BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

141 related articles for article (PubMed ID: 34218000)

  • 1. Synthesis, bioevaluation and docking studies of new imidamide derivatives as nitric oxide synthase inhibitors.
    Arias F; Franco-Montalban F; Romero M; Carrión MD; Camacho ME
    Bioorg Med Chem; 2021 Aug; 44():116294. PubMed ID: 34218000
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Development of urea and thiourea kynurenamine derivatives: synthesis, molecular modeling, and biological evaluation as nitric oxide synthase inhibitors.
    Chayah M; Carrión MD; Gallo MA; Jiménez R; Duarte J; Camacho ME
    ChemMedChem; 2015 May; 10(5):874-82. PubMed ID: 25801086
    [TBL] [Abstract][Full Text] [Related]  

  • 3. 1,3,4-Thiadiazole derivatives as selective inhibitors of iNOS versus nNOS: Synthesis and structure-activity dependence.
    López-Cara LC; Carrión MD; Entrena A; Gallo MA; Espinosa A; López A; Escames G; Acuña-Castroviejo D; Camacho ME
    Eur J Med Chem; 2012 Apr; 50():129-39. PubMed ID: 22336385
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Phenylpyrrole derivatives as neural and inducible nitric oxide synthase (nNOS and iNOS) inhibitors.
    López Cara LC; Camacho ME; Carrión MD; Tapias V; Gallo MA; Escames G; Acuña-Castroviejo D; Espinosa A; Entrena A
    Eur J Med Chem; 2009 Jun; 44(6):2655-66. PubMed ID: 19117642
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and biological evaluation of 4,5-dihydro-1H-pyrazole derivatives as potential nNOS/iNOS selective inhibitors. Part 2: Influence of diverse substituents in both the phenyl moiety and the acyl group.
    Carrión MD; Chayah M; Entrena A; López A; Gallo MA; Acuña-Castroviejo D; Camacho ME
    Bioorg Med Chem; 2013 Jul; 21(14):4132-42. PubMed ID: 23735830
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Discovery of a series of aminopiperidines as novel iNOS inhibitors.
    Le Bourdonnec B; Leister LK; Ajello CA; Cassel JA; Seida PR; O'Hare H; Gu M; Chu GH; Tuthill PA; DeHaven RN; Dolle RE
    Bioorg Med Chem Lett; 2008 Jan; 18(1):336-43. PubMed ID: 18024030
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Pyrazoles and pyrazolines as neural and inducible nitric oxide synthase (nNOS and iNOS) potential inhibitors (III).
    Carrión MD; López Cara LC; Camacho ME; Tapias V; Escames G; Acuña-Castroviejo D; Espinosa A; Gallo MA; Entrena A
    Eur J Med Chem; 2008 Nov; 43(11):2579-91. PubMed ID: 18325637
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Bioactive imidamide-based compounds targeted against nitric oxide synthase.
    Arias F; Franco-Montalban F; Romero M; Duarte J; Dora Carrión M; Encarnación Camacho M
    Bioorg Chem; 2022 Mar; 120():105637. PubMed ID: 35131617
    [TBL] [Abstract][Full Text] [Related]  

  • 9. N-Phenylamidines as selective inhibitors of human neuronal nitric oxide synthase: structure-activity studies and demonstration of in vivo activity.
    Collins JL; Shearer BG; Oplinger JA; Lee S; Garvey EP; Salter M; Duffy C; Burnette TC; Furfine ES
    J Med Chem; 1998 Jul; 41(15):2858-71. PubMed ID: 9667974
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Phenyl Ether- and Aniline-Containing 2-Aminoquinolines as Potent and Selective Inhibitors of Neuronal Nitric Oxide Synthase.
    Cinelli MA; Li H; Pensa AV; Kang S; Roman LJ; Martásek P; Poulos TL; Silverman RB
    J Med Chem; 2015 Nov; 58(21):8694-712. PubMed ID: 26469213
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Chiral linkers to improve selectivity of double-headed neuronal nitric oxide synthase inhibitors.
    Jing Q; Li H; Chreifi G; Roman LJ; Martásek P; Poulos TL; Silverman RB
    Bioorg Med Chem Lett; 2013 Oct; 23(20):5674-9. PubMed ID: 23993333
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Heteroalicyclic carboxamidines as inhibitors of inducible nitric oxide synthase; the identification of (2R)-2-pyrrolidinecarboxamidine as a potent and selective haem-co-ordinating inhibitor.
    Young RJ; Alderton W; Angell AD; Beswick PJ; Brown D; Chambers CL; Crowe MC; Dawson J; Hamlett CC; Hodgson ST; Kleanthous S; Knowles RG; Russell LJ; Stocker R; Woolven JM
    Bioorg Med Chem Lett; 2011 May; 21(10):3037-40. PubMed ID: 21482467
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Screening of novel and selective inhibitors for neuronal nitric oxide synthase (nNOS) via structure-based drug design techniques.
    Boumezber S; Yelekçi K
    J Biomol Struct Dyn; 2023 May; 41(8):3607-3629. PubMed ID: 35322764
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Contribution of nitric oxide synthase isoforms to cholinergic vasodilation in murine retinal arterioles.
    Gericke A; Goloborodko E; Sniatecki JJ; Steege A; Wojnowski L; Pfeiffer N
    Exp Eye Res; 2013 Apr; 109():60-6. PubMed ID: 23434456
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Potent and selective double-headed thiophene-2-carboximidamide inhibitors of neuronal nitric oxide synthase for the treatment of melanoma.
    Huang H; Li H; Yang S; Chreifi G; Martásek P; Roman LJ; Meyskens FL; Poulos TL; Silverman RB
    J Med Chem; 2014 Feb; 57(3):686-700. PubMed ID: 24447275
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Discovery of N-{3-[(ethanimidoylamino)methyl]benzyl}-l-prolinamide dihydrochloride: A new potent and selective inhibitor of the inducible nitric oxide synthase as a promising agent for the therapy of malignant glioma.
    Maccallini C; Di Matteo M; Gallorini M; Montagnani M; Graziani V; Ammazzalorso A; Amoia P; De Filippis B; Di Silvestre S; Fantacuzzi M; Giampietro L; Potenza MA; Re N; Pandolfi A; Cataldi A; Amoroso R
    Eur J Med Chem; 2018 May; 152():53-64. PubMed ID: 29689474
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 1,5-Disubstituted indole derivatives as selective human neuronal nitric oxide synthase inhibitors.
    Renton P; Speed J; Maddaford S; Annedi SC; Ramnauth J; Rakhit S; Andrews J
    Bioorg Med Chem Lett; 2011 Sep; 21(18):5301-4. PubMed ID: 21813276
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and biological evaluation of indazole derivatives.
    Claramunt RM; López C; López A; Pérez-Medina C; Pérez-Torralba M; Alkorta I; Elguero J; Escames G; Acuña-Castroviejo D
    Eur J Med Chem; 2011 Apr; 46(4):1439-47. PubMed ID: 21334118
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis, biological evaluation, and docking studies of N-substituted acetamidines as selective inhibitors of inducible nitric oxide synthase.
    Maccallini C; Patruno A; Besker N; Alì JI; Ammazzalorso A; De Filippis B; Franceschelli S; Giampietro L; Pesce M; Reale M; Tricca ML; Re N; Felaco M; Amoroso R
    J Med Chem; 2009 Mar; 52(5):1481-5. PubMed ID: 19203270
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Insights into the structural determinants for selective inhibition of nitric oxide synthase isoforms.
    Oliveira BL; Moreira IS; Fernandes PA; Ramos MJ; Santos I; Correia JD
    J Mol Model; 2013 Apr; 19(4):1537-51. PubMed ID: 23263357
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.