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4. Enol lactone inhibitors of serine proteases. The effect of regiochemistry on the inactivation behavior of phenyl-substituted (halomethylene)tetra- and -dihydrofuranones and (halomethylene)tetrahydropyranones toward alpha-chymotrypsin: stable acyl enzyme intermediate. Sofia MJ; Katzenellenbogen JA J Med Chem; 1986 Feb; 29(2):230-8. PubMed ID: 3512826 [TBL] [Abstract][Full Text] [Related]
5. Inhibition of human leukocyte elastase, cathepsin G, chymotrypsin A alpha, and porcine pancreatic elastase with substituted isobenzofuranones and benzopyrandiones. Hemmi K; Harper JW; Powers JC Biochemistry; 1985 Apr; 24(8):1841-8. PubMed ID: 3848330 [TBL] [Abstract][Full Text] [Related]
6. Reaction of serine proteases with substituted 3-alkoxy-4-chloroisocoumarins and 3-alkoxy-7-amino-4-chloroisocoumarins: new reactive mechanism-based inhibitors. Harper JW; Powers JC Biochemistry; 1985 Dec; 24(25):7200-13. PubMed ID: 3910097 [TBL] [Abstract][Full Text] [Related]
7. A new class of heterocyclic serine protease inhibitors. Inhibition of human leukocyte elastase, porcine pancreatic elastase, cathepsin G, and bovine chymotrypsin A alpha with substituted benzoxazinones, quinazolines, and anthranilates. Teshima T; Griffin JC; Powers JC J Biol Chem; 1982 May; 257(9):5085-91. PubMed ID: 7040392 [TBL] [Abstract][Full Text] [Related]
8. Mechanism of inhibition of human leucocyte elastase by monocyclic beta-lactams. Chabin R; Green BG; Gale P; Maycock AL; Weston H; Dorn CP; Finke PE; Hagmann WK; Hale JJ; MacCoss M Biochemistry; 1993 Aug; 32(34):8970-80. PubMed ID: 8364042 [TBL] [Abstract][Full Text] [Related]
10. Reaction of serine proteases with substituted isocoumarins: discovery of 3,4-dichloroisocoumarin, a new general mechanism based serine protease inhibitor. Harper JW; Hemmi K; Powers JC Biochemistry; 1985 Apr; 24(8):1831-41. PubMed ID: 3893537 [TBL] [Abstract][Full Text] [Related]
11. Inhibition of the human leukocyte endopeptidases elastase and cathepsin G and of porcine pancreatic elastase by N-oleoyl derivatives of heparin. Baici A; Diczházi C; Neszmélyi A; Móczár E; Hornebeck W Biochem Pharmacol; 1993 Nov; 46(9):1545-9. PubMed ID: 8240409 [TBL] [Abstract][Full Text] [Related]
12. Mechanism for slow-binding inhibition of human leukocyte elastase by valine-derived benzoxazinones. Stein RL; Strimpler AM; Viscarello BR; Wildonger RA; Mauger RC; Trainor DA Biochemistry; 1987 Jun; 26(13):4126-30. PubMed ID: 3651441 [TBL] [Abstract][Full Text] [Related]
13. Halo enol lactones: studies on the mechanism of inactivation of alpha-chymotrypsin. Daniels SB; Katzenellenbogen JA Biochemistry; 1986 Mar; 25(6):1436-44. PubMed ID: 3964685 [TBL] [Abstract][Full Text] [Related]
14. Inhibition of serine proteases by benzoxazinones: effects of electron withdrawal and 5-substitution. Spencer RW; Copp LJ; Bonaventura B; Tam TF; Liak TJ; Billedeau RJ; Krantz A Biochem Biophys Res Commun; 1986 Nov; 140(3):928-33. PubMed ID: 3535800 [TBL] [Abstract][Full Text] [Related]
15. Substituted 3-oxo-1,2,5-thiadiazolidine 1,1-dioxides: a new class of potential mechanism-based inhibitors of human leukocyte elastase and cathepsin G. Groutas WC; Kuang R; Venkataraman R Biochem Biophys Res Commun; 1994 Jan; 198(1):341-9. PubMed ID: 8292039 [TBL] [Abstract][Full Text] [Related]
16. Active site mapping of the serine proteases human leukocyte elastase, cathepsin G, porcine pancreatic elastase, rat mast cell proteases I and II. Bovine chymotrypsin A alpha, and Staphylococcus aureus protease V-8 using tripeptide thiobenzyl ester substrates. Harper JW; Cook RR; Roberts CJ; McLaughlin BJ; Powers JC Biochemistry; 1984 Jun; 23(13):2995-3002. PubMed ID: 6380580 [TBL] [Abstract][Full Text] [Related]
17. Irreversible inhibition of serine proteases by peptide derivatives of (alpha-aminoalkyl)phosphonate diphenyl esters. Oleksyszyn J; Powers JC Biochemistry; 1991 Jan; 30(2):485-93. PubMed ID: 1988040 [TBL] [Abstract][Full Text] [Related]
18. The Lossen rearrangement in biological systems. Inactivation of leukocyte elastase and alpha-chymotrypsin by (dl)-3-benzyl-N-(methanesulfonyloxy) succinimide. Groutas WC; Giri PK; Crowley JP; Castrisos JC; Brubaker MJ Biochem Biophys Res Commun; 1986 Dec; 141(2):741-8. PubMed ID: 3643025 [TBL] [Abstract][Full Text] [Related]
19. Mechanism of inhibition of human leucocyte elastase by beta-lactams. 2. Stability, reactivation kinetics, and products of beta-lactam-derived E-I complexes. Green BG; Chabin R; Mills S; Underwood DJ; Shah SK; Kuo D; Gale P; Maycock AL; Liesch J; Burgey CS Biochemistry; 1995 Nov; 34(44):14331-43. PubMed ID: 7578037 [TBL] [Abstract][Full Text] [Related]
20. Catalysis by human leukocyte elastase: proton inventory as a mechanistic probe. Stein RL; Strimpler AM; Hori H; Powers JC Biochemistry; 1987 Mar; 26(5):1305-14. PubMed ID: 3032250 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]