184 related articles for article (PubMed ID: 34339714)
1. Insights into agonist-elicited activation of the human glucose-dependent insulinotropic polypeptide receptor.
Yuliantie E; van der Velden WJC; Labroska V; Dai A; Zhao F; Darbalaei S; Deganutti G; Xu T; Zhou Q; Yang D; Rosenkilde MM; Sexton PM; Wang MW; Wootten D
Biochem Pharmacol; 2021 Oct; 192():114715. PubMed ID: 34339714
[TBL] [Abstract][Full Text] [Related]
2. Human GIP(3-30)NH
Gabe MBN; Sparre-Ulrich AH; Pedersen MF; Gasbjerg LS; Inoue A; Bräuner-Osborne H; Hartmann B; Rosenkilde MM
Biochem Pharmacol; 2018 Apr; 150():97-107. PubMed ID: 29378179
[TBL] [Abstract][Full Text] [Related]
3. Pharmacological characterization of mono-, dual- and tri-peptidic agonists at GIP and GLP-1 receptors.
Yuliantie E; Darbalaei S; Dai A; Zhao P; Yang D; Sexton PM; Wang MW; Wootten D
Biochem Pharmacol; 2020 Jul; 177():114001. PubMed ID: 32360365
[TBL] [Abstract][Full Text] [Related]
4. Molecular basis of signal transduction mediated by the human GIPR splice variants.
Zhao F; Hang K; Zhou Q; Shao L; Li H; Li W; Lin S; Dai A; Cai X; Liu Y; Xu Y; Feng W; Yang D; Wang MW
Proc Natl Acad Sci U S A; 2023 Oct; 120(41):e2306145120. PubMed ID: 37792509
[TBL] [Abstract][Full Text] [Related]
5. Genetic and biased agonist-mediated reductions in β-arrestin recruitment prolong cAMP signaling at glucagon family receptors.
Jones B; McGlone ER; Fang Z; Pickford P; Corrêa IR; Oishi A; Jockers R; Inoue A; Kumar S; Görlitz F; Dunsby C; French PMW; Rutter GA; Tan T; Tomas A; Bloom SR
J Biol Chem; 2021; 296():100133. PubMed ID: 33268378
[TBL] [Abstract][Full Text] [Related]
6. Investigating GIPR (ant)agonism: A structural analysis of GIP and its receptor.
Smit FX; van der Velden WJC; Kizilkaya HS; Nørskov A; Lückmann M; Hansen TN; Sparre-Ulrich AH; Qvotrup K; Frimurer TM; Rosenkilde MM
Structure; 2021 Jul; 29(7):679-693.e6. PubMed ID: 33891864
[TBL] [Abstract][Full Text] [Related]
7. Identification of determinants of glucose-dependent insulinotropic polypeptide receptor that interact with N-terminal biologically active region of the natural ligand.
Yaqub T; Tikhonova IG; Lättig J; Magnan R; Laval M; Escrieut C; Boulègue C; Hewage C; Fourmy D
Mol Pharmacol; 2010 Apr; 77(4):547-58. PubMed ID: 20061446
[TBL] [Abstract][Full Text] [Related]
8. Tyr1 and Ile7 of glucose-dependent insulinotropic polypeptide (GIP) confer differential ligand selectivity toward GIP and glucagon-like peptide-1 receptors.
Moon MJ; Kim HY; Kim SG; Park J; Choi DS; Hwang JI; Seong JY
Mol Cells; 2010 Aug; 30(2):149-54. PubMed ID: 20799012
[TBL] [Abstract][Full Text] [Related]
9. Functional elements of the gastric inhibitory polypeptide receptor: Comparison between secretin- and rhodopsin-like G protein-coupled receptors.
Cordomí A; Ismail S; Matsoukas MT; Escrieut C; Gherardi MJ; Pardo L; Fourmy D
Biochem Pharmacol; 2015 Aug; 96(3):237-46. PubMed ID: 26043830
[TBL] [Abstract][Full Text] [Related]
10. Structural and pharmacological characterization of novel potent and selective monoclonal antibody antagonists of glucose-dependent insulinotropic polypeptide receptor.
Ravn P; Madhurantakam C; Kunze S; Matthews E; Priest C; O'Brien S; Collinson A; Papworth M; Fritsch-Fredin M; Jermutus L; Benthem L; Gruetter M; Jackson RH
J Biol Chem; 2013 Jul; 288(27):19760-72. PubMed ID: 23689510
[TBL] [Abstract][Full Text] [Related]
11. Internalized Receptor for Glucose-dependent Insulinotropic Peptide stimulates adenylyl cyclase on early endosomes.
Ismail S; Gherardi MJ; Froese A; Zanoun M; Gigoux V; Clerc P; Gaits-Iacovoni F; Steyaert J; Nikolaev VO; Fourmy D
Biochem Pharmacol; 2016 Nov; 120():33-45. PubMed ID: 27641811
[TBL] [Abstract][Full Text] [Related]
12. Understanding interactions of gastric inhibitory polypeptide (GIP) with its G-protein coupled receptor through NMR and molecular modeling.
Malde AK; Srivastava SS; Coutinho EC
J Pept Sci; 2007 May; 13(5):287-300. PubMed ID: 17437246
[TBL] [Abstract][Full Text] [Related]
13. Internalization and desensitization of the human glucose-dependent-insulinotropic receptor is affected by N-terminal acetylation of the agonist.
Ismail S; Dubois-Vedrenne I; Laval M; Tikhonova IG; D'Angelo R; Sanchez C; Clerc P; Gherardi MJ; Gigoux V; Magnan R; Fourmy D
Mol Cell Endocrinol; 2015 Oct; 414():202-15. PubMed ID: 26225752
[TBL] [Abstract][Full Text] [Related]
14. Structural insights into hormone recognition by the human glucose-dependent insulinotropic polypeptide receptor.
Zhao F; Zhang C; Zhou Q; Hang K; Zou X; Chen Y; Wu F; Rao Q; Dai A; Yin W; Shen DD; Zhang Y; Xia T; Stevens RC; Xu HE; Yang D; Zhao L; Wang MW
Elife; 2021 Jul; 10():. PubMed ID: 34254582
[TBL] [Abstract][Full Text] [Related]
15. The GIP receptor displays higher basal activity than the GLP-1 receptor but does not recruit GRK2 or arrestin3 effectively.
Al-Sabah S; Al-Fulaij M; Shaaban G; Ahmed HA; Mann RJ; Donnelly D; Bünemann M; Krasel C
PLoS One; 2014; 9(9):e106890. PubMed ID: 25191754
[TBL] [Abstract][Full Text] [Related]
16. Downregulation of a GPCR by β-Arrestin2-Mediated Switch from an Endosomal to a TGN Recycling Pathway.
Abdullah N; Beg M; Soares D; Dittman JS; McGraw TE
Cell Rep; 2016 Dec; 17(11):2966-2978. PubMed ID: 27974210
[TBL] [Abstract][Full Text] [Related]
17. Mapping interactions of gastric inhibitory polypeptide with GIPR N-terminus using NMR and molecular dynamics simulations.
Tikhele SH; Pissurlenkar RR; Srivastava S; Saran A; Coutinho EC
J Pept Sci; 2010 Aug; 16(8):383-91. PubMed ID: 20607844
[TBL] [Abstract][Full Text] [Related]
18. Conformational, receptor interaction and alanine scan studies of glucose-dependent insulinotropic polypeptide.
Venneti KC; Malthouse JP; O'Harte FP; Hewage CM
Biochim Biophys Acta; 2011 Jul; 1814(7):882-8. PubMed ID: 21539943
[TBL] [Abstract][Full Text] [Related]
19. Enhanced agonist residence time, internalization rate and signalling of the GIP receptor variant [E354Q] facilitate receptor desensitization and long-term impairment of the GIP system.
Gabe MBN; van der Velden WJC; Gadgaard S; Smit FX; Hartmann B; Bräuner-Osborne H; Rosenkilde MM
Basic Clin Pharmacol Toxicol; 2020 Jun; 126 Suppl 6(Suppl 6):122-132. PubMed ID: 31299132
[TBL] [Abstract][Full Text] [Related]
20. Localization of the domains involved in ligand binding and activation of the glucose-dependent insulinotropic polypeptide receptor.
Gelling RW; Wheeler MB; Xue J; Gyomorey S; Nian C; Pederson RA; McIntosh CH
Endocrinology; 1997 Jun; 138(6):2640-3. PubMed ID: 9165060
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]