362 related articles for article (PubMed ID: 35157454)
1. Advances in the Development of Nonpeptide Small Molecules Targeting Ghrelin Receptor.
Giorgioni G; Del Bello F; Quaglia W; Botticelli L; Cifani C; Micioni Di Bonaventura E; Micioni Di Bonaventura MV; Piergentili A
J Med Chem; 2022 Feb; 65(4):3098-3118. PubMed ID: 35157454
[TBL] [Abstract][Full Text] [Related]
2. Small-molecule ghrelin receptor antagonists improve glucose tolerance, suppress appetite, and promote weight loss.
Esler WP; Rudolph J; Claus TH; Tang W; Barucci N; Brown SE; Bullock W; Daly M; Decarr L; Li Y; Milardo L; Molstad D; Zhu J; Gardell SJ; Livingston JN; Sweet LJ
Endocrinology; 2007 Nov; 148(11):5175-85. PubMed ID: 17656463
[TBL] [Abstract][Full Text] [Related]
3. Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling.
M'Kadmi C; Leyris JP; Onfroy L; Galés C; Saulière A; Gagne D; Damian M; Mary S; Maingot M; Denoyelle S; Verdié P; Fehrentz JA; Martinez J; Banères JL; Marie J
J Biol Chem; 2015 Nov; 290(45):27021-27039. PubMed ID: 26363071
[TBL] [Abstract][Full Text] [Related]
4. Ghrelin Receptor Ligands Reaching Clinical Trials: From Peptides to Peptidomimetics; from Agonists to Antagonists.
Vodnik M; Štrukelj B; Lunder M
Horm Metab Res; 2016 Jan; 48(1):1-15. PubMed ID: 26551992
[TBL] [Abstract][Full Text] [Related]
5. Recent developments in ghrelin receptor ligands.
Moulin A; Ryan J; Martinez J; Fehrentz JA
ChemMedChem; 2007 Sep; 2(9):1242-59. PubMed ID: 17520591
[TBL] [Abstract][Full Text] [Related]
6. Ghrelin control of GH secretion and feeding behaviour: the role of the GHS-R1a receptor studied in vivo and in vitro using novel non-peptide ligands.
Bresciani E; Tamiazzo L; Torsello A; Bulgarelli I; Rapetti D; Caporali S; Perrissoud D; Moulin A; Fehrentz JA; Martinez J; Locatelli V
Eat Weight Disord; 2008 Sep; 13(3):e67-74. PubMed ID: 19011367
[TBL] [Abstract][Full Text] [Related]
7. LEAP-2: An Emerging Endogenous Ghrelin Receptor Antagonist in the Pathophysiology of Obesity.
Lu X; Huang L; Huang Z; Feng D; Clark RJ; Chen C
Front Endocrinol (Lausanne); 2021; 12():717544. PubMed ID: 34512549
[TBL] [Abstract][Full Text] [Related]
8. The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist.
Moulin A; Brunel L; Boeglin D; Demange L; Ryan J; M'Kadmi C; Denoyelle S; Martinez J; Fehrentz JA
Amino Acids; 2013 Feb; 44(2):301-14. PubMed ID: 22798076
[TBL] [Abstract][Full Text] [Related]
9. Long-term treatment with the ghrelin receptor antagonist [d-Lys3]-GHRP-6 does not improve glucose homeostasis in nonobese diabetic MKR mice.
Mosa R; Huang L; Li H; Grist M; LeRoith D; Chen C
Am J Physiol Regul Integr Comp Physiol; 2018 Jan; 314(1):R71-R83. PubMed ID: 28903914
[TBL] [Abstract][Full Text] [Related]
10. Promiscuous dimerization of the growth hormone secretagogue receptor (GHS-R1a) attenuates ghrelin-mediated signaling.
Schellekens H; van Oeffelen WE; Dinan TG; Cryan JF
J Biol Chem; 2013 Jan; 288(1):181-91. PubMed ID: 23161547
[TBL] [Abstract][Full Text] [Related]
11. Sequence, genomic organization and expression of ghrelin receptor in grass carp, Ctenopharyngodon idellus.
Cai WJ; Yuan XC; Yuan YC; Xie SQ; Gong Y; Su H; Qiao Y
Comp Biochem Physiol A Mol Integr Physiol; 2015 Jan; 179():54-61. PubMed ID: 25242546
[TBL] [Abstract][Full Text] [Related]
12. Anorexigenic and electrophysiological actions of novel ghrelin receptor (GHS-R1A) antagonists in rats.
Salomé N; Haage D; Perrissoud D; Moulin A; Demange L; Egecioglu E; Fehrentz JA; Martinez J; Dickson SL
Eur J Pharmacol; 2009 Jun; 612(1-3):167-73. PubMed ID: 19356720
[TBL] [Abstract][Full Text] [Related]
13. Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a.
Leyris JP; Roux T; Trinquet E; Verdié P; Fehrentz JA; Oueslati N; Douzon S; Bourrier E; Lamarque L; Gagne D; Galleyrand JC; M'kadmi C; Martinez J; Mary S; Banères JL; Marie J
Anal Biochem; 2011 Jan; 408(2):253-62. PubMed ID: 20937574
[TBL] [Abstract][Full Text] [Related]
14. Modification of ghrelin receptor signaling by somatostatin receptor-5 regulates insulin release.
Park S; Jiang H; Zhang H; Smith RG
Proc Natl Acad Sci U S A; 2012 Nov; 109(46):19003-8. PubMed ID: 23112170
[TBL] [Abstract][Full Text] [Related]
15. Somatostatin, cortistatin, ghrelin and glucose metabolism.
Gauna C; van der Lely AJ
J Endocrinol Invest; 2005; 28(11 Suppl International):127-31. PubMed ID: 16625861
[TBL] [Abstract][Full Text] [Related]
16. The ghrelin receptors (GHS-R1a and GHS-R1b).
Albarrán-Zeckler RG; Smith RG
Endocr Dev; 2013; 25():5-15. PubMed ID: 23652387
[TBL] [Abstract][Full Text] [Related]
17. Ghrelin receptor in Japanese fire belly newt, Cynops pyrrhogaster.
Kaiya H; Kangawa K; Miyazato M
Comp Biochem Physiol B Biochem Mol Biol; 2015 Nov; 189():15-22. PubMed ID: 26172570
[TBL] [Abstract][Full Text] [Related]
18. Growth hormone-releasing hormone as an agonist of the ghrelin receptor GHS-R1a.
Casanueva FF; Camiña JP; Carreira MC; Pazos Y; Varga JL; Schally AV
Proc Natl Acad Sci U S A; 2008 Dec; 105(51):20452-7. PubMed ID: 19088192
[TBL] [Abstract][Full Text] [Related]
19. Food restriction, ghrelin, its antagonist and obestatin control expression of ghrelin and its receptor in chicken hypothalamus and ovary.
Sirotkin AV; Pavlova S; Tena-Sempere M; Grossmann R; Jiménez MR; Rodriguez JM; Valenzuela F
Comp Biochem Physiol A Mol Integr Physiol; 2013 Jan; 164(1):141-53. PubMed ID: 22877785
[TBL] [Abstract][Full Text] [Related]
20. Semagacestat, a γ-secretase inhibitor, activates the growth hormone secretagogue (GHS-R1a) receptor.
Schellekens H; McNamara O; Dinan TG; McCarthy JV; McGlacken GP; Cryan JF
J Pharm Pharmacol; 2013 Apr; 65(4):528-38. PubMed ID: 23488781
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]