182 related articles for article (PubMed ID: 32044580)
21. A potentiated cooperation of carbonic anhydrase IX and histone deacetylase inhibitors against cancer.
Ruzzolini J; Laurenzana A; Andreucci E; Peppicelli S; Bianchini F; Carta F; Supuran CT; Romanelli MN; Nediani C; Calorini L
J Enzyme Inhib Med Chem; 2020 Dec; 35(1):391-397. PubMed ID: 31865754
[TBL] [Abstract][Full Text] [Related]
22. Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: Design, synthesis and anti-proliferative activity.
Higazy S; Samir N; El-Khouly A; Giovannuzzi S; Begines P; Gaber HM; Supuran CT; Abouzid KAM
Bioorg Chem; 2024 Mar; 144():107089. PubMed ID: 38237393
[TBL] [Abstract][Full Text] [Related]
23. Design, synthesis and mechanism study of coumarin-sulfonamide derivatives as carbonic anhydrase IX inhibitors with anticancer activity.
Lv Q; Zhang J; Cai J; Chen L; Liang J; Zhang T; Lin J; Chen R; Zhang Z; Guo P; Hong Y; Pan L; Ji H
Chem Biol Interact; 2024 Apr; 393():110947. PubMed ID: 38479716
[TBL] [Abstract][Full Text] [Related]
24. Cancer Drug Development of Carbonic Anhydrase Inhibitors beyond the Active Site.
Singh S; Lomelino CL; Mboge MY; Frost SC; McKenna R
Molecules; 2018 Apr; 23(5):. PubMed ID: 29710858
[TBL] [Abstract][Full Text] [Related]
25. Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX.
Leitans J; Kazaks A; Bogans J; Supuran CT; Akopjana I; Ivanova J; Zalubovskis R; Tars K
ChemMedChem; 2023 Nov; 18(22):e202300454. PubMed ID: 37837260
[TBL] [Abstract][Full Text] [Related]
26. Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors.
Sufian MA; Zamanova S; Shabana AM; Kemp B; Mondal UK; Supuran CT; Ilies MA
Int J Mol Sci; 2023 Feb; 24(5):. PubMed ID: 36902027
[TBL] [Abstract][Full Text] [Related]
27. A sucrose-binding site provides a lead towards an isoform-specific inhibitor of the cancer-associated enzyme carbonic anhydrase IX.
Pinard MA; Aggarwal M; Mahon BP; Tu C; McKenna R
Acta Crystallogr F Struct Biol Commun; 2015 Oct; 71(Pt 10):1352-8. PubMed ID: 26457530
[TBL] [Abstract][Full Text] [Related]
28. 1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory Activities.
Elsawi AE; Elbadawi MM; Nocentini A; Almahli H; Giovannuzzi S; Shaldam M; Salem R; Ibrahim TM; Abdel-Aziz HA; Supuran CT; Eldehna WM
J Med Chem; 2023 Aug; 66(15):10558-10578. PubMed ID: 37501287
[TBL] [Abstract][Full Text] [Related]
29. The carbonic anhydrase IX inhibitor SLC-0111 sensitises cancer cells to conventional chemotherapy.
Andreucci E; Ruzzolini J; Peppicelli S; Bianchini F; Laurenzana A; Carta F; Supuran CT; Calorini L
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):117-123. PubMed ID: 30362384
[TBL] [Abstract][Full Text] [Related]
30. Targeting carbonic anhydrases for the management of hypoxic metastatic tumors.
Supuran CT
Expert Opin Ther Pat; 2023 Nov; 33(11):701-720. PubMed ID: 37545058
[TBL] [Abstract][Full Text] [Related]
31. A novel class of phenylpyrazolone-sulphonamides rigid synthetic anticancer molecules selectively inhibit the isoform IX of carbonic anhydrases guided by molecular docking and orbital analyses.
Khayat MT; Ahmed HEA; Omar AM; Muhammad YA; Mohammad KA; Malebari AM; Khayyat AN; Halawa AH; Abulkhair HS; Al-Karmalawy AA; Almaghrabi M; Alharbi M; Aljahdali AS; El-Agrody AM
J Biomol Struct Dyn; 2023; 41(24):15243-15261. PubMed ID: 36914238
[TBL] [Abstract][Full Text] [Related]
32. Inhibitor binding to metal-substituted metalloenzyme: Sulfonamide affinity for carbonic anhydrase IX.
Baronas D; Knašienė B; Mickevičiūtė A; Jachno J; Naujalis E; Zubrienė A; Matulis D
J Inorg Biochem; 2024 Jul; 256():112547. PubMed ID: 38581802
[TBL] [Abstract][Full Text] [Related]
33. Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases.
Fuentes-Aguilar A; González-Bakker A; Jovanović M; Stojanov SJ; Puerta A; Gargano A; Dinić J; Vega-Báez JL; Merino-Montiel P; Montiel-Smith S; Alcaro S; Nocentini A; Pešić M; Supuran CT; Padrón JM; Fernández-Bolaños JG; López Ó
Bioorg Chem; 2024 Apr; 145():107168. PubMed ID: 38354500
[TBL] [Abstract][Full Text] [Related]
34. Insights towards sulfonamide drug specificity in α-carbonic anhydrases.
Aggarwal M; Kondeti B; McKenna R
Bioorg Med Chem; 2013 Mar; 21(6):1526-33. PubMed ID: 22985956
[TBL] [Abstract][Full Text] [Related]
35. Carbonic anhydrase IX: An atypical target for innovative therapies in cancer.
Ronca R; Supuran CT
Biochim Biophys Acta Rev Cancer; 2024 Jul; 1879(4):189120. PubMed ID: 38801961
[TBL] [Abstract][Full Text] [Related]
36. Design and synthesis of new adamantyl derivatives as promising antiproliferative agents.
Shahin AI; Zaraei SO; AlKubaisi BO; Ullah S; Anbar HS; El-Gamal R; Menon V; Abdel-Maksoud MS; Oh CH; El-Awady R; Gelsleichter NE; Pelletier J; Sévigny J; Iqbal J; Al-Tel TH; El-Gamal MI
Eur J Med Chem; 2023 Jan; 246():114958. PubMed ID: 36470105
[TBL] [Abstract][Full Text] [Related]
37. Identification of 3-(5-cyano-6-oxo-pyridin-2-yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity.
Shaldam MA; Khalil AF; Almahli H; Jaballah MY; Angeli A; Khaleel EF; Badi RM; Elkaeed EB; Supuran CT; Eldehna WM; Tawfik HO
Arch Pharm (Weinheim); 2024 Jan; 357(1):e2300449. PubMed ID: 37828544
[TBL] [Abstract][Full Text] [Related]
38. Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma.
Tawfik HO; Saleh MM; Ammara A; Khaleel EF; Badi R; Khater YTT; Rasheed RA; Attia AA; Hefny SM; Elkaeed EB; Nocentini A; Supuran CT; Eldehna WM; Shaldam MA
J Med Chem; 2024 Jan; 67(2):1611-1623. PubMed ID: 38207099
[TBL] [Abstract][Full Text] [Related]
39. High-Affinity NIR-Fluorescent Inhibitors for Tumor Imaging via Carbonic Anhydrase IX.
Žvinys G; Petrosiute A; Zakšauskas A; Zubrienė A; Ščerbavičienė A; Kalnina Z; Čapkauskaitė E; Juozapaitienė V; Mickevičiu Tė A; Shubin K; Grincevičienė Š; Raišys S; Tars K; Matulienė J; Matulis D
Bioconjug Chem; 2024 Jun; 35(6):790-803. PubMed ID: 38750635
[TBL] [Abstract][Full Text] [Related]
40. A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation.
Supuran CT
Bioorg Med Chem Lett; 2023 Sep; 93():129411. PubMed ID: 37507055
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
