BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

164 related articles for article (PubMed ID: 34082225)

  • 1. Thiophene-2-carboxamide derivatives of anthraquinone: A new potent antitumor chemotype.
    Volodina YL; Tikhomirov AS; Dezhenkova LG; Ramonova AA; Kononova AV; Andreeva DV; Kaluzhny DN; Schols D; Moisenovich MM; Shchekotikhin AE; Shtil AA
    Eur J Med Chem; 2021 Oct; 221():113521. PubMed ID: 34082225
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Amides of pyrrole- and thiophene-fused anthraquinone derivatives: A role of the heterocyclic core in antitumor properties.
    Tikhomirov AS; Litvinova VA; Andreeva DV; Tsvetkov VB; Dezhenkova LG; Volodina YL; Kaluzhny DN; Treshalin ID; Schols D; Ramonova AA; Moisenovich MM; Shtil AA; Shchekotikhin AE
    Eur J Med Chem; 2020 Aug; 199():112294. PubMed ID: 32428792
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New antitumor anthra[2,3-b]furan-3-carboxamides: Synthesis and structure-activity relationship.
    Tikhomirov AS; Lin CY; Volodina YL; Dezhenkova LG; Tatarskiy VV; Schols D; Shtil AA; Kaur P; Chueh PJ; Shchekotikhin AE
    Eur J Med Chem; 2018 Mar; 148():128-139. PubMed ID: 29459273
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 5-Nitro-Thiophene-Thiosemicarbazone Derivatives Present Antitumor Activity Mediated by Apoptosis and DNA Intercalation.
    Roque Marques KM; do Desterro MR; de Arruda SM; de Araújo Neto LN; do Carmo Alves de Lima M; de Almeida SMV; da Silva ECD; de Aquino TM; da Silva-Júnior EF; de Araújo-Júnior JX; de M Silva M; de A Dantas MD; Santos JCC; Figueiredo IM; Bazin MA; Marchand P; da Silva TG; Mendonça Junior FJB
    Curr Top Med Chem; 2019; 19(13):1075-1091. PubMed ID: 31223089
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Concise synthesis and biological evaluation of 2-Aryl-3-Anilinobenzo[b]thiophene derivatives as potent apoptosis-inducing agents.
    Romagnoli R; Preti D; Hamel E; Bortolozzi R; Viola G; Brancale A; Ferla S; Morciano G; Pinton P
    Bioorg Chem; 2021 Jul; 112():104919. PubMed ID: 33957538
    [TBL] [Abstract][Full Text] [Related]  

  • 6. New anthra[2,3-b]furancarboxamides: A role of positioning of the carboxamide moiety in antitumor properties.
    Volodina YL; Dezhenkova LG; Tikhomirov AS; Tatarskiy VV; Kaluzhny DN; Moisenovich AM; Moisenovich MM; Isagulieva AK; Shtil AA; Tsvetkov VB; Shchekotikhin AE
    Eur J Med Chem; 2019 Mar; 165():31-45. PubMed ID: 30659997
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents.
    Romagnoli R; Baraldi PG; Lopez-Cara C; Salvador MK; Preti D; Tabrizi MA; Balzarini J; Nussbaumer P; Bassetto M; Brancale A; Fu XH; Yang-Gao ; Li J; Zhang SZ; Hamel E; Bortolozzi R; Basso G; Viola G
    Bioorg Med Chem; 2014 Sep; 22(18):5097-109. PubMed ID: 24398384
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Discovery of antitumor anthra[2,3-b]furan-3-carboxamides: Optimization of synthesis and evaluation of antitumor properties.
    Shchekotikhin AE; Dezhenkova LG; Tsvetkov VB; Luzikov YN; Volodina YL; Tatarskiy VV; Kalinina AA; Treshalin MI; Treshalina HM; Romanenko VI; Kaluzhny DN; Kubbutat M; Schols D; Pommier Y; Shtil AA; Preobrazhenskaya MN
    Eur J Med Chem; 2016 Apr; 112():114-129. PubMed ID: 26890118
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel Tetrahydrobenzo [b] Thiophene Compounds Exhibit Anticancer Activity through Enhancing Apoptosis and Inhibiting Tyrosine Kinase.
    El-Metwally SA; Khalil AK; El-Naggar AM; El-Sayed WM
    Anticancer Agents Med Chem; 2018; 18(12):1761-1769. PubMed ID: 30101717
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Annulation of substituted anthracene-9,10-diones yields promising selectively antiproliferative compounds.
    Castro-Castillo V; Suárez-Rozas C; Castro-Loiza N; Theoduloz C; Cassels BK
    Eur J Med Chem; 2013 Apr; 62():688-92. PubMed ID: 23454511
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Heterocyclic ring expansion yields anthraquinone derivatives potent against multidrug resistant tumor cells.
    Tikhomirov AS; Tsvetkov VB; Volodina YL; Litvinova VA; Andreeva DV; Dezhenkova LG; Kaluzhny DN; Treshalin ID; Shtil AA; Shchekotikhin AE
    Bioorg Chem; 2022 Oct; 127():105925. PubMed ID: 35728293
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and cytotoxic effect of 1,3-dihydroxy-9,10-anthraquinone derivatives.
    Wei BL; Wu SH; Chung MI; Won SJ; Lin CN
    Eur J Med Chem; 2000 Dec; 35(12):1089-98. PubMed ID: 11248407
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Upregulation of p53 through induction of MDM2 degradation: Anthraquinone analogs.
    Draganov AB; Yang X; Anifowose A; De La Cruz LKC; Dai C; Ni N; Chen W; De Los Santos Z; Gu L; Zhou M; Wang B
    Bioorg Med Chem; 2019 Sep; 27(17):3860-3865. PubMed ID: 31324563
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Novel multi-targeting anthra[2,3-b]thiophene-5,10-diones with guanidine-containing side chains: interaction with telomeric G-quadruplex, inhibition of telomerase and topoisomerase I and cytotoxic properties.
    Ilyinsky NS; Shchyolkina AK; Borisova OF; Mamaeva OK; Zvereva MI; Azhibek DM; Livshits MA; Mitkevich VA; Balzarini J; Sinkevich YB; Luzikov YN; Dezhenkova LG; Kolotova ES; Shtil AA; Shchekotikhin AE; Kaluzhny DN
    Eur J Med Chem; 2014 Oct; 85():605-14. PubMed ID: 25127152
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and biological evaluation of 2-(3',4',5'-trimethoxybenzoyl)-3-aryl/arylaminobenzo[b]thiophene derivatives as a novel class of antiproliferative agents.
    Romagnoli R; Baraldi PG; Cara CL; Hamel E; Basso G; Bortolozzi R; Viola G
    Eur J Med Chem; 2010 Dec; 45(12):5781-91. PubMed ID: 20933308
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of thiophene-thiosemicarbazone derivatives and evaluation of their in vitro and in vivo antitumor activities.
    de Oliveira JF; da Silva AL; Vendramini-Costa DB; da Cruz Amorim CA; Campos JF; Ribeiro AG; Olímpio de Moura R; Neves JL; Ruiz AL; Ernesto de Carvalho J; Alves de Lima Mdo C
    Eur J Med Chem; 2015 Nov; 104():148-56. PubMed ID: 26454648
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition.
    Romagnoli R; Kimatrai Salvador M; Schiaffino Ortega S; Baraldi PG; Oliva P; Baraldi S; Lopez-Cara LC; Brancale A; Ferla S; Hamel E; Balzarini J; Liekens S; Mattiuzzo E; Basso G; Viola G
    Eur J Med Chem; 2018 Jan; 143():683-698. PubMed ID: 29220790
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design, synthesis and cytotoxic effect of hydroxy- and 3-alkylaminopropoxy-9,10-anthraquinone derivatives.
    Teng CH; Won SJ; Lin CN
    Bioorg Med Chem; 2005 May; 13(10):3439-45. PubMed ID: 15848756
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis, antitumor screening and cell cycle analysis of novel benzothieno[3,2-b]pyran derivatives.
    Zaher AF; Abuel-Maaty SM; El-Nassan HB; Amer SA; Abdelghany TM
    J Enzyme Inhib Med Chem; 2016; 31(sup4):145-153. PubMed ID: 27590401
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis of novel bis-anthraquinone derivatives and their biological evaluation as antitumor agents.
    Taher AT; Hegazy GH
    Arch Pharm Res; 2013 May; 36(5):573-8. PubMed ID: 23471561
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.