These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
4. TROPION-Breast01: Datopotamab deruxtecan vs chemotherapy in pre-treated inoperable or metastatic HR+/HER2- breast cancer. Bardia A; Jhaveri K; Kalinsky K; Pernas S; Tsurutani J; Xu B; Hamilton E; Im SA; Nowecki Z; Sohn J; Laurentiis M; Jañez NM; Adamo B; Lee KS; Jung KH; Rubovszky G; Tseng LM; Lu YS; Yuan Y; Maxwell MJ; Haddad V; Khan SS; Rugo HS; Pistilli B Future Oncol; 2024 Mar; 20(8):423-436. PubMed ID: 37387213 [TBL] [Abstract][Full Text] [Related]
5. TROPION-Lung08: phase III study of datopotamab deruxtecan plus pembrolizumab as first-line therapy for advanced NSCLC. Levy BP; Felip E; Reck M; Yang JC; Cappuzzo F; Yoneshima Y; Zhou C; Rawat S; Xie J; Basak P; Xu L; Sands J Future Oncol; 2023 Jul; 19(21):1461-1472. PubMed ID: 37249038 [TBL] [Abstract][Full Text] [Related]
6. DS-7300a, a DNA Topoisomerase I Inhibitor, DXd-Based Antibody-Drug Conjugate Targeting B7-H3, Exerts Potent Antitumor Activities in Preclinical Models. Yamato M; Hasegawa J; Maejima T; Hattori C; Kumagai K; Watanabe A; Nishiya Y; Shibutani T; Aida T; Hayakawa I; Nakada T; Abe Y; Agatsuma T Mol Cancer Ther; 2022 Apr; 21(4):635-646. PubMed ID: 35149548 [TBL] [Abstract][Full Text] [Related]
7. TROPION-Breast03: a randomized phase III global trial of datopotamab deruxtecan ± durvalumab in patients with triple-negative breast cancer and residual invasive disease at surgical resection after neoadjuvant therapy. Bardia A; Pusztai L; Albain K; Ciruelos EM; Im SA; Hershman D; Kalinsky K; Isaacs C; Loirat D; Testa L; Tokunaga E; Wu J; Dry H; Barlow W; Kozarski R; Maxwell M; Harbeck N; Sharma P Ther Adv Med Oncol; 2024; 16():17588359241248336. PubMed ID: 38686016 [TBL] [Abstract][Full Text] [Related]
8. A Novel HER3-Targeting Antibody-Drug Conjugate, U3-1402, Exhibits Potent Therapeutic Efficacy through the Delivery of Cytotoxic Payload by Efficient Internalization. Hashimoto Y; Koyama K; Kamai Y; Hirotani K; Ogitani Y; Zembutsu A; Abe M; Kaneda Y; Maeda N; Shiose Y; Iguchi T; Ishizaka T; Karibe T; Hayakawa I; Morita K; Nakada T; Nomura T; Wakita K; Kagari T; Abe Y; Murakami M; Ueno S; Agatsuma T Clin Cancer Res; 2019 Dec; 25(23):7151-7161. PubMed ID: 31471314 [TBL] [Abstract][Full Text] [Related]
9. Raludotatug Deruxtecan, a CDH6-Targeting Antibody-Drug Conjugate with a DNA Topoisomerase I Inhibitor DXd, Is Efficacious in Human Ovarian and Kidney Cancer Models. Suzuki H; Nagase S; Saito C; Takatsuka A; Nagata M; Honda K; Kaneda Y; Nishiya Y; Honda T; Ishizaka T; Nakamura K; Nakada T; Abe Y; Agatsuma T Mol Cancer Ther; 2024 Mar; 23(3):257-271. PubMed ID: 38205802 [TBL] [Abstract][Full Text] [Related]
10. Clinical management, monitoring, and prophylaxis of adverse events of special interest associated with datopotamab deruxtecan. Heist RS; Sands J; Bardia A; Shimizu T; Lisberg A; Krop I; Yamamoto N; Kogawa T; Al-Hashimi S; Fung SSM; Galor A; Pisetzky F; Basak P; Lau C; Meric-Bernstam F Cancer Treat Rev; 2024 Apr; 125():102720. PubMed ID: 38502995 [TBL] [Abstract][Full Text] [Related]
12. Datopotamab Deruxtecan in Advanced or Metastatic HR+/HER2- and Triple-Negative Breast Cancer: Results From the Phase I TROPION-PanTumor01 Study. Bardia A; Krop IE; Kogawa T; Juric D; Tolcher AW; Hamilton EP; Mukohara T; Lisberg A; Shimizu T; Spira AI; Tsurutani J; Damodaran S; Papadopoulos KP; Greenberg J; Kobayashi F; Zebger-Gong H; Wong R; Kawasaki Y; Nakamura T; Meric-Bernstam F J Clin Oncol; 2024 Jul; 42(19):2281-2294. PubMed ID: 38652877 [TBL] [Abstract][Full Text] [Related]
13. Blockade of SIRPα-CD47 axis by anti-SIRPα antibody enhances anti-tumor activity of DXd antibody-drug conjugates. Sue M; Tsubaki T; Ishimoto Y; Hayashi S; Ishida S; Otsuka T; Isumi Y; Kawase Y; Yamaguchi J; Nakada T; Ishiguro J; Nakamura K; Kawaida R; Ohtsuka T; Wada T; Agatsuma T; Kawasaki N PLoS One; 2024; 19(6):e0304985. PubMed ID: 38843278 [TBL] [Abstract][Full Text] [Related]
14. DB-1310, an ADC comprised of a novel anti-HER3 antibody conjugated to a DNA topoisomerase I inhibitor, is highly effective for the treatment of HER3-positive solid tumors. Li X; Yao J; Qu C; Luo L; Li B; Zhang Y; Zhu Z; Qiu Y; Hua H J Transl Med; 2024 Apr; 22(1):362. PubMed ID: 38632563 [TBL] [Abstract][Full Text] [Related]
15. DS-8201a, A Novel HER2-Targeting ADC with a Novel DNA Topoisomerase I Inhibitor, Demonstrates a Promising Antitumor Efficacy with Differentiation from T-DM1. Ogitani Y; Aida T; Hagihara K; Yamaguchi J; Ishii C; Harada N; Soma M; Okamoto H; Oitate M; Arakawa S; Hirai T; Atsumi R; Nakada T; Hayakawa I; Abe Y; Agatsuma T Clin Cancer Res; 2016 Oct; 22(20):5097-5108. PubMed ID: 27026201 [TBL] [Abstract][Full Text] [Related]
16. Antibody-drug conjugates targeting TROP-2: Clinical development in metastatic breast cancer. Shastry M; Jacob S; Rugo HS; Hamilton E Breast; 2022 Dec; 66():169-177. PubMed ID: 36302269 [TBL] [Abstract][Full Text] [Related]
17. Datopotamab Deruxtecan Versus Chemotherapy in Previously Treated Inoperable/Metastatic Hormone Receptor-Positive Human Epidermal Growth Factor Receptor 2-Negative Breast Cancer: Primary Results From TROPION-Breast01. Bardia A; Jhaveri K; Im SA; Pernas S; De Laurentiis M; Wang S; Martínez Jañez N; Borges G; Cescon DW; Hattori M; Lu YS; Hamilton E; Zhang Q; Tsurutani J; Kalinsky K; Rubini Liedke PE; Xu L; Fairhurst RM; Khan S; Denduluri N; Rugo HS; Xu B; Pistilli B; J Clin Oncol; 2024 Sep; ():JCO2400920. PubMed ID: 39265124 [TBL] [Abstract][Full Text] [Related]
18. Safety evaluation of Datopotamab deruxtecan for triple-negative breast cancer: a meta-analysis. Gadaleta-Caldarola G; Lanotte L; Infusino S; Gadaleta-Caldarola A; Schipilliti FM; Citrigno C; Petrarota C; Cusmai A; Rizzo A Cancer Treat Res Commun; 2023; 37():100775. PubMed ID: 37956525 [TBL] [Abstract][Full Text] [Related]
19. Datopotamab deruxtecan: A novel antibody drug conjugate for triple-negative breast cancer. Schipilliti FM; Drittone D; Mazzuca F; La Forgia D; Guven DC; Rizzo A Heliyon; 2024 Apr; 10(7):e28385. PubMed ID: 38560142 [TBL] [Abstract][Full Text] [Related]
20. Comprehensive preclinical pharmacokinetic evaluations of trastuzumab deruxtecan (DS-8201a), a HER2-targeting antibody-drug conjugate, in cynomolgus monkeys. Nagai Y; Oitate M; Shiozawa H; Ando O Xenobiotica; 2019 Sep; 49(9):1086-1096. PubMed ID: 30351177 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]