BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

190 related articles for article (PubMed ID: 36167735)

  • 1. Bis-pharmacophore of cinnamaldehyde-clubbed thiosemicarbazones as potent carbonic anhydrase-II inhibitors.
    Rasool A; Batool Z; Khan M; Halim SA; Shafiq Z; Temirak A; Salem MA; Ali TE; Khan A; Al-Harrasi A
    Sci Rep; 2022 Sep; 12(1):16095. PubMed ID: 36167735
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, Synthesis and Molecular Docking Study of Novel 3-Phenyl-β-Alanine-Based Oxadiazole Analogues as Potent Carbonic Anhydrase II Inhibitors.
    Rafiq K; Ur Rehman N; Halim SA; Khan M; Khan A; Al-Harrasi A
    Molecules; 2022 Jan; 27(3):. PubMed ID: 35164091
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Inhibitory Efficacy of Thiosemicarbazones for Carbonic Anhydrase II (Bovine and Human) as a Target of Calcification and Tumorigenicity.
    Khan M; Halim SA; Shafiq Z; Islam M; Shehzad MT; Ibrar A; Khan FA; Marraiki N; Uddin J; Khan A; Al-Harrasi A
    Curr Pharm Des; 2022; 28(36):3010-3022. PubMed ID: 35909284
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Utilization of the common functional groups in bioactive molecules: Exploring dual inhibitory potential and computational analysis of keto esters against α-glucosidase and carbonic anhydrase-II enzymes.
    Khan I; Khan A; Halim SA; Khan M; Zaib S; Al-Yahyaei BEM; Al-Harrasi A; Ibrar A
    Int J Biol Macromol; 2021 Jan; 167():233-244. PubMed ID: 33249154
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel 2-substituted thioquinazoline-benzenesulfonamide derivatives as carbonic anhydrase inhibitors with potential anticancer activity.
    Abdel-Mohsen HT; Omar MA; Petreni A; Supuran CT
    Arch Pharm (Weinheim); 2022 Dec; 355(12):e2200180. PubMed ID: 36056903
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysis.
    Ahmed A; Channar PA; Saeed A; Kalesse M; Kazi MA; Larik FA; Abbas Q; Hassan M; Raza H; Seo SY
    Bioorg Chem; 2019 May; 86():624-630. PubMed ID: 30807935
    [TBL] [Abstract][Full Text] [Related]  

  • 7. New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies.
    Abdel-Mohsen HT; El Kerdawy AM; Omar MA; Berrino E; Abdelsamie AS; El Diwani HI; Supuran CT
    Bioorg Med Chem; 2020 Mar; 28(5):115329. PubMed ID: 32007388
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, carbonic anhydrase inhibitory activity and antioxidant activity of some 1,3-oxazine derivatives.
    Qamar R; Saeed A; Saeed M; Ashraf Z; Abbas Q; Hassan M; Albericio F
    Drug Dev Res; 2018 Nov; 79(7):352-361. PubMed ID: 30302774
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Potential inhibitors of human carbonic anhydrase isozymes I and II: Design, synthesis and docking studies of new 1,3,4-thiadiazole derivatives.
    Altıntop MD; Sever B; Özdemir A; Kucukoglu K; Onem H; Nadaroglu H; Kaplancıklı ZA
    Bioorg Med Chem; 2017 Jul; 25(13):3547-3554. PubMed ID: 28511907
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, Synthesis, Kinetic Analysis and Pharmacophore-Directed Discovery of 3-Ethylaniline Hybrid Imino-Thiazolidinone as Potential Inhibitor of Carbonic Anhydrase II: An Emerging Biological Target for Treatment of Cancer.
    Ahmed A; Aziz M; Ejaz SA; Channar PA; Saeed A; Zargar S; Wani TA; Hamad A; Abbas Q; Raza H; Kim SJ
    Biomolecules; 2022 Nov; 12(11):. PubMed ID: 36421710
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of novel bisindolylmethanes: New carbonic anhydrase II inhibitors, docking, and 3D pharmacophore studies.
    Imran S; Taha M; Ismail NH; Fayyaz S; Khan KM; Choudhary MI
    Bioorg Chem; 2016 Oct; 68():90-104. PubMed ID: 27474804
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Pharmacophores Modeling in Terms of Prediction of Theoretical Physicochemical Properties and Verification by EXPERIMENTAL correlations of Carbacylamidophosphates (CAPh) and Sulfanylamidophosphates (SAPh) Tested as New Carbonic Anhydrase Inhibitors.
    Amirkhanov V; Rauf A; Hadda TB; Ovchynnikov V; Trush V; Saleem M; Raza M; Rehman T; Zgou H; Shaheen U; Farghaly TA
    Mini Rev Med Chem; 2019; 19(12):1015-1027. PubMed ID: 30806314
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis, molecular docking analysis and carbonic anhydrase I-II inhibitory evaluation of new sulfonamide derivatives.
    Sağlık BN; Çevik UA; Osmaniye D; Levent S; Çavuşoğlu BK; Demir Y; Ilgın S; Özkay Y; Koparal AS; Beydemir Ş; Kaplancıklı ZA
    Bioorg Chem; 2019 Oct; 91():103153. PubMed ID: 31382057
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.
    Di Fiore A; De Simone G; Menchise V; Pedone C; Casini A; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2005 Apr; 15(7):1937-42. PubMed ID: 15780637
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Effect of incorporating a thiophene tail in the scaffold of acetazolamide on the inhibition of human carbonic anhydrase isoforms I, II, IX and XII.
    Biswas S; McKenna R; Supuran CT
    Bioorg Med Chem Lett; 2013 Oct; 23(20):5646-9. PubMed ID: 23993330
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Enzyme inhibition, molecular docking, and density functional theory studies of new thiosemicarbazones incorporating the 4-hydroxy-3,5-dimethoxy benzaldehyde motif.
    Demir Y; Türkeş C; Çavuş MS; Erdoğan M; Muğlu H; Yakan H; Beydemir Ş
    Arch Pharm (Weinheim); 2023 Apr; 356(4):e2200554. PubMed ID: 36575148
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis, Biological Evaluation, and Molecular Dynamics of Carbothioamides Derivatives as Carbonic Anhydrase II and 15-Lipoxygenase Inhibitors.
    Channar PA; Alharthy RD; Ejaz SA; Saeed A; Iqbal J
    Molecules; 2022 Dec; 27(24):. PubMed ID: 36557863
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Inhibition of carbonic anhydrase II by sulfonamide derivatives.
    Xuan GS; Zhan JH; Zhang AM; Li W; Zheng K
    Pharmazie; 2021 Sep; 76(9):412-415. PubMed ID: 34481530
    [TBL] [Abstract][Full Text] [Related]  

  • 19. New Carbonic Anhydrase-II Inhibitors from Marine Macro Brown Alga
    Rafiq K; Khan A; Ur Rehman N; Halim SA; Khan M; Ali L; Hilal Al-Balushi A; Al-Busaidi HK; Al-Harrasi A
    Molecules; 2021 Nov; 26(23):. PubMed ID: 34885658
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of arjunolic acid as a novel non-zinc binding carbonic anhydrase II inhibitor.
    Kalyanavenkataraman S; Nanjan P; Banerji A; Nair BG; Kumar GB
    Bioorg Chem; 2016 Jun; 66():72-9. PubMed ID: 27038848
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.