These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

156 related articles for article (PubMed ID: 33202687)

  • 1. Novel 1-Amidino-4-Phenylpiperazines as Potent Agonists at Human TAAR1 Receptor: Rational Design, Synthesis, Biological Evaluation and Molecular Docking Studies.
    Francesconi V; Cichero E; Kanov EV; Laurini E; Pricl S; Gainetdinov RR; Tonelli M
    Pharmaceuticals (Basel); 2020 Nov; 13(11):. PubMed ID: 33202687
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling.
    Grossi G; Scarano N; Musumeci F; Tonelli M; Kanov E; Carbone A; Fossa P; Gainetdinov RR; Cichero E; Schenone S
    Molecules; 2024 Apr; 29(8):. PubMed ID: 38675561
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Novel biguanide-based derivatives scouted as TAAR1 agonists: Synthesis, biological evaluation, ADME prediction and molecular docking studies.
    Tonelli M; Espinoza S; Gainetdinov RR; Cichero E
    Eur J Med Chem; 2017 Feb; 127():781-792. PubMed ID: 27823885
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Rational design, chemical synthesis and biological evaluation of novel biguanides exploring species-specificity responsiveness of TAAR1 agonists.
    Guariento S; Tonelli M; Espinoza S; Gerasimov AS; Gainetdinov RR; Cichero E
    Eur J Med Chem; 2018 Feb; 146():171-184. PubMed ID: 29407948
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Pharmacologic characterization of the cloned human trace amine-associated receptor1 (TAAR1) and evidence for species differences with the rat TAAR1.
    Wainscott DB; Little SP; Yin T; Tu Y; Rocco VP; He JX; Nelson DL
    J Pharmacol Exp Ther; 2007 Jan; 320(1):475-85. PubMed ID: 17038507
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Trace amine associated receptor 1 (TAAR1) modulators: a patent review (2010-present).
    Tonelli M; Cichero E
    Expert Opin Ther Pat; 2020 Feb; 30(2):137-145. PubMed ID: 31865810
    [No Abstract]   [Full Text] [Related]  

  • 7. Further insights into the pharmacology of the human trace amine-associated receptors: discovery of novel ligands for TAAR1 by a virtual screening approach.
    Cichero E; Espinoza S; Franchini S; Guariento S; Brasili L; Gainetdinov RR; Fossa P
    Chem Biol Drug Des; 2014 Dec; 84(6):712-20. PubMed ID: 24894156
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Insights into the structure and pharmacology of the human trace amine-associated receptor 1 (hTAAR1): homology modelling and docking studies.
    Cichero E; Espinoza S; Gainetdinov RR; Brasili L; Fossa P
    Chem Biol Drug Des; 2013 Apr; 81(4):509-16. PubMed ID: 22883051
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Discovery of Guanfacine as a Novel TAAR1 Agonist: A Combination Strategy through Molecular Modeling Studies and Biological Assays.
    Cichero E; Francesconi V; Casini B; Casale M; Kanov E; Gerasimov AS; Sukhanov I; Savchenko A; Espinoza S; Gainetdinov RR; Tonelli M
    Pharmaceuticals (Basel); 2023 Nov; 16(11):. PubMed ID: 38004497
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Interaction analyses of hTAAR1 and mTAAR1 with antagonist EPPTB.
    Liao S; Pino MJ; Deleon C; Lindner-Jackson M; Wu C
    Life Sci; 2022 Jul; 300():120553. PubMed ID: 35452636
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Targeting species-specific trace amine-associated receptor 1 ligands: to date perspective of the rational drug design process.
    Cichero E; Tonelli M
    Future Med Chem; 2017 Sep; 9(13):1507-1527. PubMed ID: 28791911
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Biological evaluation and
    Wang Y; Liu Z; Lu J; Wang W; Wang L; Yang Y; Wang H; Ye L; Zhang J; Tian J
    Front Pharmacol; 2023; 14():1161964. PubMed ID: 37153799
    [No Abstract]   [Full Text] [Related]  

  • 13. In Vitro Characterization of Psychoactive Substances at Rat, Mouse, and Human Trace Amine-Associated Receptor 1.
    Simmler LD; Buchy D; Chaboz S; Hoener MC; Liechti ME
    J Pharmacol Exp Ther; 2016 Apr; 357(1):134-44. PubMed ID: 26791601
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Evolutionary Conservation of 3-Iodothyronamine as an Agonist at the Trace Amine-Associated Receptor 1.
    Cöster M; Biebermann H; Schöneberg T; Stäubert C
    Eur Thyroid J; 2015 Sep; 4(Suppl 1):9-20. PubMed ID: 26601069
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Trace amine-associated receptor 1 partial agonism reveals novel paradigm for neuropsychiatric therapeutics.
    Revel FG; Moreau JL; Gainetdinov RR; Ferragud A; Velázquez-Sánchez C; Sotnikova TD; Morairty SR; Harmeier A; Groebke Zbinden K; Norcross RD; Bradaia A; Kilduff TS; Biemans B; Pouzet B; Caron MG; Canales JJ; Wallace TL; Wettstein JG; Hoener MC
    Biol Psychiatry; 2012 Dec; 72(11):934-42. PubMed ID: 22705041
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists.
    Chiellini G; Nesi G; Digiacomo M; Malvasi R; Espinoza S; Sabatini M; Frascarelli S; Laurino A; Cichero E; Macchia M; Gainetdinov RR; Fossa P; Raimondi L; Zucchi R; Rapposelli S
    J Med Chem; 2015 Jun; 58(12):5096-107. PubMed ID: 26010728
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Identification of a Potent Human Trace Amine-Associated Receptor 1 Antagonist.
    Decker AM; Brackeen MF; Mohammadkhani A; Kormos CM; Hesk D; Borgland SL; Blough BE
    ACS Chem Neurosci; 2022 Apr; 13(7):1082-1095. PubMed ID: 35325532
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class.
    Lewin AH; Miller GM; Gilmour B
    Bioorg Med Chem; 2011 Dec; 19(23):7044-8. PubMed ID: 22037049
    [TBL] [Abstract][Full Text] [Related]  

  • 19. A rapid functional assay for the human trace amine-associated receptor 1 based on the mobilization of internal calcium.
    Navarro HA; Gilmour BP; Lewin AH
    J Biomol Screen; 2006 Sep; 11(6):688-93. PubMed ID: 16831861
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of Trace Amine Associated Receptor 1 (TAAR1) Agonist 2-(5-(4'-Chloro-[1,1'-biphenyl]-4-yl)-4
    Krasavin M; Lukin A; Sukhanov I; Gerasimov AS; Kuvarzin S; Efimova EV; Dorofeikova M; Nichugovskaya A; Matveev A; Onokhin K; Zakharov K; Gureev M; Gainetdinov RR
    Biomolecules; 2022 Nov; 12(11):. PubMed ID: 36359001
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.