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4. Randomized Trial of Verubecestat for Prodromal Alzheimer's Disease. Egan MF; Kost J; Voss T; Mukai Y; Aisen PS; Cummings JL; Tariot PN; Vellas B; van Dyck CH; Boada M; Zhang Y; Li W; Furtek C; Mahoney E; Harper Mozley L; Mo Y; Sur C; Michelson D N Engl J Med; 2019 Apr; 380(15):1408-1420. PubMed ID: 30970186 [TBL] [Abstract][Full Text] [Related]
5. Efficacy and Safety of Lanabecestat for Treatment of Early and Mild Alzheimer Disease: The AMARANTH and DAYBREAK-ALZ Randomized Clinical Trials. Wessels AM; Tariot PN; Zimmer JA; Selzler KJ; Bragg SM; Andersen SW; Landry J; Krull JH; Downing AM; Willis BA; Shcherbinin S; Mullen J; Barker P; Schumi J; Shering C; Matthews BR; Stern RA; Vellas B; Cohen S; MacSweeney E; Boada M; Sims JR JAMA Neurol; 2020 Feb; 77(2):199-209. PubMed ID: 31764959 [TBL] [Abstract][Full Text] [Related]
6. Lessons that can be learnt from the failure of verubecestat in Alzheimer's disease. Doggrell SA Expert Opin Pharmacother; 2019 Dec; 20(17):2095-2099. PubMed ID: 31423903 [No Abstract] [Full Text] [Related]
7. Further analyses of the safety of verubecestat in the phase 3 EPOCH trial of mild-to-moderate Alzheimer's disease. Egan MF; Mukai Y; Voss T; Kost J; Stone J; Furtek C; Mahoney E; Cummings JL; Tariot PN; Aisen PS; Vellas B; Lines C; Michelson D Alzheimers Res Ther; 2019 Aug; 11(1):68. PubMed ID: 31387606 [TBL] [Abstract][Full Text] [Related]
8. Retinal Optical Coherence Tomography Metrics Are Unchanged in Verubecestat Alzheimer's Disease Clinical Trial but Correlate with Baseline Regional Brain Atrophy. Sergott RC; Raji A; Kost J; Sur C; Jackson S; Locco A; Patel A; Furtek C; Mattson B; Egan MF J Alzheimers Dis; 2021; 79(1):275-287. PubMed ID: 33252075 [TBL] [Abstract][Full Text] [Related]
9. Chronic Verubecestat Treatment Suppresses Amyloid Accumulation in Advanced Aged Tg2576-AβPPswe Mice Without Inducing Microhemorrhage. Villarreal S; Zhao F; Hyde LA; Holder D; Forest T; Sondey M; Chen X; Sur C; Parker EM; Kennedy ME J Alzheimers Dis; 2017; 59(4):1393-1413. PubMed ID: 28800329 [TBL] [Abstract][Full Text] [Related]
10. Neuropathology of a patient with Alzheimer disease treated with low doses of verubecestat. Querol-Vilaseca M; Sirisi S; Molina-Porcel L; Molina B; Pegueroles J; Ferrer-Raventós P; Nuñez-Llaves R; Dols-Icardo O; Balasa M; Iulita MF; Blesa R; Belbin O; Clarimon J; Fortea J; Gelpi E; Sánchez-Valle R; Lleó A Neuropathol Appl Neurobiol; 2022 Apr; 48(3):e12781. PubMed ID: 34825396 [TBL] [Abstract][Full Text] [Related]
11. Merck ends trial of potential Alzheimer's drug verubecestat. Hawkes N BMJ; 2017 Feb; 356():j845. PubMed ID: 28202490 [No Abstract] [Full Text] [Related]
13. β-secretase inhibitors for Alzheimer's disease: heading in the wrong direction? Selkoe D Lancet Neurol; 2019 Jul; 18(7):624-626. PubMed ID: 31202466 [No Abstract] [Full Text] [Related]
14. Future Therapeutics in Alzheimer's Disease: Development Status of BACE Inhibitors. Evin G BioDrugs; 2016 Jun; 30(3):173-94. PubMed ID: 27023706 [TBL] [Abstract][Full Text] [Related]
16. Emerging drugs to reduce abnormal β-amyloid protein in Alzheimer's disease patients. Panza F; Seripa D; Solfrizzi V; Imbimbo BP; Lozupone M; Leo A; Sardone R; Gagliardi G; Lofano L; Creanza BC; Bisceglia P; Daniele A; Bellomo A; Greco A; Logroscino G Expert Opin Emerg Drugs; 2016 Dec; 21(4):377-391. PubMed ID: 27678025 [TBL] [Abstract][Full Text] [Related]
17. BACE inhibitors in clinical development for the treatment of Alzheimer's disease. Panza F; Lozupone M; Solfrizzi V; Sardone R; Piccininni C; Dibello V; Stallone R; Giannelli G; Bellomo A; Greco A; Daniele A; Seripa D; Logroscino G; Imbimbo BP Expert Rev Neurother; 2018 Nov; 18(11):847-857. PubMed ID: 30277096 [TBL] [Abstract][Full Text] [Related]
18. BACE inhibitor bust in Alzheimer trial. Mullard A Nat Rev Drug Discov; 2017 Mar; 16(3):155. PubMed ID: 28248932 [No Abstract] [Full Text] [Related]
19. Synthesis and evaluation of multi-target-directed ligands with BACE-1 inhibitory and Nrf2 agonist activities as potential agents against Alzheimer's disease. Qu L; Ji L; Wang C; Luo H; Li S; Peng W; Yin F; Lu D; Liu X; Kong L; Wang X Eur J Med Chem; 2021 Jul; 219():113441. PubMed ID: 33862517 [TBL] [Abstract][Full Text] [Related]
20. Evaluation of the efficacy, safety and tolerability of orally administered BI 409306, a novel phosphodiesterase type 9 inhibitor, in two randomised controlled phase II studies in patients with prodromal and mild Alzheimer's disease. Frölich L; Wunderlich G; Thamer C; Roehrle M; Garcia M; Dubois B Alzheimers Res Ther; 2019 Feb; 11(1):18. PubMed ID: 30755255 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]