIA; Kafafy AN; Farghaly HSM
    Bioorg Chem; 2018 Aug; 78():80-93. PubMed ID: 29550533
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Design, synthesis and pharmacobiological evaluation of novel acrylic acid derivatives acting as lipoxygenase and cyclooxygenase-1 inhibitors with antioxidant and anti-inflammatory activities.
    Pontiki E; Hadjipavlou-Litina D; Litinas K; Nicolotti O; Carotti A
    Eur J Med Chem; 2011 Jan; 46(1):191-200. PubMed ID: 21106277
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Thiopyranol[2,3,4-c,d]indoles as inhibitors of 5-lipoxygenase, 5-lipoxygenase-activating protein, and leukotriene C4 synthase.
    Hutchinson JH; Charleson S; Evans JF; Falgueyret JP; Hoogsteen K; Jones TR; Kargman S; Macdonald D; McFarlane CS; Nicholson DW
    J Med Chem; 1995 Oct; 38(22):4538-47. PubMed ID: 7473582
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Aspirin analogues as dual cyclooxygenase-2/5-lipoxygenase inhibitors: synthesis, nitric oxide release, molecular modeling, and biological evaluation as anti-inflammatory agents.
    Kaur J; Bhardwaj A; Huang Z; Knaus EE
    ChemMedChem; 2012 Jan; 7(1):144-50. PubMed ID: 22095955
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Synthesis and biological evaluation of a class of 5-benzylidene-2-phenyl-thiazolinones as potent 5-lipoxygenase inhibitors.
    Barzen S; Rödl CB; Lill A; Steinhilber D; Stark H; Hofmann B
    Bioorg Med Chem; 2012 Jun; 20(11):3575-83. PubMed ID: 22551629
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 7.