These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

134 related articles for article (PubMed ID: 34878728)

  • 1. Chalcone-inspired rA
    Matthee C; Terre'Blanche G; Janse van Rensburg HD; Aucamp J; Legoabe LJ
    Chem Biol Drug Des; 2022 Mar; 99(3):416-437. PubMed ID: 34878728
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 2-Benzylidene-1-Indanone Analogues as Dual Adenosine A1/A2a Receptor Antagonists for the Potential Treatment of Neurological Conditions.
    van Rensburg HJ; Legoabe L; Terre'Blanche G; Van der Walt M
    Drug Res (Stuttg); 2019 Jul; 69(7):382-391. PubMed ID: 30616250
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Adenosine Receptor Ligands: Coumarin-Chalcone Hybrids as Modulating Agents on the Activity of
    Vazquez-Rodriguez S; Vilar S; Kachler S; Klotz KN; Uriarte E; Borges F; Matos MJ
    Molecules; 2020 Sep; 25(18):. PubMed ID: 32961824
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Evaluation of 2-benzylidene-1-tetralone derivatives as antagonists of A
    Legoabe LJ; Van der Walt MM; Terre'Blanche G
    Chem Biol Drug Des; 2018 Jan; 91(1):234-244. PubMed ID: 28734058
    [TBL] [Abstract][Full Text] [Related]  

  • 5. 5-Substituted 2-benzylidene-1-tetralone analogues as A
    Janse van Rensburg HD; Terre'Blanche G; van der Walt MM; Legoabe LJ
    Bioorg Chem; 2017 Oct; 74():251-259. PubMed ID: 28881253
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and evaluation of methoxy substituted 2-benzoyl-1-benzofuran derivatives as lead compounds for the development adenosine A
    Janse van Rensburg HD; Legoabe LJ; Terre'Blanche G; Aucamp J
    Bioorg Chem; 2020 Jan; 94():103459. PubMed ID: 31818481
    [TBL] [Abstract][Full Text] [Related]  

  • 7. C2-substituted quinazolinone derivatives exhibit A
    Pieterse L; van der Walt MM; Terre'Blanche G
    Bioorg Med Chem Lett; 2020 Aug; 30(16):127274. PubMed ID: 32631506
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Benzopyrone represents a privilege scaffold to identify novel adenosine A
    van der Walt MM; Terre'Blanche G
    Bioorg Chem; 2018 Apr; 77():136-143. PubMed ID: 29353730
    [TBL] [Abstract][Full Text] [Related]  

  • 9. New fused pyrroles with rA1/A2A antagonistic activity as potential therapeutics for neurodegenerative disorders.
    van Vuuren NJ; van Rensburg HDJ; Terre'Blanche G; Legoabe LJ
    Mol Divers; 2022 Aug; 26(4):2211-2220. PubMed ID: 34741275
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Discovery of 1,3-diethyl-7-methyl-8-(phenoxymethyl)-xanthine derivatives as novel adenosine A
    Harmse R; van der Walt MM; Petzer JP; Terre'Blanche G
    Bioorg Med Chem Lett; 2016 Dec; 26(24):5951-5955. PubMed ID: 27836398
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Chalcone-based derivatives as new scaffolds for hA3 adenosine receptor antagonists.
    Vazquez-Rodriguez S; Matos MJ; Santana L; Uriarte E; Borges F; Kachler S; Klotz KN
    J Pharm Pharmacol; 2013 May; 65(5):697-703. PubMed ID: 23600387
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Carbamate substituted 2-amino-4,6-diphenylpyrimidines as adenosine receptor antagonists.
    Robinson SJ; Petzer JP; Rousseau AL; Terre'Blanche G; Petzer A; Lourens ACU
    Bioorg Med Chem Lett; 2016 Feb; 26(3):734-738. PubMed ID: 26776359
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Design, synthesis, and biological evaluation of a second generation of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as potent and selective A2A adenosine receptor antagonists.
    Baraldi PG; Cacciari B; Spalluto G; Bergonzoni M; Dionisotti S; Ongini E; Varani K; Borea PA
    J Med Chem; 1998 Jun; 41(12):2126-33. PubMed ID: 9622554
    [TBL] [Abstract][Full Text] [Related]  

  • 14. C3 amino-substituted chalcone derivative with selective adenosine
    Janse van Rensburg HD; Legoabe LJ; Terre'Blanche G
    Chem Zvesti; 2021; 75(4):1581-1605. PubMed ID: 33223599
    [TBL] [Abstract][Full Text] [Related]  

  • 15. 2-Aminopyrimidines as dual adenosine A1/A2A antagonists.
    Robinson SJ; Petzer JP; Terre'Blanche G; Petzer A; van der Walt MM; Bergh JJ; Lourens AC
    Eur J Med Chem; 2015 Nov; 104():177-88. PubMed ID: 26462195
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Identification of novel thiazolo[5,4-d]pyrimidine derivatives as human A
    Varano F; Catarzi D; Falsini M; Vincenzi F; Pasquini S; Varani K; Colotta V
    Bioorg Med Chem; 2018 Jul; 26(12):3688-3695. PubMed ID: 29880250
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and Structure Activity Relationships of Chalcone based Benzocycloalkanone Derivatives as Adenosine A1 and/or A2A Receptor Antagonists.
    Janse van Rensburg HD; Legoabe LJ; Terre'Blanche G
    Drug Res (Stuttg); 2020 Jun; 70(6):243-256. PubMed ID: 32349128
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Structures of Human A
    Cheng RKY; Segala E; Robertson N; Deflorian F; Doré AS; Errey JC; Fiez-Vandal C; Marshall FH; Cooke RM
    Structure; 2017 Aug; 25(8):1275-1285.e4. PubMed ID: 28712806
    [TBL] [Abstract][Full Text] [Related]  

  • 19. JNJ-40255293, a novel adenosine A2A/A1 antagonist with efficacy in preclinical models of Parkinson's disease.
    Atack JR; Shook BC; Rassnick S; Jackson PF; Rhodes K; Drinkenburg WH; Ahnaou A; Te Riele P; Langlois X; Hrupka B; De Haes P; Hendrickx H; Aerts N; Hens K; Wellens A; Vermeire J; Megens AA
    ACS Chem Neurosci; 2014 Oct; 5(10):1005-19. PubMed ID: 25203719
    [TBL] [Abstract][Full Text] [Related]  

  • 20. N9-benzyl-substituted 1,3-dimethyl- and 1,3-dipropyl-pyrimido[2,1-f]purinediones: synthesis and structure-activity relationships at adenosine A1 and A2A receptors.
    Drabczyńska A; Müller CE; Karolak-Wojciechowska J; Schumacher B; Schiedel A; Yuzlenko O; Kieć-Kononowicz K
    Bioorg Med Chem; 2007 Jul; 15(14):5003-17. PubMed ID: 17499511
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.