286 related articles for article (PubMed ID: 32209254)
1. Identification of protein tyrosine phosphatase 1B (PTP1B) inhibitors through De Novo Evoluton, synthesis, biological evaluation and molecular dynamics simulation.
Wu J; Ma Y; Zhou H; Zhou L; Du S; Sun Y; Li W; Dong W; Wang R
Biochem Biophys Res Commun; 2020 May; 526(1):273-280. PubMed ID: 32209254
[TBL] [Abstract][Full Text] [Related]
2. Design, synthesis, biological activity and molecular dynamics studies of specific protein tyrosine phosphatase 1B inhibitors over SHP-2.
Sun SX; Li XB; Liu WB; Ma Y; Wang RL; Cheng XC; Wang SQ; Liu W
Int J Mol Sci; 2013 Jun; 14(6):12661-74. PubMed ID: 23774838
[TBL] [Abstract][Full Text] [Related]
3. Discovery and evaluation of the hybrid of bromophenol and saccharide as potent and selective protein tyrosine phosphatase 1B inhibitors.
Zhang R; Yu R; Xu Q; Li X; Luo J; Jiang B; Wang L; Guo S; Wu N; Shi D
Eur J Med Chem; 2017 Jul; 134():24-33. PubMed ID: 28395151
[TBL] [Abstract][Full Text] [Related]
4. Design and Biological Evaluation of Novel Imidazolyl Flavonoids as Potent and Selective Protein Tyrosine Phosphatase Inhibitors.
Han RY; Ge Y; Zhang L; Wang QM
Med Chem; 2020; 16(4):563-574. PubMed ID: 31208312
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
Sun LP; Gao LX; Ma WP; Nan FJ; Li J; Piao HR
Chem Biol Drug Des; 2012 Oct; 80(4):584-90. PubMed ID: 22805439
[TBL] [Abstract][Full Text] [Related]
6. Synthesis, biological evaluation and in silico studies of 5-(3-methoxybenzylidene)thiazolidine-2,4-dione analogues as PTP1B inhibitors.
Mahapatra MK; Kumar R; Kumar M
Bioorg Chem; 2017 Apr; 71():1-9. PubMed ID: 28126289
[TBL] [Abstract][Full Text] [Related]
7. Discovery of novel, high potent, ABC type PTP1B inhibitors with TCPTP selectivity and cellular activity.
Liu P; Du Y; Song L; Shen J; Li Q
Eur J Med Chem; 2016 Aug; 118():27-33. PubMed ID: 27123900
[TBL] [Abstract][Full Text] [Related]
8. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
[TBL] [Abstract][Full Text] [Related]
9. Design, synthesis, biological evaluation and molecular dynamics studies of 4-thiazolinone derivatives as protein tyrosine phosphatase 1B (PTP1B) inhibitors.
Liu WS; Wang RR; Yue H; Zheng ZH; Lu XH; Wang SQ; Dong WL; Wang RL
J Biomol Struct Dyn; 2020 Aug; 38(13):3814-3824. PubMed ID: 31490104
[TBL] [Abstract][Full Text] [Related]
10. Toward a treatment of diabesity: Rational design, synthesis and biological evaluation of benzene-sulfonamide derivatives as a new class of PTP-1B inhibitors.
Ghareb N; El-Sayed NM; Abdelhameed R; Yamada K; Elgawish MS
Bioorg Chem; 2019 May; 86():322-338. PubMed ID: 30743173
[TBL] [Abstract][Full Text] [Related]
11. Design, synthesis, biological evaluation and molecular dynamics simulation studies of imidazolidine-2,4-dione derivatives as novel PTP1B inhibitors.
Ma Y; Ding TT; Liu YY; Zheng ZH; Sun SX; Zhang LS; Zhang H; Lu XH; Cheng XC; Wang RL
Biochem Biophys Res Commun; 2021 Nov; 579():40-46. PubMed ID: 34583194
[TBL] [Abstract][Full Text] [Related]
12. Design and synthesis of paracaseolide A analogues as selective protein tyrosine phosphatase 1B inhibitors.
Yin JP; Tang CL; Gao LX; Ma WP; Li JY; Li Y; Li J; Nan FJ
Org Biomol Chem; 2014 Jun; 12(21):3441-5. PubMed ID: 24752625
[TBL] [Abstract][Full Text] [Related]
13. Flavonoids as potent allosteric inhibitors of protein tyrosine phosphatase 1B: molecular dynamics simulation and free energy calculation.
Zargari F; Lotfi M; Shahraki O; Nikfarjam Z; Shahraki J
J Biomol Struct Dyn; 2018 Nov; 36(15):4126-4142. PubMed ID: 29216799
[TBL] [Abstract][Full Text] [Related]
14. Discovery of novel high potent and cellular active ADC type PTP1B inhibitors with selectivity over TC-PTP via modification interacting with C site.
Du Y; Zhang Y; Ling H; Li Q; Shen J
Eur J Med Chem; 2018 Jan; 144():692-700. PubMed ID: 29289892
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors.
Campos-Almazán MI; Flores-Ramos M; Hernández-Campos A; Castillo R; Sierra-Campos E; Torgeson K; Peti W; Valdez-Solana M; Oria-Hernández J; Méndez ST; Castillo-Villanueva A; Jiménez-de Jesús H; Avitia-Domínguez C; Téllez-Valencia A
Bioorg Med Chem; 2021 Oct; 48():116418. PubMed ID: 34563877
[TBL] [Abstract][Full Text] [Related]
16. Identification and characterization of potent and selective inhibitors targeting protein tyrosine phosphatase 1B (PTP1B).
Jin J; Ye X; Boateng D; Dai K; Ye F; Du P; Yu H
Bioorg Med Chem Lett; 2019 Aug; 29(16):2358-2363. PubMed ID: 31221555
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and biological evaluation of novel N-aryl-ω-(benzoazol-2-yl)-sulfanylalkanamides as dual inhibitors of α-glucosidase and protein tyrosine phosphatase 1B.
Wang MY; Cheng XC; Chen XB; Li Y; Zang LL; Duan YQ; Chen MZ; Yu P; Sun H; Wang RL
Chem Biol Drug Des; 2018 Sep; 92(3):1647-1656. PubMed ID: 29745030
[TBL] [Abstract][Full Text] [Related]
18. Pyrazoles as novel protein tyrosine phosphatase 1B (PTP1B) inhibitors: An in vitro and in silico study.
Rocha S; Lucas M; Silva VLM; Gomes PMO; Silva AMS; Araújo AN; Aniceto N; Guedes RC; Corvo ML; Fernandes E; Freitas M
Int J Biol Macromol; 2021 Jun; 181():1171-1182. PubMed ID: 33857515
[TBL] [Abstract][Full Text] [Related]
19. Synthesis of small peptide compounds, molecular docking, and inhibitory activity evaluation against phosphatases PTP1B and SHP2.
Kostrzewa T; Sahu KK; Gorska-Ponikowska M; Tuszynski JA; Kuban-Jankowska A
Drug Des Devel Ther; 2018; 12():4139-4147. PubMed ID: 30584278
[TBL] [Abstract][Full Text] [Related]
20. Design and synthesis of imidazolidine-2,4-dione derivatives as selective inhibitors by targeting protein tyrosine phosphatase-1B over T-cell protein tyrosine phosphatase.
Ma Y; Sun SX; Cheng XC; Wang SQ; Dong WL; Wang RL; Xu WR
Chem Biol Drug Des; 2013 Nov; 82(5):595-602. PubMed ID: 23848232
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]