BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

502 related articles for article (PubMed ID: 32711085)

  • 1. Novel bis(pyrazole-benzofuran) hybrids possessing piperazine linker: Synthesis of potent bacterial biofilm and MurB inhibitors.
    Mekky AEM; Sanad SMH
    Bioorg Chem; 2020 Sep; 102():104094. PubMed ID: 32711085
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Hydrazonoyl bromide precursors as DHFR inhibitors for the synthesis of bis-thiazolyl pyrazole derivatives; antimicrobial activities, antibiofilm, and drug combination studies against MRSA.
    Ibrahim SA; Fayed EA; Rizk HF; Desouky SE; Ragab A
    Bioorg Chem; 2021 Nov; 116():105339. PubMed ID: 34530234
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Novel ciprofloxacin hybrids using biology oriented drug synthesis (BIODS) approach: Anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis, topoisomerase II inhibition, and antibacterial activity.
    Kassab AE; Gedawy EM
    Eur J Med Chem; 2018 Apr; 150():403-418. PubMed ID: 29547830
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Design, synthesis and biological evaluation of novel pleuromutilin derivatives containing piperazine and 1,2,3-triazole linker.
    Zhang GY; Zhang Z; Li K; Liu J; Li B; Jin Z; Liu YH; Tang YZ
    Bioorg Chem; 2020 Dec; 105():104398. PubMed ID: 33137559
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Discovery of New Schiff Bases Tethered Pyrazole Moiety: Design, Synthesis, Biological Evaluation, and Molecular Docking Study as Dual Targeting DHFR/DNA Gyrase Inhibitors with Immunomodulatory Activity.
    Hassan AS; Askar AA; Naglah AM; Almehizia AA; Ragab A
    Molecules; 2020 Jun; 25(11):. PubMed ID: 32498469
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and antimicrobial evaluation of 1-(benzofuran-2-yl)-4-nitro-3-arylbutan-1-ones and 3-(benzofuran-2-yl)-4,5-dihydro-5-aryl-1-[4-(aryl)-1,3-thiazol-2-yl]-1H-pyrazoles.
    Abdel-Wahab BF; Abdel-Aziz HA; Ahmed EM
    Eur J Med Chem; 2009 Jun; 44(6):2632-5. PubMed ID: 18995932
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and evaluation of antimicrobial and anticancer activities of 3-phenyl-1-phenylsulfonyl pyrazoles containing an aminoguanidine moiety.
    Huang Y; Hu H; Yan R; Lin L; Song M; Yao X
    Arch Pharm (Weinheim); 2021 Feb; 354(2):e2000165. PubMed ID: 33047391
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Pyrazolidine-3,5-diones and 5-hydroxy-1H-pyrazol-3(2H)-ones, inhibitors of UDP-N-acetylenolpyruvyl glucosamine reductase.
    Gilbert AM; Failli A; Shumsky J; Yang Y; Severin A; Singh G; Hu W; Keeney D; Petersen PJ; Katz AH
    J Med Chem; 2006 Oct; 49(20):6027-36. PubMed ID: 17004716
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and anti-staphylococcal activity of new 4-diazopyrazole derivatives.
    Raimondi MV; Maggio B; Raffa D; Plescia F; Cascioferro S; Cancemi G; Schillaci D; Cusimano MG; Vitale M; Daidone G
    Eur J Med Chem; 2012 Dec; 58():64-71. PubMed ID: 23088933
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis of novel 1,2-diarylpyrazolidin-3-one-based compounds and their evaluation as broad spectrum antibacterial agents.
    Mokbel SA; Fathalla RK; El-Sharkawy LY; Abadi AH; Engel M; Abdel-Halim M
    Bioorg Chem; 2020 Jun; 99():103759. PubMed ID: 32220665
    [TBL] [Abstract][Full Text] [Related]  

  • 11. 3,5-dioxopyrazolidines, novel inhibitors of UDP-N- acetylenolpyruvylglucosamine reductase (MurB) with activity against gram-positive bacteria.
    Yang Y; Severin A; Chopra R; Krishnamurthy G; Singh G; Hu W; Keeney D; Svenson K; Petersen PJ; Labthavikul P; Shlaes DM; Rasmussen BA; Failli AA; Shumsky JS; Kutterer KM; Gilbert A; Mansour TS
    Antimicrob Agents Chemother; 2006 Feb; 50(2):556-64. PubMed ID: 16436710
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis, antimicrobial, anti-cancer and in silico studies of new urea derivatives.
    Sroor FM; Othman AM; Tantawy MA; Mahrous KF; El-Naggar ME
    Bioorg Chem; 2021 Jul; 112():104953. PubMed ID: 33964581
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Optimization of activity localization of quinoline derivatives: Design, synthesis, and dual evaluation of biological activity for potential antitumor and antibacterial agents.
    Jin G; Li Z; Xiao F; Qi X; Sun X
    Bioorg Chem; 2020 Jun; 99():103837. PubMed ID: 32299019
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis, in-vitro and in-silico study of novel thiazoles as potent antibacterial agents and MurB inhibitors.
    Sanad SMH; Ahmed AAM; Mekky AEM
    Arch Pharm (Weinheim); 2020 Apr; 353(4):e1900309. PubMed ID: 31967349
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of 3,5-Bis(trifluoromethyl)phenyl-Substituted Pyrazole Derivatives as Potent Growth Inhibitors of Drug-Resistant Bacteria.
    Alkhaibari IS; Kc HR; Roy S; Abu-Gazleh MK; Gilmore DF; Alam MA
    Molecules; 2021 Aug; 26(16):. PubMed ID: 34443670
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and antibacterial and cytotoxic activities of new N-3 substituted thiazolidine-2,4-dione derivatives bearing the pyrazole moiety.
    Desai NC; Satodiya HM; Kotadiya GM; Vaghani HV
    Arch Pharm (Weinheim); 2014 Jul; 347(7):523-32. PubMed ID: 24729458
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 4-4-(Anilinomethyl)-3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-ylbenzoic acid derivatives as potent anti-gram-positive bacterial agents.
    Hansa RK; Khan MMK; Frangie MM; Gilmore DF; Shelton RS; Savenka AV; Basnakian AG; Shuttleworth SL; Smeltzer MS; Alam MA
    Eur J Med Chem; 2021 Jul; 219():113402. PubMed ID: 33845234
    [TBL] [Abstract][Full Text] [Related]  

  • 18. 1-Substituted carbamoyl and thiocarbamoyl-4,5-dihydro-1H-pyrazoles as possible cytotoxic and antimicrobial agents.
    Khan KA; Faidallah HM
    J Enzyme Inhib Med Chem; 2016 Aug; 31(4):619-27. PubMed ID: 26114308
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis, anticancer and antimicrobial evaluation of new benzofuran based derivatives: PI3K inhibition, quorum sensing and molecular modeling study.
    El-Khouly OA; Henen MA; El-Sayed MA; Shabaan MI; El-Messery SM
    Bioorg Med Chem; 2021 Feb; 31():115976. PubMed ID: 33388654
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis, antitumor activity and molecular docking study of novel benzofuran-2-yl pyrazole pyrimidine derivatives.
    El-Zahar MI; Adb El-Karim SS; Haiba ME; Khedr MA
    Acta Pol Pharm; 2011; 68(3):357-73. PubMed ID: 21648190
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 26.