BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

186 related articles for article (PubMed ID: 33798546)

  • 1. COR758, a negative allosteric modulator of GABA
    Porcu A; Mostallino R; Serra V; Melis M; Sogos V; Beggiato S; Ferraro L; Manetti F; Gianibbi B; Bettler B; Corelli F; Mugnaini C; Castelli MP
    Neuropharmacology; 2021 May; 189():108537. PubMed ID: 33798546
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Pharmacological characterization of GABAB receptor subtypes assembled with auxiliary KCTD subunits.
    Rajalu M; Fritzius T; Adelfinger L; Jacquier V; Besseyrias V; Gassmann M; Bettler B
    Neuropharmacology; 2015 Jan; 88():145-54. PubMed ID: 25196734
    [TBL] [Abstract][Full Text] [Related]  

  • 3. In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator.
    Porcu A; Lobina C; Giunta D; Solinas M; Mugnaini C; Castelli MP
    Eur J Pharmacol; 2016 Nov; 791():115-123. PubMed ID: 27578262
    [TBL] [Abstract][Full Text] [Related]  

  • 4. KK-92A, a novel GABA
    Li X; Sturchler E; Kaczanowska K; Cameron M; Finn MG; Griffin P; McDonald P; Markou A
    Psychopharmacology (Berl); 2017 May; 234(9-10):1633-1644. PubMed ID: 28382542
    [TBL] [Abstract][Full Text] [Related]  

  • 5. The GABA
    Olianas MC; Dedoni S; Onali P
    Eur J Pharmacol; 2017 Jan; 794():135-146. PubMed ID: 27876620
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a Gα
    Porcu A; Melis M; Turecek R; Ullrich C; Mocci I; Bettler B; Gessa GL; Castelli MP
    Neuropharmacology; 2018 May; 133():107-120. PubMed ID: 29407764
    [TBL] [Abstract][Full Text] [Related]  

  • 7. GABA
    de Miguel E; Vekovischeva O; Kuokkanen K; Vesajoki M; Paasikoski N; Kaskinoro J; Myllymäki M; Lainiola M; Janhunen SK; Hyytiä P; Linden AM; Korpi ER
    Addict Biol; 2019 Nov; 24(6):1191-1203. PubMed ID: 30421860
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Mechanisms of allosteric modulation at GABAB receptors by CGP7930 and GS39783: effects on affinities and efficacies of orthosteric ligands with distinct intrinsic properties.
    Urwyler S; Gjoni T; Koljatić J; Dupuis DS
    Neuropharmacology; 2005 Mar; 48(3):343-53. PubMed ID: 15721166
    [TBL] [Abstract][Full Text] [Related]  

  • 9. In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE).
    Perdona' E; Costantini VJ; Tessari M; Martinelli P; Carignani C; Valerio E; Mok MH; Zonzini L; Visentini F; Gianotti M; Gordon L; Rocheville M; Corsi M; Capelli AM
    Neuropharmacology; 2011; 61(5-6):957-66. PubMed ID: 21756923
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Selected amino acids, dipeptides and arylalkylamine derivatives do not act as allosteric modulators at GABAB receptors.
    Urwyler S; Gjoni T; Kaupmann K; Pozza MF; Mosbacher J
    Eur J Pharmacol; 2004 Jan; 483(2-3):147-53. PubMed ID: 14729102
    [TBL] [Abstract][Full Text] [Related]  

  • 11. CGP7930 - An allosteric modulator of GABA
    Hannan SB; Penzinger R; Mickute G; Smart TG
    Neuropharmacology; 2023 Nov; 238():109644. PubMed ID: 37422181
    [TBL] [Abstract][Full Text] [Related]  

  • 12. The positive allosteric GABAB receptor modulator rac-BHFF enhances baclofen-mediated analgesia in neuropathic mice.
    Zemoura K; Ralvenius WT; Malherbe P; Benke D
    Neuropharmacology; 2016 Sep; 108():172-8. PubMed ID: 27108932
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Changes in the properties of allosteric and orthosteric GABAB receptor ligands after a continuous, desensitizing agonist pretreatment.
    Gjoni T; Urwyler S
    Eur J Pharmacol; 2009 Jan; 603(1-3):37-41. PubMed ID: 19109945
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Effects of intraperitoneal administration of the GABAB receptor positive allosteric modulator 2,6-di tert-butyl-4-(2-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) on food intake in non-deprived rats.
    Ebenezer IS
    Eur J Pharmacol; 2012 Sep; 690(1-3):115-8. PubMed ID: 22652431
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Role of CA1 GABA
    Ebrahimi-Ghiri M; Rostampour M; Jamshidi-Mehr M; Nasehi M; Zarrindast MR
    Brain Res; 2018 Jan; 1678():164-173. PubMed ID: 29038006
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Receptor activation involving positive allosteric modulation, unlike full agonism, does not result in GABAB receptor desensitization.
    Gjoni T; Urwyler S
    Neuropharmacology; 2008 Dec; 55(8):1293-9. PubMed ID: 18775443
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Structure optimization of positive allosteric modulators of GABA
    Mugnaini C; Brizzi A; Mostallino R; Castelli MP; Corelli F
    Bioorg Med Chem Lett; 2020 Sep; 30(18):127443. PubMed ID: 32730942
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Positive allosteric modulators at GABAB receptors exert intrinsic actions and enhance the influence of baclofen on light-induced phase shifts of hamster circadian activity rhythms.
    Gannon RL; Millan MJ
    Pharmacol Biochem Behav; 2011 Oct; 99(4):712-7. PubMed ID: 21756929
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Positive allosteric modulation of native and recombinant gamma-aminobutyric acid(B) receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its aldehyde analog CGP13501.
    Urwyler S; Mosbacher J; Lingenhoehl K; Heid J; Hofstetter K; Froestl W; Bettler B; Kaupmann K
    Mol Pharmacol; 2001 Nov; 60(5):963-71. PubMed ID: 11641424
    [TBL] [Abstract][Full Text] [Related]  

  • 20. GABAB receptor activation inhibits exocytosis in rat pancreatic beta-cells by G-protein-dependent activation of calcineurin.
    Braun M; Wendt A; Buschard K; Salehi A; Sewing S; Gromada J; Rorsman P
    J Physiol; 2004 Sep; 559(Pt 2):397-409. PubMed ID: 15235087
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.