These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
7. Covalent Stapling of the Cereblon Sensor Loop Histidine Using Sulfur-Heterocycle Exchange. Cruite JT; Nowak RP; Donovan KA; Ficarro SB; Huang H; Liu H; Liu Y; Marto JA; Metivier RJ; Fischer ES; Jones LH ACS Med Chem Lett; 2023 Nov; 14(11):1576-1581. PubMed ID: 37974938 [TBL] [Abstract][Full Text] [Related]
8. Arylfluorosulfate-Based Electrophiles for Covalent Protein Labeling: A New Addition to the Arsenal. Martín-Gago P; Olsen CA Angew Chem Int Ed Engl; 2019 Jan; 58(4):957-966. PubMed ID: 30024079 [TBL] [Abstract][Full Text] [Related]
9. Systems analysis of protein modification and cellular responses induced by electrophile stress. Jacobs AT; Marnett LJ Acc Chem Res; 2010 May; 43(5):673-83. PubMed ID: 20218676 [TBL] [Abstract][Full Text] [Related]
10. Covalent drug discovery using sulfur(VI) fluoride exchange warheads. Huang H; Jones LH Expert Opin Drug Discov; 2023 Jul; 18(7):725-735. PubMed ID: 37243622 [TBL] [Abstract][Full Text] [Related]
11. Introducing A New Class of Sulfonyl Fluoride Hubs via Radical Chloro-Fluorosulfonylation of Alkynes. Nie X; Xu T; Hong Y; Zhang H; Mao C; Liao S Angew Chem Int Ed Engl; 2021 Sep; 60(40):22035-22042. PubMed ID: 34382306 [TBL] [Abstract][Full Text] [Related]
12. Direct Target Site Identification of a Sulfonyl-Triazole Covalent Kinase Probe by LC-MS Chemical Proteomics. McCloud RL; Yuan K; Mahoney KE; Bai DL; Shabanowitz J; Ross MM; Hunt DF; Hsu KL Anal Chem; 2021 Sep; 93(35):11946-11955. PubMed ID: 34431655 [TBL] [Abstract][Full Text] [Related]
13. Reactions of electrophiles with nucleophilic thiolate sites: relevance to pathophysiological mechanisms and remediation. LoPachin RM; Gavin T Free Radic Res; 2016; 50(2):195-205. PubMed ID: 26559119 [TBL] [Abstract][Full Text] [Related]
14. Using sulfuramidimidoyl fluorides that undergo sulfur(VI) fluoride exchange for inverse drug discovery. Brighty GJ; Botham RC; Li S; Nelson L; Mortenson DE; Li G; Morisseau C; Wang H; Hammock BD; Sharpless KB; Kelly JW Nat Chem; 2020 Oct; 12(10):906-913. PubMed ID: 32868886 [TBL] [Abstract][Full Text] [Related]
15. Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry. Dong J; Krasnova L; Finn MG; Sharpless KB Angew Chem Int Ed Engl; 2014 Sep; 53(36):9430-48. PubMed ID: 25112519 [TBL] [Abstract][Full Text] [Related]
16. Covalent drugs targeting histidine - an unexploited opportunity? Che J; Jones LH RSC Med Chem; 2022 Oct; 13(10):1121-1126. PubMed ID: 36325394 [TBL] [Abstract][Full Text] [Related]
17. Chemical and biology of sulfur fluoride exchange (SuFEx) click chemistry for drug discovery. Wilson Lucas S; Zijian Qin R; Rakesh KP; Sharath Kumar KS; Qin HL Bioorg Chem; 2023 Jan; 130():106227. PubMed ID: 36368173 [TBL] [Abstract][Full Text] [Related]
18. Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue. Fadeyi OO; Hoth LR; Choi C; Feng X; Gopalsamy A; Hett EC; Kyne RE; Robinson RP; Jones LH ACS Chem Biol; 2017 Aug; 12(8):2015-2020. PubMed ID: 28718624 [TBL] [Abstract][Full Text] [Related]