BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

80 related articles for article (PubMed ID: 3255316)

  • 1. Synthesis and aromatase inhibiting activity of aminoglutethimide analogs.
    Aboul-Enein HY
    Drug Des Deliv; 1988 Feb; 2(3):221-6. PubMed ID: 3255316
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Pharmacology of aminoglutethimide: structure/activity relationships and receptor interactions.
    Nicholls PJ; Daly MJ; Smith HJ
    Breast Cancer Res Treat; 1986; 7 Suppl():S55-67. PubMed ID: 3755630
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and structure-activity relationships of 6-substituted androst-4-ene analogs as aromatase inhibitors.
    Numazawa M; Kamiyama T; Tachibana M; Oshibe M
    J Med Chem; 1996 May; 39(11):2245-52. PubMed ID: 8667367
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and biochemical evaluation of novel inhibitors of aromatase (AR) using an enhanced representation of the active site of AR derived from the consideration of the reaction mechanism.
    Ahmed S; Amanuel Y
    Biochem Biophys Res Commun; 2000 Jan; 267(1):356-61. PubMed ID: 10623624
    [TBL] [Abstract][Full Text] [Related]  

  • 5. In vitro inhibition of aromatase by the enantiomers of aminoglutethimide and analogs.
    Ogbunude PO; Aboul-Enein HY
    Chirality; 1994; 6(8):623-6. PubMed ID: 7857773
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Analogues of aminoglutethimide based on 1-phenyl-3-azabicyclo[3.1.0]hexane-2,4-dione: selective inhibition of aromatase activity.
    Rowlands MG; Bunnett MA; Foster AB; Jarman M; Stanek J; Schweizer E
    J Med Chem; 1988 May; 31(5):971-6. PubMed ID: 3361583
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and biochemical evaluation of analogues of aminoglutethimide based on phenylpyrrolidine-2,5-dione.
    Daly MJ; Jones GW; Nicholls PJ; Smith HJ; Rowlands MG; Bunnett MA
    J Med Chem; 1986 Apr; 29(4):520-3. PubMed ID: 3754286
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Inhibition of aromatase as treatment of breast carcinoma in postmenopausal women.
    Santen RJ; Boucher AE; Santner SJ; Henderson IC; Harvey H; Lipton A
    J Lab Clin Med; 1987 Mar; 109(3):278-89. PubMed ID: 3546561
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Selective aromatase inhibition by pyridoglutethimide, an analogue of aminoglutethimide.
    Kitawaki J; Yamamoto T; Urabe M; Tamura T; Inoue S; Honjo H; Okada H
    Acta Endocrinol (Copenh); 1990 May; 122(5):592-8. PubMed ID: 2353556
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and biological evaluation of 3-(prop-2-enyl)- and 3-(prop-2-ynyl)pyrrolidine-2,5-dione derivatives as potential aromatase inhibitors.
    Barrell KJ; Woo WL; Ahmadi M; Smith HJ; Nicholls PJ
    J Pharm Pharmacol; 1996 Feb; 48(2):154-9. PubMed ID: 8935164
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Structure-activity relationships of a new family of steroidal aromatase inhibitors. 1. Synthesis and evaluation of a series of analogs related to 19-[(methylthio)methyl]androstenedione (RU54115).
    Lesuisse D; Gourvest JF; Benslimane O; Canu F; Delaisi C; Doucet B; Hartmann C; Lefrançois JM; Tric B; Mansuy D; Philibert D; Teutsch G
    J Med Chem; 1996 Feb; 39(3):757-72. PubMed ID: 8576919
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Aromatase inhibitors--mechanisms for non-steroidal inhibitors.
    Vanden Bossche HV; Moereels H; Koymans LM
    Breast Cancer Res Treat; 1994; 30(1):43-55. PubMed ID: 7949204
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Analogues of aminoglutethimide: selective inhibition of cholesterol side-chain cleavage.
    Foster AB; Jarman M; Leung CS; Rowlands MG; Taylor GN
    J Med Chem; 1983 Jan; 26(1):50-4. PubMed ID: 6827528
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Structure-activity relationships of new A,D-ring modified steroids as aromatase inhibitors: design, synthesis, and biological activity evaluation.
    Cepa MM; Tavares da Silva EJ; Correia-da-Silva G; Roleira FM; Teixeira NA
    J Med Chem; 2005 Oct; 48(20):6379-85. PubMed ID: 16190763
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and evaluation of benzimidazole and imidazole compounds as potential aromatase inhibitors.
    Hida F; Robert J; Luu-Duc C
    Farmaco; 1994; 49(7-8):489-92. PubMed ID: 7945714
    [TBL] [Abstract][Full Text] [Related]  

  • 16. [Inhibitors of aromatase. Synthesis and pharmacologic action of potential mammary tumor-inhibiting 4-alkyl-3-(4-aminophenyl)-3-ethylpiperidine-2,6-diones].
    Batzl C; Hartmann RW
    Arch Pharm (Weinheim); 1987 Jan; 320(1):51-8. PubMed ID: 3566486
    [No Abstract]   [Full Text] [Related]  

  • 17. Analogues of aminoglutethimide: selective inhibition of aromatase.
    Foster AB; Jarman M; Leung CS; Rowlands MG; Taylor GN; Plevey RG; Sampson P
    J Med Chem; 1985 Feb; 28(2):200-4. PubMed ID: 3968684
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Effects of aromatase inhibitors, aminoglutethimide, and 4-hydroxyandrostenedione on cyclic rats and rats with 7,12-dimethylbenz(a)anthracene-induced mammary tumors.
    Wing LY; Garrett WM; Brodie AM
    Cancer Res; 1985 Jun; 45(6):2425-8. PubMed ID: 3921242
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Aromatase inhibition by an 11,13-dihydroderivative of a sesquiterpene lactone.
    Blanco JG; Gil RR; Bocco JL; Meragelman TL; Genti-Raimondi S; Flury A
    J Pharmacol Exp Ther; 2001 Jun; 297(3):1099-105. PubMed ID: 11356934
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Analogues of 3-ethyl-3-(4-pyridyl)piperidine-2,6-dione as selective inhibitors of aromatase: derivatives with variable 1-alkyl and 3-alkyl substituents.
    Leung CS; Rowlands MG; Jarman M; Foster AB; Griggs LJ; Wilman DE
    J Med Chem; 1987 Sep; 30(9):1550-4. PubMed ID: 3625703
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 4.