137 related articles for article (PubMed ID: 32009412)
1. Rapid Access to Kinase Inhibitor Pharmacophores by Regioselective C-H Arylation of Thieno[2,3-
Yamada S; Flesch KN; Murakami K; Itami K
Org Lett; 2020 Feb; 22(4):1547-1551. PubMed ID: 32009412
[TBL] [Abstract][Full Text] [Related]
2. Catalyst-Switchable Regiocontrol in the Direct Arylation of Remote C-H Groups in Pyrazolo[1,5-a]pyrimidines.
Bedford RB; Durrant SJ; Montgomery M
Angew Chem Int Ed Engl; 2015 Jul; 54(30):8787-90. PubMed ID: 26095315
[TBL] [Abstract][Full Text] [Related]
3. Palladium-catalyzed direct arylation of azine and azole N-oxides: reaction development, scope and applications in synthesis.
Campeau LC; Stuart DR; Leclerc JP; Bertrand-Laperle M; Villemure E; Sun HY; Lasserre S; Guimond N; Lecavallier M; Fagnou K
J Am Chem Soc; 2009 Mar; 131(9):3291-306. PubMed ID: 19215128
[TBL] [Abstract][Full Text] [Related]
4. Pd-catalyzed regioselective arylation on the C-5 position of N-aryl 1,2,3-triazoles.
Yamajala KD; Patil M; Banerjee S
J Org Chem; 2015 Mar; 80(6):3003-11. PubMed ID: 25710598
[TBL] [Abstract][Full Text] [Related]
5. Divergent synthesis of kinase inhibitor derivatives, leading to discovery of selective Gck inhibitors.
Matsumaru T; Inai M; Ishigami K; Iwamatsu T; Maita H; Otsuguro S; Nomura T; Matsuda A; Ichikawa S; Sakaitani M; Shuto S; Maenaka K; Kan T
Bioorg Med Chem Lett; 2017 May; 27(10):2144-2147. PubMed ID: 28385506
[TBL] [Abstract][Full Text] [Related]
6. Palladium-catalyzed direct C-H arylation of cyclic enaminones with aryl iodides.
Yu YY; Bi L; Georg GI
J Org Chem; 2013 Jun; 78(12):6163-9. PubMed ID: 23750615
[TBL] [Abstract][Full Text] [Related]
7. Completely N1-selective palladium-catalyzed arylation of unsymmetric imidazoles: application to the synthesis of nilotinib.
Ueda S; Su M; Buchwald SL
J Am Chem Soc; 2012 Jan; 134(1):700-6. PubMed ID: 22126442
[TBL] [Abstract][Full Text] [Related]
8. Highly regioselective palladium-catalyzed direct arylation of oxazole at C-2 or C-5 with aryl bromides, chlorides, and triflates.
Strotman NA; Chobanian HR; Guo Y; He J; Wilson JE
Org Lett; 2010 Aug; 12(16):3578-81. PubMed ID: 20704397
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and biological evaluation of benzo[4,5]imidazo[1,2-c]pyrimidine and benzo[4,5]imidazo[1,2-a]pyrazine derivatives as anaplastic lymphoma kinase inhibitors.
Tardy S; Orsato A; Mologni L; Bisson WH; Donadoni C; Gambacorti-Passerini C; Scapozza L; Gueyrard D; Goekjian PG
Bioorg Med Chem; 2014 Feb; 22(4):1303-12. PubMed ID: 24468632
[TBL] [Abstract][Full Text] [Related]
10. Aromaticity-Dependent Regioselectivity in Pd(II)-Catalyzed C-H Direct Arylation of Aryl Ureas.
Jiang P; Li F; Xu Y; Liu Q; Wang J; Ding H; Yu R; Wang Q
Org Lett; 2015 Dec; 17(23):5918-21. PubMed ID: 26575848
[TBL] [Abstract][Full Text] [Related]
11. Access and regioselective transformations of 6-substituted 4-aryl-2,8-dichloropyrido[3,2-d]pyrimidine compounds.
Bouscary-Desforges G; Bombrun A; Augustine JK; Bernardinelli G; Quattropani A
J Org Chem; 2012 May; 77(10):4586-95. PubMed ID: 22500580
[TBL] [Abstract][Full Text] [Related]
12. C-H bond functionalization under metalation-deprotonation process: regioselective direct arylation of 3-aminoimidazo[1,2-a]pyrazine.
Guchhait SK; Kandekar S; Kashyap M; Taxak N; Bharatam PV
J Org Chem; 2012 Sep; 77(18):8321-8. PubMed ID: 22928611
[TBL] [Abstract][Full Text] [Related]
13. One-pot synthesis of pyrimido[1,6-a]indol-1(2H)-one derivatives by a nucleophilic addition/Cu-catalyzed N-arylation/Pd-catalyzed C-H activation sequential process.
Wang ZJ; Yang JG; Yang F; Bao W
Org Lett; 2010 Jul; 12(13):3034-7. PubMed ID: 20527777
[TBL] [Abstract][Full Text] [Related]
14. Palladium-catalyzed regioselective C-5 arylation of protected L-histidine: microwave-assisted C-H activation adjacent to donor arm.
Mahindra A; Bagra N; Jain R
J Org Chem; 2013 Nov; 78(21):10954-9. PubMed ID: 24098973
[TBL] [Abstract][Full Text] [Related]
15. Synthetic strategy for increasing solubility of potential FLT3 inhibitor thieno[2,3-d]pyrimidine derivatives through structural modifications at the C
Oh C; Kim H; Kang JS; Yun J; Sim J; Kim HM; Han G
Bioorg Med Chem Lett; 2017 Feb; 27(3):496-500. PubMed ID: 28043794
[TBL] [Abstract][Full Text] [Related]
16. Regioselective Synthesis of New 2,4-(Het)aryl-3H-pyrido[1',2':1,5]pyrazolo[4,3-d]pyrimidines Involving Palladium-Catalyzed Cross-Coupling Reactions.
Ejjoummany A; Belaroussi R; El Hakmaoui A; Akssira M; Guillaumet G; Buron F; Routier S
Molecules; 2018 Oct; 23(11):. PubMed ID: 30360579
[TBL] [Abstract][Full Text] [Related]
17. Palladium-assisted regioselective C-H cyanation of heteroarenes using isonitrile as cyanide source.
Xu S; Huang X; Hong X; Xu B
Org Lett; 2012 Sep; 14(17):4614-7. PubMed ID: 22905784
[TBL] [Abstract][Full Text] [Related]
18. Design and synthesis of novel protein kinase CK2 inhibitors on the base of 4-aminothieno[2,3-d]pyrimidines.
Ostrynska OV; Balanda AO; Bdzhola VG; Golub AG; Kotey IM; Kukharenko OP; Gryshchenko AA; Briukhovetska NV; Yarmoluk SM
Eur J Med Chem; 2016 Jun; 115():148-60. PubMed ID: 27017545
[TBL] [Abstract][Full Text] [Related]
19. Efficient one-pot synthesis of 2,4-di(het)aryl and 2,4-diamino pyrido[3,2-d]pyrimidines involving regioselective S(N)Ar and palladium-catalyzed reactions.
Tikad A; Routier S; Akssira M; Guillaumet G
Org Biomol Chem; 2009 Dec; 7(24):5113-8. PubMed ID: 20024106
[TBL] [Abstract][Full Text] [Related]
20. Regioselective direct C-3 arylation of imidazo[1,2-a]pyridines with aryl tosylates and mesylates promoted by palladium-phosphine complexes.
Choy PY; Luk KC; Wu Y; So CM; Wang LL; Kwong FY
J Org Chem; 2015 Feb; 80(3):1457-63. PubMed ID: 25607730
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
