These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
43. 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: solution and X-ray crystallographic studies. Leitans J; Sprudza A; Tanc M; Vozny I; Zalubovskis R; Tars K; Supuran CT Bioorg Med Chem; 2013 Sep; 21(17):5130-8. PubMed ID: 23859774 [TBL] [Abstract][Full Text] [Related]
44. Iodoquinazolinones bearing benzenesulfonamide as human carbonic anhydrase I, II, IX and XII inhibitors: Synthesis, biological evaluation and radiosensitizing activity. Soliman AM; Ghorab MM; Bua S; Supuran CT Eur J Med Chem; 2020 Aug; 200():112449. PubMed ID: 32485534 [TBL] [Abstract][Full Text] [Related]
45. Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX. Garaj V; Puccetti L; Fasolis G; Winum JY; Montero JL; Scozzafava A; Vullo D; Innocenti A; Supuran CT Bioorg Med Chem Lett; 2005 Jun; 15(12):3102-8. PubMed ID: 15905091 [TBL] [Abstract][Full Text] [Related]
46. Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors. Clima L; Craciun BF; Angeli A; Petreni A; Bonardi A; Nocentini A; Carta F; Gratteri P; Pinteala M; Supuran CT ChemMedChem; 2020 Nov; 15(21):2052-2057. PubMed ID: 32744806 [TBL] [Abstract][Full Text] [Related]
47. In Vivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents. Bruno E; Buemi MR; De Luca L; Ferro S; Monforte AM; Supuran CT; Vullo D; De Sarro G; Russo E; Gitto R ChemMedChem; 2016 Aug; 11(16):1812-8. PubMed ID: 26915563 [TBL] [Abstract][Full Text] [Related]
48. Structural investigations on coumarins leading to chromeno[4,3-c]pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII. Bonardi A; Falsini M; Catarzi D; Varano F; Di Cesare Mannelli L; Tenci B; Ghelardini C; Angeli A; Supuran CT; Colotta V Eur J Med Chem; 2018 Feb; 146():47-59. PubMed ID: 29407972 [TBL] [Abstract][Full Text] [Related]
50. Carbonic anhydrase inhibitors: X-ray and molecular modeling study for the interaction of a fluorescent antitumor sulfonamide with isozyme II and IX. Alterio V; Vitale RM; Monti SM; Pedone C; Scozzafava A; Cecchi A; De Simone G; Supuran CT J Am Chem Soc; 2006 Jun; 128(25):8329-35. PubMed ID: 16787097 [TBL] [Abstract][Full Text] [Related]
51. 5-Arylisothiazol-3(2H)-one-1,(1)-(di)oxides: A new class of selective tumor-associated carbonic anhydrases (hCA IX and XII) inhibitors. Cornelio B; Laronze-Cochard M; Miambo R; De Grandis M; Riccioni R; Borisova B; Dontchev D; Machado C; Ceruso M; Fontana A; Supuran CT; Sapi J Eur J Med Chem; 2019 Aug; 175():40-48. PubMed ID: 31071549 [TBL] [Abstract][Full Text] [Related]
52. 3-Hydrazinoisatin-based benzenesulfonamides as novel carbonic anhydrase inhibitors endowed with anticancer activity: Synthesis, in vitro biological evaluation and in silico insights. Abo-Ashour MF; Eldehna WM; Nocentini A; Bonardi A; Bua S; Ibrahim HS; Elaasser MM; Kryštof V; Jorda R; Gratteri P; Abou-Seri SM; Supuran CT Eur J Med Chem; 2019 Dec; 184():111768. PubMed ID: 31629164 [TBL] [Abstract][Full Text] [Related]
54. Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. Sarikaya B; Ceruso M; Carta F; Supuran CT Bioorg Med Chem; 2014 Nov; 22(21):5883-90. PubMed ID: 25267005 [TBL] [Abstract][Full Text] [Related]
55. Effects of dopaminergic compounds on carbonic anhydrase isozymes I, II, and VI. Sentürk M; Ekinci D; Göksu S; Supuran CT J Enzyme Inhib Med Chem; 2012 Jun; 27(3):365-9. PubMed ID: 21699374 [TBL] [Abstract][Full Text] [Related]
56. Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors. Mishra CB; Kumari S; Angeli A; Monti SM; Buonanno M; Prakash A; Tiwari M; Supuran CT J Enzyme Inhib Med Chem; 2016; 31(sup2):174-179. PubMed ID: 27314170 [TBL] [Abstract][Full Text] [Related]
57. Discovery of potent anti-convulsant carbonic anhydrase inhibitors: Design, synthesis, in vitro and in vivo appraisal. Mishra CB; Kumari S; Angeli A; Bua S; Buonanno M; Monti SM; Tiwari M; Supuran CT Eur J Med Chem; 2018 Aug; 156():430-443. PubMed ID: 30015076 [TBL] [Abstract][Full Text] [Related]
58. Differential in vitro inhibition effects of some antibiotics on tumor associated carbonic anhydrase isozymes of hCA-IX and hCA-XII. Ozensoy O; Arslan O; Kockar F J Enzyme Inhib Med Chem; 2008 Aug; 23(4):579-85. PubMed ID: 18666004 [TBL] [Abstract][Full Text] [Related]
59. 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors. D'Ascenzio M; Secci D; Carradori S; Zara S; Guglielmi P; Cirilli R; Pierini M; Poli G; Tuccinardi T; Angeli A; Supuran CT J Med Chem; 2020 Mar; 63(5):2470-2488. PubMed ID: 31972093 [TBL] [Abstract][Full Text] [Related]