153 related articles for article (PubMed ID: 33151676)
1. X-ray Structure and Molecular Docking Guided Discovery of Novel Chitinase Inhibitors with a Scaffold of Dipyridopyrimidine-3-carboxamide.
Yuan P; Jiang X; Wang S; Shao X; Yang Q; Qian X
J Agric Food Chem; 2020 Nov; 68(47):13584-13593. PubMed ID: 33151676
[TBL] [Abstract][Full Text] [Related]
2. Discovery of aromatic 2-(3-(methylcarbamoyl) guanidino)-N-aylacetamides as highly potent chitinase inhibitors.
Zhao Z; Li F; Chen W; Yang Q; Lu H; Zhang J
Bioorg Med Chem; 2023 Feb; 80():117172. PubMed ID: 36709570
[TBL] [Abstract][Full Text] [Related]
3. Novel Inhibitors of an Insect Pest Chitinase: Design and Optimization of 9-O-Aromatic and Heterocyclic Esters of Berberine.
Zhu L; Chen L; Shao X; Cheng J; Yang Q; Qian X
J Agric Food Chem; 2021 Jul; 69(27):7526-7533. PubMed ID: 34212716
[No Abstract] [Full Text] [Related]
4. Crystal structure-guided design of berberine-based novel chitinase inhibitors.
Chen L; Zhu L; Chen J; Chen W; Qian X; Yang Q
J Enzyme Inhib Med Chem; 2020 Dec; 35(1):1937-1943. PubMed ID: 33167737
[TBL] [Abstract][Full Text] [Related]
5. Rational Design, Synthesis, and Biological Investigations of
Zhao Z; Xu Q; Chen W; Wang S; Yang Q; Dong Y; Zhang J
J Agric Food Chem; 2022 Apr; 70(16):4889-4898. PubMed ID: 35416043
[TBL] [Abstract][Full Text] [Related]
6. A Novel Scaffold for Developing Specific or Broad-Spectrum Chitinase Inhibitors.
Jiang X; Kumar A; Liu T; Zhang KY; Yang Q
J Chem Inf Model; 2016 Dec; 56(12):2413-2420. PubMed ID: 28024404
[TBL] [Abstract][Full Text] [Related]
7. Design of Inhibitors Targeting Chitin-Degrading Enzymes by Bioisostere Substitutions and Scaffold Hopping for Selective Control of
Liang P; Li J; Chen W; Zhou H; Lai X; Li J; Xu Z; Yang Q; Zhang J
J Agric Food Chem; 2024 May; 72(19):10794-10804. PubMed ID: 38711396
[TBL] [Abstract][Full Text] [Related]
8. Discovery of Azo-Aminopyrimidines as Novel and Potent Chitinase O
Dong L; Shen S; Jiang X; Liu Y; Li J; Chen W; Wang Y; Shi J; Liu J; Ma S; Zhang L; Dong J; Yang Q
J Agric Food Chem; 2022 Sep; 70(38):12203-12210. PubMed ID: 36121180
[TBL] [Abstract][Full Text] [Related]
9. Structure, Catalysis, and Inhibition of
Liu T; Chen L; Zhou Y; Jiang X; Duan Y; Yang Q
J Biol Chem; 2017 Feb; 292(6):2080-2088. PubMed ID: 28053084
[TBL] [Abstract][Full Text] [Related]
10. A Series of Compounds Bearing a Dipyrido-Pyrimidine Scaffold Acting as Novel Human and Insect Pest Chitinase Inhibitors.
Jiang X; Kumar A; Motomura Y; Liu T; Zhou Y; Moro K; Zhang KYJ; Yang Q
J Med Chem; 2020 Feb; 63(3):987-1001. PubMed ID: 31928006
[TBL] [Abstract][Full Text] [Related]
11. Fully deacetylated chitooligosaccharides act as efficient glycoside hydrolase family 18 chitinase inhibitors.
Chen L; Zhou Y; Qu M; Zhao Y; Yang Q
J Biol Chem; 2014 Jun; 289(25):17932-40. PubMed ID: 24828498
[TBL] [Abstract][Full Text] [Related]
12. Structural analysis of group II chitinase (ChtII) catalysis completes the puzzle of chitin hydrolysis in insects.
Chen W; Qu M; Zhou Y; Yang Q
J Biol Chem; 2018 Feb; 293(8):2652-2660. PubMed ID: 29317504
[TBL] [Abstract][Full Text] [Related]
13. Pocket-based Lead Optimization Strategy for the Design and Synthesis of Chitinase Inhibitors.
Dong Y; Hu S; Jiang X; Liu T; Ling Y; He X; Yang Q; Zhang L
J Agric Food Chem; 2019 Apr; 67(13):3575-3582. PubMed ID: 30865442
[TBL] [Abstract][Full Text] [Related]
14. Structure-based virtual screening of highly potent inhibitors of the nematode chitinase
Chen W; Chen Q; Kumar A; Jiang X; Zhang KYJ; Yang Q
J Enzyme Inhib Med Chem; 2021 Dec; 36(1):1198-1204. PubMed ID: 34074203
[TBL] [Abstract][Full Text] [Related]
15. Development of Novel Pesticides Targeting Insect Chitinases: A Minireview and Perspective.
Chen W; Yang Q
J Agric Food Chem; 2020 Apr; 68(16):4559-4565. PubMed ID: 32239934
[TBL] [Abstract][Full Text] [Related]
16. Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry.
Hirose T; Sunazuka T; Sugawara A; Endo A; Iguchi K; Yamamoto T; Ui H; Shiomi K; Watanabe T; Sharpless KB; Omura S
J Antibiot (Tokyo); 2009 May; 62(5):277-82. PubMed ID: 19329983
[TBL] [Abstract][Full Text] [Related]
17. Microbial Secondary Metabolite, Phlegmacin B
Chen L; Liu T; Duan Y; Lu X; Yang Q
J Agric Food Chem; 2017 May; 65(19):3851-3857. PubMed ID: 28457127
[TBL] [Abstract][Full Text] [Related]
18. Chitinases: Therapeutic Scaffolds for Allergy and Inflammation.
Madan K; Madan M; Sharma S; Paliwal S
Recent Pat Inflamm Allergy Drug Discov; 2020; 14(1):46-57. PubMed ID: 31934842
[TBL] [Abstract][Full Text] [Related]
19. Human Chitinases: Structure, Function, and Inhibitor Discovery.
Kumar A; Zhang KYJ
Adv Exp Med Biol; 2019; 1142():221-251. PubMed ID: 31102249
[TBL] [Abstract][Full Text] [Related]
20. Discovery of ZQ-
Yang L; Chen M; Han X; Liu C; Wang C; Zhang G; Yang D; Zhao S
J Agric Food Chem; 2022 Sep; 70(36):11314-11323. PubMed ID: 36054909
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]