BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

200 related articles for article (PubMed ID: 32942905)

  • 1. Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases.
    Aspatwar A; Berrino E; Bua S; Carta F; Capasso C; Parkkila S; Supuran CT
    J Enzyme Inhib Med Chem; 2020 Dec; 35(1):1765-1772. PubMed ID: 32942905
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases.
    De Luca L; Mancuso F; Ferro S; Buemi MR; Angeli A; Del Prete S; Capasso C; Supuran CT; Gitto R
    Eur J Med Chem; 2018 Jan; 143():276-282. PubMed ID: 29197732
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Benzoxepinones: A new isoform-selective class of tumor associated carbonic anhydrase inhibitors.
    Grandane A; Nocentini A; Werner T; Zalubovskis R; Supuran CT
    Bioorg Med Chem; 2020 Jun; 28(11):115496. PubMed ID: 32327349
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile.
    Sharonova T; Zhmurov P; Kalinin S; Nocentini A; Angeli A; Ferraroni M; Korsakov M; Supuran CT; Krasavin M
    J Enzyme Inhib Med Chem; 2022 Dec; 37(1):857-865. PubMed ID: 35296197
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and carbonic anhydrase inhibitory properties of novel coumarin derivatives.
    Karatas MO; Alici B; Cakir U; Cetinkaya E; Demir D; Ergün A; Gençer N; Arslan O
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):299-304. PubMed ID: 22512727
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Coumarins inhibit η-class carbonic anhydrase from
    Giovannuzzi S; De Luca V; Nocentini A; Capasso C; Supuran CT
    J Enzyme Inhib Med Chem; 2022 Dec; 37(1):680-685. PubMed ID: 35139744
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis of coumarin-sulfonamide derivatives and determination of their cytotoxicity, carbonic anhydrase inhibitory and molecular docking studies.
    Zengin Kurt B; Sonmez F; Ozturk D; Akdemir A; Angeli A; Supuran CT
    Eur J Med Chem; 2019 Dec; 183():111702. PubMed ID: 31542715
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Metronidazole-coumarin conjugates and 3-cyano-7-hydroxy-coumarin act as isoform-selective carbonic anhydrase inhibitors.
    Bonneau A; Maresca A; Winum JY; Supuran CT
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):397-401. PubMed ID: 22299576
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Coumarins effectively inhibit bacterial α-carbonic anhydrases.
    Giovannuzzi S; Hewitt CS; Nocentini A; Capasso C; Flaherty DP; Supuran CT
    J Enzyme Inhib Med Chem; 2022 Dec; 37(1):333-338. PubMed ID: 34979838
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Carbonic anhydrase inhibition for the management of cerebral ischemia: in vivo evaluation of sulfonamide and coumarin inhibitors.
    Di Cesare Mannelli L; Micheli L; Carta F; Cozzi A; Ghelardini C; Supuran CT
    J Enzyme Inhib Med Chem; 2016 Dec; 31(6):894-9. PubMed ID: 26607399
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation.
    Kartsev V; Geronikaki A; Bua S; Nocentini A; Petrou A; Lichitsky B; Frasinyuk M; Leitans J; Kazaks A; Tars K; Supuran CT
    Molecules; 2019 Oct; 24(19):. PubMed ID: 31590289
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors.
    Angeli A; Carta F; Bartolucci G; Supuran CT
    Bioorg Med Chem; 2017 Jul; 25(13):3567-3573. PubMed ID: 28522267
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Novel sulfonamide bearing coumarin scaffolds as selective inhibitors of tumor associated carbonic anhydrase isoforms IX and XII.
    Chandak N; Ceruso M; Supuran CT; Sharma PK
    Bioorg Med Chem; 2016 Jul; 24(13):2882-2886. PubMed ID: 27137360
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis of aminocyanopyrazoles via a multi-component reaction and anti-carbonic anhydrase inhibitory activity of their sulfamide derivatives against cytosolic and transmembrane isoforms.
    Allouche F; Chabchoub F; Carta F; Supuran CT
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):343-9. PubMed ID: 23013533
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups.
    Bozdag M; Ferraroni M; Carta F; Vullo D; Lucarini L; Orlandini E; Rossello A; Nuti E; Scozzafava A; Masini E; Supuran CT
    J Med Chem; 2014 Nov; 57(21):9152-67. PubMed ID: 25310626
    [TBL] [Abstract][Full Text] [Related]  

  • 16.
    Aspatwar A; Hammaren M; Parikka M; Parkkila S; Carta F; Bozdag M; Vullo D; Supuran CT
    J Enzyme Inhib Med Chem; 2020 Dec; 35(1):65-71. PubMed ID: 31663386
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and biological evaluation of some coumarin hybrids as selective carbonic anhydrase IX and XII inhibitors.
    Thacker PS; Sridhar Goud N; Argulwar OS; Soman J; Angeli A; Alvala M; Arifuddin M; Supuran CT
    Bioorg Chem; 2020 Nov; 104():104272. PubMed ID: 32961467
    [TBL] [Abstract][Full Text] [Related]  

  • 18. New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases.
    Huentupil Y; Peña L; Novoa N; Berrino E; Arancibia R; Supuran CT
    J Enzyme Inhib Med Chem; 2019 Dec; 34(1):451-458. PubMed ID: 30734605
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes.
    Bua S; Berrino E; Del Prete S; Murthy VS; Vijayakumar V; Tamboli Y; Capasso C; Cerbai E; Mugelli A; Carta F; Supuran CT
    J Enzyme Inhib Med Chem; 2018 Dec; 33(1):1125-1136. PubMed ID: 29987956
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Spirocyclic sulfonamides with carbonic anhydrase inhibitory and anti-neuropathic pain activity.
    Kalisha Vali Y; Gundla R; Singh OV; Tamboli Y; Di Cesare Manelli L; Ghelardini C; Al-Tamimi AS; Carta F; Angeli A; Supuran CT
    Bioorg Chem; 2019 Nov; 92():103210. PubMed ID: 31473472
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.