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2. Cross-Resistance Among Next-Generation Antiandrogen Drugs Through the AKR1C3/AR-V7 Axis in Advanced Prostate Cancer. Zhao J; Ning S; Lou W; Yang JC; Armstrong CM; Lombard AP; D'Abronzo LS; Evans CP; Gao AC; Liu C Mol Cancer Ther; 2020 Aug; 19(8):1708-1718. PubMed ID: 32430485 [TBL] [Abstract][Full Text] [Related]
3. Mesoporous silica nanoparticles combined with AKR1C3 siRNA inhibited the growth of castration-resistant prostate cancer by suppressing androgen synthesis in vitro and in vivo. Chen J; Yang Y; Xu D; Li J; Wu S; Jiang Y; Wang C; Yang Z; Zhao L Biochem Biophys Res Commun; 2021 Feb; 540():83-89. PubMed ID: 33450484 [TBL] [Abstract][Full Text] [Related]
4. A 3-(4-nitronaphthen-1-yl) amino-benzoate analog as a bifunctional AKR1C3 inhibitor and AR antagonist: Head to head comparison with other advanced AKR1C3 targeted therapeutics. Wangtrakuldee P; Adeniji AO; Zang T; Duan L; Khatri B; Twenter BM; Estrada MA; Higgins TF; Winkler JD; Penning TM J Steroid Biochem Mol Biol; 2019 Sep; 192():105283. PubMed ID: 30641225 [TBL] [Abstract][Full Text] [Related]
5. Nuclear receptor ERRα contributes to castration-resistant growth of prostate cancer via its regulation of intratumoral androgen biosynthesis. Xu Z; Ma T; Zhou J; Gao W; Li Y; Yu S; Wang Y; Chan FL Theranostics; 2020; 10(9):4201-4216. PubMed ID: 32226548 [TBL] [Abstract][Full Text] [Related]
6. The AKR1C3/AR-V7 complex maintains CRPC tumour growth by repressing B4GALT1 expression. Wang B; Wu S; Fang Y; Sun G; He D; Hsieh JT; Wang X; Zeng H; Wu K J Cell Mol Med; 2020 Oct; 24(20):12032-12043. PubMed ID: 32902124 [TBL] [Abstract][Full Text] [Related]
7. Novel inhibition of AKR1C3 and androgen receptor axis by PTUPB synergizes enzalutamide treatment in advanced prostate cancer. Yang JC; Xu P; Ning S; Wasielewski LJ; Adomat H; Hwang SH; Morisseau C; Gleave M; Corey E; Gao AC; Lara PN; Evans CP; Hammock BD; Liu C Oncogene; 2023 Feb; 42(9):693-707. PubMed ID: 36596844 [TBL] [Abstract][Full Text] [Related]
8. A Mansonone Derivative Coupled with Monoclonal Antibody 4D5-Modified Chitosan Inhibit AKR1C3 to Treat Castration-Resistant Prostate Cancer. Zhou M; Wang X; Xia J; Cheng Y; Xiao L; Bei Y; Tang J; Huang Y; Xiang Q; Huang S Int J Nanomedicine; 2020; 15():3087-3098. PubMed ID: 32431503 [TBL] [Abstract][Full Text] [Related]
9. ERG/AKR1C3/AR Constitutes a Feed-Forward Loop for AR Signaling in Prostate Cancer Cells. Powell K; Semaan L; Conley-LaComb MK; Asangani I; Wu YM; Ginsburg KB; Williams J; Squire JA; Maddipati KR; Cher ML; Chinni SR Clin Cancer Res; 2015 Jun; 21(11):2569-79. PubMed ID: 25754347 [TBL] [Abstract][Full Text] [Related]
10. AKR1C3 Inhibitor KV-37 Exhibits Antineoplastic Effects and Potentiates Enzalutamide in Combination Therapy in Prostate Adenocarcinoma Cells. Verma K; Gupta N; Zang T; Wangtrakluldee P; Srivastava SK; Penning TM; Trippier PC Mol Cancer Ther; 2018 Sep; 17(9):1833-1845. PubMed ID: 29891491 [TBL] [Abstract][Full Text] [Related]
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