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13. Studies on angiotensin converting enzyme inhibitors. 4. Synthesis and angiotensin converting enzyme inhibitory activities of 3-acyl-1-alkyl-2-oxoimidazolidine-4-carboxylic acid derivatives. Hayashi K; Nunami K; Kato J; Yoneda N; Kubo M; Ochiai T; Ishida R J Med Chem; 1989 Feb; 32(2):289-97. PubMed ID: 2913292 [TBL] [Abstract][Full Text] [Related]
14. Pharmacological profiles of CS-622, a novel angiotensin converting enzyme inhibitor. Oizumi K; Koike H; Sada T; Miyamoto M; Nishino H; Matsushita Y; Iijima Y; Yanagisawa H Jpn J Pharmacol; 1988 Nov; 48(3):349-56. PubMed ID: 2851680 [TBL] [Abstract][Full Text] [Related]
15. Temocaprilat, a novel angiotensin-converting enzyme inhibitor, is excreted in bile via an ATP-dependent active transporter (cMOAT) that is deficient in Eisai hyperbilirubinemic mutant rats (EHBR). Ishizuka H; Konno K; Naganuma H; Sasahara K; Kawahara Y; Niinuma K; Suzuki H; Sugiyama Y J Pharmacol Exp Ther; 1997 Mar; 280(3):1304-11. PubMed ID: 9067317 [TBL] [Abstract][Full Text] [Related]
16. Angiotensin-converting enzyme inhibitors: new orally active 1,4-thiazepine-2,5-diones, 1,4-thiazine-2,5-diones, and 1,4-benzothiazepine-2,5-diones possessing antihypertensive activity. Skiles JW; Suh JT; Williams BE; Menard PR; Barton JN; Loev B; Jones H; Neiss ES; Schwab A; Mann WS J Med Chem; 1986 May; 29(5):784-96. PubMed ID: 3009814 [TBL] [Abstract][Full Text] [Related]
17. Angiotensin converting enzyme inhibitors: structure-activity profile of 1-benzazepin-2-one derivatives. Stanton JL; Watthey JW; Desai MN; Finn BM; Babiarz JE; Tomaselli HC J Med Chem; 1985 Nov; 28(11):1603-6. PubMed ID: 2999394 [TBL] [Abstract][Full Text] [Related]
18. Synthesis and structure-activity relationships of potent new angiotensin converting enzyme inhibitors containing saturated bicyclic amino acids. Blankley CJ; Kaltenbronn JS; DeJohn DE; Werner A; Bennett LR; Bobowski G; Krolls U; Johnson DR; Pearlman WM; Hoefle ML J Med Chem; 1987 Jun; 30(6):992-8. PubMed ID: 3035180 [TBL] [Abstract][Full Text] [Related]
19. Synthesis of 2-substituted-N-carboxymethyl-1,5-benzothiazepin-4-ones and -1,4-benzothiazin-3-ones and their evaluation as angiotensin converting enzyme inhibitors. Trapani G; Latrofa A; Franco M; Liso G Farmaco; 1995 Feb; 50(2):107-12. PubMed ID: 7766274 [TBL] [Abstract][Full Text] [Related]
20. Synthesis and angiotensin converting enzyme-inhibitory activity of 1,5-benzothiazepine and 1,5-benzoxazepine derivatives. III. Itoh K; Kori M; Inada Y; Nishikawa K; Kawamatsu Y; Sugihara H Chem Pharm Bull (Tokyo); 1986 Sep; 34(9):3747-61. PubMed ID: 3028653 [No Abstract] [Full Text] [Related] [Next] [New Search]