207 related articles for article (PubMed ID: 33823393)
21. Tag-Convertible Photocrosslinker with Click-On/Off N-Acylsulfonamide Linkage for Protein Identification.
Hayashi R; Morimoto S; Tomohiro T
Chem Asian J; 2019 Sep; 14(18):3145-3148. PubMed ID: 31359597
[TBL] [Abstract][Full Text] [Related]
22. Evaluation of the cyclopentane-1,2-dione as a potential bio-isostere of the carboxylic acid functional group.
Ballatore C; Gay B; Huang L; Robinson KH; James MJ; Trojanowski JQ; Lee VM; Brunden KR; Smith AB
Bioorg Med Chem Lett; 2014 Sep; 24(17):4171-5. PubMed ID: 25127105
[TBL] [Abstract][Full Text] [Related]
23. Discovery of new indole-based acylsulfonamide Na
Wu YJ; Venables B; Guernon J; Chen J; Sit SY; Rajamani R; Knox RJ; Matchett M; Pieschl RL; Herrington J; Bristow LJ; Meanwell NA; Thompson LA; Dzierba C
Bioorg Med Chem Lett; 2019 Feb; 29(4):659-663. PubMed ID: 30638874
[TBL] [Abstract][Full Text] [Related]
24. Synthesis and evaluation of potent and selective beta(3) adrenergic receptor agonists containing acylsulfonamide, sulfonylsulfonamide, and sulfonylurea carboxylic acid isosteres.
Uehling DE; Donaldson KH; Deaton DN; Hyman CE; Sugg EE; Barrett DG; Hughes RG; Reitter B; Adkison KK; Lancaster ME; Lee F; Hart R; Paulik MA; Sherman BW; True T; Cowan C
J Med Chem; 2002 Jan; 45(3):567-83. PubMed ID: 11806709
[TBL] [Abstract][Full Text] [Related]
25. Bioisoteres for carboxylic acids: From ionized isosteres to novel unionized replacements.
Hall A; Chatzopoulou M; Frost J
Bioorg Med Chem; 2024 Apr; 104():117653. PubMed ID: 38579492
[TBL] [Abstract][Full Text] [Related]
26. Discovery and preclinical evaluation of potent, orally bioavailable, metabolically stable cyclopropylindolobenzazepine acylsulfonamides as thumb site 1 inhibitors of the hepatitis c virus NS5B RNA-dependent, RNA polymerase.
Hewawasam P; Tu Y; Gao M; Hanumegowda U; Knipe J; Lemm JA; Parker DD; Rigat KL; Roberts SB; Meanwell NA; Kadow JF
Bioorg Med Chem Lett; 2016 Feb; 26(3):936-940. PubMed ID: 26747393
[TBL] [Abstract][Full Text] [Related]
27. Recognition properties of carboxylic acid bioisosteres: anion binding by tetrazoles, aryl sulfonamides, and acyl sulfonamides on a calix[4]arene scaffold.
Pinter T; Jana S; Courtemanche RJ; Hof F
J Org Chem; 2011 May; 76(10):3733-41. PubMed ID: 21462934
[TBL] [Abstract][Full Text] [Related]
28. 2-Oxabicyclo[2.2.2]octane as a new bioisostere of the phenyl ring.
Levterov VV; Panasiuk Y; Sahun K; Stashkevych O; Badlo V; Shablykin O; Sadkova I; Bortnichuk L; Klymenko-Ulianov O; Holota Y; Lachmann L; Borysko P; Horbatok K; Bodenchuk I; Bas Y; Dudenko D; Mykhailiuk PK
Nat Commun; 2023 Oct; 14(1):5608. PubMed ID: 37783681
[TBL] [Abstract][Full Text] [Related]
29. Recent Developments in the Practical Application of Novel Carboxylic Acid Bioisosteres.
Horgan C; O'Sullivan TP
Curr Med Chem; 2022; 29(13):2203-2234. PubMed ID: 34420501
[TBL] [Abstract][Full Text] [Related]
30. Functional and structural analyses of N-acylsulfonamide-linked dinucleoside inhibitors of RNase A.
Thiyagarajan N; Smith BD; Raines RT; Acharya KR
FEBS J; 2011 Feb; 278(3):541-9. PubMed ID: 21205197
[TBL] [Abstract][Full Text] [Related]
31. Thiazolone-acylsulfonamides as novel HCV NS5B polymerase allosteric inhibitors: convergence of structure-based drug design and X-ray crystallographic study.
Yan S; Appleby T; Larson G; Wu JZ; Hamatake RK; Hong Z; Yao N
Bioorg Med Chem Lett; 2007 Apr; 17(7):1991-5. PubMed ID: 17276060
[TBL] [Abstract][Full Text] [Related]
32. Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors.
Graham TH; Shu M; Verras A; Chen Q; Garcia-Calvo M; Li X; Lisnock J; Tong X; Tung EC; Wiltsie J; Hale JJ; Pinto S; Shen DM
Bioorg Med Chem Lett; 2014 Apr; 24(7):1657-60. PubMed ID: 24636945
[TBL] [Abstract][Full Text] [Related]
33. Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design.
Subbaiah MAM; Meanwell NA
J Med Chem; 2021 Oct; 64(19):14046-14128. PubMed ID: 34591488
[TBL] [Abstract][Full Text] [Related]
34. [Strategy of molecular design of drugs: the unification of macro-properties and micro-structures of a molecule].
Guo ZR
Yao Xue Xue Bao; 2008 Mar; 43(3):227-33. PubMed ID: 18630256
[TBL] [Abstract][Full Text] [Related]
35. Application of the bicyclo[1.1.1]pentane motif as a nonclassical phenyl ring bioisostere in the design of a potent and orally active γ-secretase inhibitor.
Stepan AF; Subramanyam C; Efremov IV; Dutra JK; O'Sullivan TJ; DiRico KJ; McDonald WS; Won A; Dorff PH; Nolan CE; Becker SL; Pustilnik LR; Riddell DR; Kauffman GW; Kormos BL; Zhang L; Lu Y; Capetta SH; Green ME; Karki K; Sibley E; Atchison KP; Hallgren AJ; Oborski CE; Robshaw AE; Sneed B; O'Donnell CJ
J Med Chem; 2012 Apr; 55(7):3414-24. PubMed ID: 22420884
[TBL] [Abstract][Full Text] [Related]
36. Theoretical study of gas-phase acidity, pKa, lipophilicity, and solubility of some biologically active sulfonamides.
Remko M; von der Lieth CW
Bioorg Med Chem; 2004 Oct; 12(20):5395-403. PubMed ID: 15388166
[TBL] [Abstract][Full Text] [Related]
37. O,N,N'-trialkylisoureas as mild activating reagents for N-acylsulfonamide anchors.
Zohrabi-Kalantari V; Heidler P; Larsen T; Link A
Org Lett; 2005 Dec; 7(25):5665-7. PubMed ID: 16321017
[TBL] [Abstract][Full Text] [Related]
38. Structure-activity relationships and key structural feature of pyridyloxybenzene-acylsulfonamides as new, potent, and selective peroxisome proliferator-activated receptor (PPAR) γ Agonists.
Rikimaru K; Wakabayashi T; Abe H; Tawaraishi T; Imoto H; Yonemori J; Hirose H; Murase K; Matsuo T; Matsumoto M; Nomura C; Tsuge H; Arimura N; Kawakami K; Sakamoto J; Funami M; Mol CD; Snell GP; Bragstad KA; Sang BC; Dougan DR; Tanaka T; Katayama N; Horiguchi Y; Momose Y
Bioorg Med Chem; 2012 May; 20(10):3332-58. PubMed ID: 22503460
[TBL] [Abstract][Full Text] [Related]
39. Sulfonimidamides in Medicinal and Agricultural Chemistry.
Chinthakindi PK; Naicker T; Thota N; Govender T; Kruger HG; Arvidsson PI
Angew Chem Int Ed Engl; 2017 Apr; 56(15):4100-4109. PubMed ID: 27958674
[TBL] [Abstract][Full Text] [Related]
40. Carboxylate Surrogates Enhance the Antimycobacterial Activity of UDP-Galactopyranose Mutase Probes.
Winton VJ; Aldrich C; Kiessling LL
ACS Infect Dis; 2016 Aug; 2(8):538-43. PubMed ID: 27626294
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
