BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

140 related articles for article (PubMed ID: 34313342)

  • 1. Nanomolar potency of imidazo[2,1-b]thiazole analogs as indoleamine 2,3-dioxygenase inhibitors.
    Ewida MA; Ewida HA; Ahmed MS; Allam HA; ElBagary RI; George RF; Georgey HH; El-Subbagh HI
    Arch Pharm (Weinheim); 2021 Nov; 354(11):e2100202. PubMed ID: 34313342
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of Benzo[d]imidazo[2,1-b]thiazole-Propenone Conjugates as Cytotoxic and Apoptotic Inducing Agents.
    Shaik SP; Reddy TS; Sunkari S; Rao AVS; Babu KS; Bhargava SK; Kamal A
    Anticancer Agents Med Chem; 2019; 19(3):347-355. PubMed ID: 30479221
    [TBL] [Abstract][Full Text] [Related]  

  • 3. 3-Methyl-imidazo[2,1-b]thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations.
    Ewida MA; Ewida HA; Ahmed MS; Allam HA; ElBagary RI; George RF; Georgey HH; El-Subbagh HI
    Bioorg Chem; 2021 Oct; 115():105205. PubMed ID: 34329992
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and biological evaluation of imidazo[2,1-b]thiazole-benzimidazole conjugates as microtubule-targeting agents.
    Baig MF; Nayak VL; Budaganaboyina P; Mullagiri K; Sunkari S; Gour J; Kamal A
    Bioorg Chem; 2018 Apr; 77():515-526. PubMed ID: 29459129
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors.
    Serafini M; Torre E; Aprile S; Massarotti A; Fallarini S; Pirali T
    Molecules; 2019 May; 24(10):. PubMed ID: 31096672
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Unique Sulfur-Aromatic Interactions Contribute to the Binding of Potent Imidazothiazole Indoleamine 2,3-Dioxygenase Inhibitors.
    Peng YH; Liao FY; Tseng CT; Kuppusamy R; Li AS; Chen CH; Fan YS; Wang SY; Wu MH; Hsueh CC; Chang JY; Lee LC; Shih C; Shia KS; Yeh TK; Hung MS; Kuo CC; Song JS; Wu SY; Ueng SH
    J Med Chem; 2020 Feb; 63(4):1642-1659. PubMed ID: 31961685
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design and synthesis of 1,2,3-triazolo linked benzo[d]imidazo[2,1-b]thiazole conjugates as tubulin polymerization inhibitors.
    Shaik SP; Vishnuvardhan MVPS; Sultana F; Subba Rao AV; Bagul C; Bhattacharjee D; Kapure JS; Jain N; Kamal A
    Bioorg Med Chem; 2017 Jul; 25(13):3285-3297. PubMed ID: 28462842
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies.
    Griglio A; Torre E; Serafini M; Bianchi A; Schmid R; Coda Zabetta G; Massarotti A; Sorba G; Pirali T; Fallarini S
    Bioorg Med Chem Lett; 2018 Feb; 28(4):651-657. PubMed ID: 29398544
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis and biological evaluation of imidazo[2,1-b]thiazole and benzo[d]imidazo[2,1-b]thiazole derivatives as Mycobacterium tuberculosis pantothenate synthetase inhibitors.
    Samala G; Devi PB; Saxena S; Meda N; Yogeeswari P; Sriram D
    Bioorg Med Chem; 2016 Mar; 24(6):1298-307. PubMed ID: 26867485
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Harmine-inspired design and synthesis of benzo[d]imidazo[2,1-b]thiazole derivatives bearing 1,3,4-oxadiazole moiety as potential tumor suppressors.
    Zhao T; Yang Y; Yang J; Cui Y; Cao Z; Zuo D; Zhai X
    Bioorg Med Chem; 2021 Sep; 46():116367. PubMed ID: 34425477
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of benzo[d]imidazo[2,1-b]thiazole-chalcone conjugates as microtubule targeting and apoptosis inducing agents.
    Sultana F; Reddy Bonam S; Reddy VG; Nayak VL; Akunuri R; Rani Routhu S; Alarifi A; Halmuthur MSK; Kamal A
    Bioorg Chem; 2018 Feb; 76():1-12. PubMed ID: 29102724
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and Antitumor Activity of New Thiazole Nortopsentin Analogs.
    Spanò V; Attanzio A; Cascioferro S; Carbone A; Montalbano A; Barraja P; Tesoriere L; Cirrincione G; Diana P; Parrino B
    Mar Drugs; 2016 Dec; 14(12):. PubMed ID: 27983614
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Potential antitumor agents. 37. Synthesis and antitumor activity of guanylhydrazones from imidazo[2,1-b]thiazoles and from the new heterocyclic system thiazolo[2',3':2,3]imidazo[4,5-c]quinoline.
    Andreani A; Granaiola M; Leoni A; Locatelli A; Morigi R; Rambaldi M; Lenaz G; Fato R; Bergamini C; Farruggia G
    J Med Chem; 2005 Apr; 48(8):3085-9. PubMed ID: 15828848
    [TBL] [Abstract][Full Text] [Related]  

  • 14. New imidazo[2,1-b]thiazole derivatives: synthesis, in vitro anticancer evaluation, and in silico studies.
    Park JH; El-Gamal MI; Lee YS; Oh CH
    Eur J Med Chem; 2011 Dec; 46(12):5769-77. PubMed ID: 22033063
    [TBL] [Abstract][Full Text] [Related]  

  • 15. New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues.
    Andreani A; Burnelli S; Granaiola M; Leoni A; Locatelli A; Morigi R; Rambaldi M; Varoli L; Calonghi N; Cappadone C; Farruggia G; Zini M; Stefanelli C; Masotti L; Radin NS; Shoemaker RH
    J Med Chem; 2008 Feb; 51(4):809-16. PubMed ID: 18251494
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, in vitro anticancer evaluation and in silico studies of novel imidazo[2,1-b]thiazole derivatives bearing pyrazole moieties.
    Ali AR; El-Bendary ER; Ghaly MA; Shehata IA
    Eur J Med Chem; 2014 Mar; 75():492-500. PubMed ID: 24576591
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Design, synthesis and antiproliferative activity of novel heterobivalent hybrids based on imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b][1,3]thiazole scaffolds.
    Romagnoli R; Baraldi PG; Prencipe F; Balzarini J; Liekens S; Estévez F
    Eur J Med Chem; 2015 Aug; 101():205-17. PubMed ID: 26141911
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design and synthesis of imidazo[2,1-b]thiazole linked triazole conjugates: Microtubule-destabilizing agents.
    Shaik SP; Nayak VL; Sultana F; Rao AVS; Shaik AB; Babu KS; Kamal A
    Eur J Med Chem; 2017 Jan; 126():36-51. PubMed ID: 27744185
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis of imidazothiazole-chalcone derivatives as anticancer and apoptosis inducing agents.
    Kamal A; Dastagiri D; Ramaiah MJ; Reddy JS; Bharathi EV; Srinivas C; Pushpavalli SN; Pal D; Pal-Bhadra M
    ChemMedChem; 2010 Nov; 5(11):1937-47. PubMed ID: 20836120
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design and Synthesis of Indoleamine 2,3-Dioxygenase 1 Inhibitors and Evaluation of Their Use as Anti-Tumor Agents.
    Wen H; Liu Y; Wang S; Wang T; Zhang G; Chen X; Li Y; Cui H; Lai F; Sheng L
    Molecules; 2019 Jun; 24(11):. PubMed ID: 31195673
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.