190 related articles for article (PubMed ID: 32150343)
1. Detection of Small-Molecule Aggregation with High-Throughput Microplate Biophysical Methods.
Allen SJ; Dower CM; Liu AX; Lumb KJ
Curr Protoc Chem Biol; 2020 Mar; 12(1):e78. PubMed ID: 32150343
[TBL] [Abstract][Full Text] [Related]
2. Applications of Biophysics in High-Throughput Screening Hit Validation.
Genick CC; Barlier D; Monna D; Brunner R; Bé C; Scheufler C; Ottl J
J Biomol Screen; 2014 Jun; 19(5):707-14. PubMed ID: 24695619
[TBL] [Abstract][Full Text] [Related]
3. Solubility at the molecular level: development of a critical aggregation concentration (CAC) assay for estimating compound monomer solubility.
Wang J; Matayoshi E
Pharm Res; 2012 Jul; 29(7):1745-54. PubMed ID: 22422319
[TBL] [Abstract][Full Text] [Related]
4. Fragment screening using X-ray crystallography.
Davies TG; Tickle IJ
Top Curr Chem; 2012; 317():33-59. PubMed ID: 21678136
[TBL] [Abstract][Full Text] [Related]
5. Phenotypic approaches to small-molecule discovery in chemical biology.
Wagner BK; Dey M
Cell Chem Biol; 2021 Mar; 28(3):245. PubMed ID: 33740431
[No Abstract] [Full Text] [Related]
6. Open access high throughput drug discovery in the public domain: a Mount Everest in the making.
Roy A; McDonald PR; Sittampalam S; Chaguturu R
Curr Pharm Biotechnol; 2010 Nov; 11(7):764-78. PubMed ID: 20809896
[TBL] [Abstract][Full Text] [Related]
7. Addressing Compound Reactivity and Aggregation Assay Interferences: Case Studies of Biochemical High-Throughput Screening Campaigns Benefiting from the National Institutes of Health
Coussens NP; Auld DS; Thielman JR; Wagner BK; Dahlin JL
SLAS Discov; 2021 Dec; 26(10):1280-1290. PubMed ID: 34218710
[TBL] [Abstract][Full Text] [Related]
8. Frequent hitters: nuisance artifacts in high-throughput screening.
Yang ZY; He JH; Lu AP; Hou TJ; Cao DS
Drug Discov Today; 2020 Apr; 25(4):657-667. PubMed ID: 31987936
[TBL] [Abstract][Full Text] [Related]
9. Review article: high-throughput affinity-based technologies for small-molecule drug discovery.
Zhu Z; Cuozzo J
J Biomol Screen; 2009 Dec; 14(10):1157-64. PubMed ID: 19822881
[TBL] [Abstract][Full Text] [Related]
10. Data-driven approaches used for compound library design, hit triage and bioactivity modeling in high-throughput screening.
Paricharak S; Méndez-Lucio O; Chavan Ravindranath A; Bender A; IJzerman AP; van Westen GJP
Brief Bioinform; 2018 Mar; 19(2):277-285. PubMed ID: 27789427
[TBL] [Abstract][Full Text] [Related]
11. The European Lead Factory: An updated HTS compound library for innovative drug discovery.
van Vlijmen H; Ortholand JY; Li VM; de Vlieger JSB
Drug Discov Today; 2021 Oct; 26(10):2406-2413. PubMed ID: 33892142
[TBL] [Abstract][Full Text] [Related]
12. Solid-phase biological assays for drug discovery.
Forsberg EM; Sicard C; Brennan JD
Annu Rev Anal Chem (Palo Alto Calif); 2014; 7():337-59. PubMed ID: 25000820
[TBL] [Abstract][Full Text] [Related]
13. Non-stoichiometric inhibition in integrated lead finding - a literature review.
Klumpp M
Expert Opin Drug Discov; 2016; 11(2):149-62. PubMed ID: 26653534
[TBL] [Abstract][Full Text] [Related]
14. Learning from our mistakes: the 'unknown knowns' in fragment screening.
Davis BJ; Erlanson DA
Bioorg Med Chem Lett; 2013 May; 23(10):2844-52. PubMed ID: 23562240
[TBL] [Abstract][Full Text] [Related]
15. Resonant waveguide grating based assays for colloidal aggregate detection and promiscuity characterization in natural products.
Wang R; Wang J; Liu Y; Zhang X; Liang X
RSC Adv; 2019 Nov; 9(65):38055-38064. PubMed ID: 35541809
[TBL] [Abstract][Full Text] [Related]
16. A Guide to Run Affinity Screens Using Differential Scanning Fluorimetry and Surface Plasmon Resonance Assays.
Bergsdorf C; Wright SK
Methods Enzymol; 2018; 610():135-165. PubMed ID: 30390797
[TBL] [Abstract][Full Text] [Related]
17. High Throughput Differential Scanning Fluorimetry (DSF) Formulation Screening with Complementary Dyes to Assess Protein Unfolding and Aggregation in Presence of Surfactants.
McClure SM; Ahl PL; Blue JT
Pharm Res; 2018 Mar; 35(4):81. PubMed ID: 29508082
[TBL] [Abstract][Full Text] [Related]
18. Cheminformatics approaches to analyze diversity in compound screening libraries.
Akella LB; DeCaprio D
Curr Opin Chem Biol; 2010 Jun; 14(3):325-30. PubMed ID: 20457001
[TBL] [Abstract][Full Text] [Related]
19. Covalent hits and where to find them.
Lucas SCC; Blackwell JH; Hewitt SH; Semple H; Whitehurst BC; Xu H
SLAS Discov; 2024 Apr; 29(3):100142. PubMed ID: 38278484
[TBL] [Abstract][Full Text] [Related]
20. Brief Guide: Experimental Strategies for High-Quality Hit Selection from Small-Molecule Screening Campaigns.
Rothenaigner I; Hadian K
SLAS Discov; 2021 Aug; 26(7):851-854. PubMed ID: 33882754
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]