BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

119 related articles for article (PubMed ID: 34897776)

  • 1. Synthesis of novel hybrid pharmacophore of N-((4-sulfamoylphenyl)carbamothioyl)alkanamides as potent carbonic anhydrase-II and 15-lipoxygenase inhibitors.
    Saeed A; Khan SU; Saeed M; Shabir G; Hasan A; Khera RA; El-Seedi H; Halim SA; Khan A; Al-Harrasi A; Iqbal J
    Drug Dev Res; 2022 May; 83(3):745-754. PubMed ID: 34897776
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Substituted (E)-2-(2-benzylidenehydrazinyl)-4-methylthiazole-5-carboxylates as dual inhibitors of 15-lipoxygenase & carbonic anhydrase II: synthesis, biochemical evaluation and docking studies.
    Saeed A; Khan SU; Mahesar PA; Channar PA; Shabir G; Iqbal J
    Biochem Biophys Res Commun; 2017 Jan; 482(1):176-181. PubMed ID: 27836541
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis, Biological Evaluation, and Molecular Dynamics of Carbothioamides Derivatives as Carbonic Anhydrase II and 15-Lipoxygenase Inhibitors.
    Channar PA; Alharthy RD; Ejaz SA; Saeed A; Iqbal J
    Molecules; 2022 Dec; 27(24):. PubMed ID: 36557863
    [TBL] [Abstract][Full Text] [Related]  

  • 4. New aminobenzenesulfonamide-thiourea conjugates: synthesis and carbonic anhydrase inhibition and docking studies.
    Zaib S; Saeed A; Stolte K; Flörke U; Shahid M; Iqbal J
    Eur J Med Chem; 2014 May; 78():140-50. PubMed ID: 24681391
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Inhibitory Efficacy of Thiosemicarbazones for Carbonic Anhydrase II (Bovine and Human) as a Target of Calcification and Tumorigenicity.
    Khan M; Halim SA; Shafiq Z; Islam M; Shehzad MT; Ibrar A; Khan FA; Marraiki N; Uddin J; Khan A; Al-Harrasi A
    Curr Pharm Des; 2022; 28(36):3010-3022. PubMed ID: 35909284
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Carbonic anhydrase inhibition by 1-aroyl-3-(4-aminosulfonylphenyl)thioureas.
    Saeed A; Al-Rashida M; Hamayoun M; Mumtaz A; Iqbal J
    J Enzyme Inhib Med Chem; 2014 Dec; 29(6):901-5. PubMed ID: 24666305
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, Synthesis, Kinetic Analysis and Pharmacophore-Directed Discovery of 3-Ethylaniline Hybrid Imino-Thiazolidinone as Potential Inhibitor of Carbonic Anhydrase II: An Emerging Biological Target for Treatment of Cancer.
    Ahmed A; Aziz M; Ejaz SA; Channar PA; Saeed A; Zargar S; Wani TA; Hamad A; Abbas Q; Raza H; Kim SJ
    Biomolecules; 2022 Nov; 12(11):. PubMed ID: 36421710
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, biological evaluation and molecular docking of novel pyrazole derivatives as potent carbonic anhydrase and acetylcholinesterase inhibitors.
    Turkan F; Cetin A; Taslimi P; Karaman M; Gulçin İ
    Bioorg Chem; 2019 May; 86():420-427. PubMed ID: 30769267
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis, carbonic anhydrase inhibitory activity and antioxidant activity of some 1,3-oxazine derivatives.
    Qamar R; Saeed A; Saeed M; Ashraf Z; Abbas Q; Hassan M; Albericio F
    Drug Dev Res; 2018 Nov; 79(7):352-361. PubMed ID: 30302774
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, Synthesis and Molecular Docking Study of Novel 3-Phenyl-β-Alanine-Based Oxadiazole Analogues as Potent Carbonic Anhydrase II Inhibitors.
    Rafiq K; Ur Rehman N; Halim SA; Khan M; Khan A; Al-Harrasi A
    Molecules; 2022 Jan; 27(3):. PubMed ID: 35164091
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of isoxazole-containing sulfonamides with potent carbonic anhydrase II and VII inhibitory properties.
    Altug C; Güneş H; Nocentini A; Monti SM; Buonanno M; Supuran CT
    Bioorg Med Chem; 2017 Feb; 25(4):1456-1464. PubMed ID: 28111158
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design, synthesis, characterization, in vitro and in silico evaluation of novel imidazo[2,1-b][1,3,4]thiadiazoles as highly potent acetylcholinesterase and non-classical carbonic anhydrase inhibitors.
    Askin S; Tahtaci H; Türkeş C; Demir Y; Ece A; Akalın Çiftçi G; Beydemir Ş
    Bioorg Chem; 2021 Aug; 113():105009. PubMed ID: 34052739
    [TBL] [Abstract][Full Text] [Related]  

  • 13. New Carbonic Anhydrase-II Inhibitors from Marine Macro Brown Alga
    Rafiq K; Khan A; Ur Rehman N; Halim SA; Khan M; Ali L; Hilal Al-Balushi A; Al-Busaidi HK; Al-Harrasi A
    Molecules; 2021 Nov; 26(23):. PubMed ID: 34885658
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Utilization of the common functional groups in bioactive molecules: Exploring dual inhibitory potential and computational analysis of keto esters against α-glucosidase and carbonic anhydrase-II enzymes.
    Khan I; Khan A; Halim SA; Khan M; Zaib S; Al-Yahyaei BEM; Al-Harrasi A; Ibrar A
    Int J Biol Macromol; 2021 Jan; 167():233-244. PubMed ID: 33249154
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysis.
    Ahmed A; Channar PA; Saeed A; Kalesse M; Kazi MA; Larik FA; Abbas Q; Hassan M; Raza H; Seo SY
    Bioorg Chem; 2019 May; 86():624-630. PubMed ID: 30807935
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, biological evaluation and computational studies of novel iminothiazolidinone benzenesulfonamides as potent carbonic anhydrase II and IX inhibitors.
    Mahmood SU; Saeed A; Bua S; Nocentini A; Gratteri P; Supuran CT
    Bioorg Chem; 2018 Apr; 77():381-386. PubMed ID: 29421714
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and investigation of inhibition effect of fluorinated sulfonamide derivatives on carbonic anhydrase.
    Benfodda Z; Guillen F; Romestand B; Dahmani A; Blancou H
    Eur J Med Chem; 2010 Mar; 45(3):1225-9. PubMed ID: 20036446
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis, biological evaluation, and docking studies of novel thiourea derivatives of bisindolylmethane as carbonic anhydrase II inhibitor.
    Imran S; Taha M; Ismail NH; Fayyaz S; Khan KM; Choudhary MI
    Bioorg Chem; 2015 Oct; 62():83-93. PubMed ID: 26275866
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Sulfonamides containing curcumin scaffold: Synthesis, characterization, carbonic anhydrase inhibition and molecular docking studies.
    Ahmed M; Qadir MA; Hameed A; Arshad MN; Asiri AM; Muddassar M
    Bioorg Chem; 2018 Feb; 76():218-227. PubMed ID: 29190478
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Sulfonamides incorporating ketene N,S-acetal bioisosteres as potent carbonic anhydrase and acetylcholinesterase inhibitors.
    Istrefi Q; Türkeş C; Arslan M; Demir Y; Nixha AR; Beydemir Ş; Küfrevioğlu ÖI
    Arch Pharm (Weinheim); 2020 Jun; 353(6):e1900383. PubMed ID: 32285537
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.