153 related articles for article (PubMed ID: 35833378)
1. Discovery of novel mRNA demethylase FTO inhibitors against esophageal cancer.
Qin B; Bai Q; Yan D; Yin F; Zhu Z; Xia C; Yang Y; Zhao Y
J Enzyme Inhib Med Chem; 2022 Dec; 37(1):1995-2003. PubMed ID: 35833378
[TBL] [Abstract][Full Text] [Related]
2. Anti-cancer effect of entacaponeon esophageal cancer cells via apoptosis induction and cell cycle modulation.
Ramedani F; Jafari SM; Saghaeian Jazi M; Mohammadi Z; Asadi J
Cancer Rep (Hoboken); 2023 Mar; 6(3):e1759. PubMed ID: 36534072
[TBL] [Abstract][Full Text] [Related]
3. Rational Design and Optimization of m
Huff S; Kummetha IR; Zhang L; Wang L; Bray W; Yin J; Kelley V; Wang Y; Rana TM
J Med Chem; 2022 Aug; 65(16):10920-10937. PubMed ID: 35939803
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis and molecular docking studies of thymol based 1,2,3-triazole hybrids as thymidylate synthase inhibitors and apoptosis inducers against breast cancer cells.
Alam MM; Malebari AM; Syed N; Neamatallah T; Almalki ASA; Elhenawy AA; Obaid RJ; Alsharif MA
Bioorg Med Chem; 2021 May; 38():116136. PubMed ID: 33894490
[TBL] [Abstract][Full Text] [Related]
5. LPE-1, an orally active pyrimidine derivative, inhibits growth and mobility of human esophageal cancers by targeting LSD1.
Wang B; Zhao B; Pang LP; Zhao YD; Guo Q; Wang JW; Zheng YC; Zhang XH; Liu Y; Liu GY; Guo WG; Wang C; Li ZH; Mao XJ; Yu B; Ma LY; Liu HM
Pharmacol Res; 2017 Aug; 122():66-77. PubMed ID: 28571892
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and biological evaluation of some novel 1,2,3-triazole hybrids of myrrhanone B isolated from Commiphora mukul gum resin: Identification of potent antiproliferative leads active against prostate cancer cells (PC-3).
Madasu C; Karri S; Sangaraju R; Sistla R; Uppuluri MV
Eur J Med Chem; 2020 Feb; 188():111974. PubMed ID: 31883489
[TBL] [Abstract][Full Text] [Related]
7. Alisertib, an Aurora kinase A inhibitor, induces apoptosis and autophagy but inhibits epithelial to mesenchymal transition in human epithelial ovarian cancer cells.
Ding YH; Zhou ZW; Ha CF; Zhang XY; Pan ST; He ZX; Edelman JL; Wang D; Yang YX; Zhang X; Duan W; Yang T; Qiu JX; Zhou SF
Drug Des Devel Ther; 2015; 9():425-64. PubMed ID: 25624750
[TBL] [Abstract][Full Text] [Related]
8. Small-Molecule Inhibitors of the RNA M6A Demethylases FTO Potently Support the Survival of Dopamine Neurons.
Selberg S; Yu LY; Bondarenko O; Kankuri E; Seli N; Kovaleva V; Herodes K; Saarma M; Karelson M
Int J Mol Sci; 2021 Apr; 22(9):. PubMed ID: 33926120
[TBL] [Abstract][Full Text] [Related]
9. Novel benzotriazole N-acylarylhydrazone hybrids: Design, synthesis, anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis and FAK inhibition.
Kassab AE; Hassan RA
Bioorg Chem; 2018 Oct; 80():531-544. PubMed ID: 30014921
[TBL] [Abstract][Full Text] [Related]
10. Identifying the novel inhibitors of lysine-specific demethylase 1 (LSD1) combining pharmacophore-based and structure-based virtual screening.
Sun XD; Zheng YC; Ma CY; Yang J; Gao QB; Yan Y; Wang ZZ; Li W; Zhao W; Liu HM; Ding L
J Biomol Struct Dyn; 2019 Oct; 37(16):4200-4214. PubMed ID: 30366512
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and Preclinical Evaluation of Indole Triazole Conjugates as Microtubule Targeting Agents that are Effective against MCF-7 Breast Cancer Cell Lines.
Yele V; Pindiprolu SKSS; Sana S; Ramamurty DSVNM; Madasi JRK; Vadlamani S
Anticancer Agents Med Chem; 2021; 21(8):1047-1055. PubMed ID: 32981511
[TBL] [Abstract][Full Text] [Related]
12. Downregulation of the FTO m
Jeschke J; Collignon E; Al Wardi C; Krayem M; Bizet M; Jia Y; Garaud S; Wimana Z; Calonne E; Hassabi B; Morandini R; Deplus R; Putmans P; Dube G; Singh NK; Koch A; Shostak K; Rizzotto L; Ross RL; Desmedt C; Bareche Y; Rothé F; Lehmann-Che J; Duterque-Coquillaud M; Leroy X; Menschaert G; Teixeira L; Guo M; Limbach PA; Close P; Chariot A; Leucci E; Ghanem G; Yuan BF; Willard-Gallo K; Sotiriou C; Marine JC; Fuks F
Nat Cancer; 2021 Jun; 2(6):611-628. PubMed ID: 35121941
[TBL] [Abstract][Full Text] [Related]
13. Structure-based design and evaluation of novel N-phenyl-1H-indol-2-amine derivatives for fat mass and obesity-associated (FTO) protein inhibition.
Padariya M; Kalathiya U
Comput Biol Chem; 2016 Oct; 64():414-425. PubMed ID: 27644082
[TBL] [Abstract][Full Text] [Related]
14. Vitamin E succinate induces apoptosis via the PI3K/AKT signaling pathways in EC109 esophageal cancer cells.
Yang P; Zhao J; Hou L; Yang L; Wu K; Zhang L
Mol Med Rep; 2016 Aug; 14(2):1531-7. PubMed ID: 27357907
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis and molecular docking studies of novel N-benzenesulfonyl-1,2,3,4-tetrahydroisoquinoline-based triazoles with potential anticancer activity.
Pingaew R; Mandi P; Nantasenamat C; Prachayasittikul S; Ruchirawat S; Prachayasittikul V
Eur J Med Chem; 2014 Jun; 81():192-203. PubMed ID: 24836071
[TBL] [Abstract][Full Text] [Related]
16. Synthesis, anticancer activity and molecular modeling studies of 1,2,4-triazole derivatives as EGFR inhibitors.
El-Sherief HAM; Youssif BGM; Abbas Bukhari SN; Abdelazeem AH; Abdel-Aziz M; Abdel-Rahman HM
Eur J Med Chem; 2018 Aug; 156():774-789. PubMed ID: 30055463
[TBL] [Abstract][Full Text] [Related]
17. The m6A demethylase FTO promotes the growth of lung cancer cells by regulating the m6A level of USP7 mRNA.
Li J; Han Y; Zhang H; Qian Z; Jia W; Gao Y; Zheng H; Li B
Biochem Biophys Res Commun; 2019 May; 512(3):479-485. PubMed ID: 30905413
[TBL] [Abstract][Full Text] [Related]
18. Structural characteristics of small-molecule inhibitors targeting
Gao S; Li X; Zhang M; Zhang N; Wang R; Chang J
Future Med Chem; 2021 Sep; 13(17):1475-1489. PubMed ID: 34240624
[TBL] [Abstract][Full Text] [Related]
19. Bardoxolone methyl induces apoptosis and autophagy and inhibits epithelial-to-mesenchymal transition and stemness in esophageal squamous cancer cells.
Wang YY; Yang YX; Zhao R; Pan ST; Zhe H; He ZX; Duan W; Zhang X; Yang T; Qiu JX; Zhou SF
Drug Des Devel Ther; 2015; 9():993-1026. PubMed ID: 25733817
[TBL] [Abstract][Full Text] [Related]
20. FTO m6A Demethylase in Obesity and Cancer: Implications and Underlying Molecular Mechanisms.
Azzam SK; Alsafar H; Sajini AA
Int J Mol Sci; 2022 Mar; 23(7):. PubMed ID: 35409166
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
