114 related articles for article (PubMed ID: 3625701)
1. Indazoles as indole bioisosteres: synthesis and evaluation of the tropanyl ester and amide of indazole-3-carboxylate as antagonists at the serotonin 5HT3 receptor.
Fludzinski P; Evrard DA; Bloomquist WE; Lacefield WB; Pfeifer W; Jones ND; Deeter JB; Cohen ML
J Med Chem; 1987 Sep; 30(9):1535-7. PubMed ID: 3625701
[No Abstract] [Full Text] [Related]
2. Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
Robertson DW; Bloomquist W; Cohen ML; Reid LR; Schenck K; Wong DT
J Med Chem; 1990 Dec; 33(12):3176-81. PubMed ID: 2258903
[TBL] [Abstract][Full Text] [Related]
3. 5-Hydroxytryptamine (5-HT3) receptor antagonists. 3. Ortho-substituted phenylureas.
Bermudez J; Dabbs S; King FD
J Med Chem; 1990 Jul; 33(7):1932-5. PubMed ID: 2362272
[TBL] [Abstract][Full Text] [Related]
4. 5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives.
Bermudez J; Fake CS; Joiner GF; Joiner KA; King FD; Miner WD; Sanger GJ
J Med Chem; 1990 Jul; 33(7):1924-9. PubMed ID: 2362270
[TBL] [Abstract][Full Text] [Related]
5. 5-Hydroxytryptamine (5-HT3) receptor antagonists. 2. 1-Indolinecarboxamides.
Bermudez J; Dabbs S; Joiner KA; King FD
J Med Chem; 1990 Jul; 33(7):1929-32. PubMed ID: 2362271
[TBL] [Abstract][Full Text] [Related]
6. BRL 43694, a new 5HT3 receptor antagonist, prevents cisplatin-induced emesis in dogs.
Bhandari P; Gupta YK; Seth SD
Methods Find Exp Clin Pharmacol; 1989 May; 11(5):361-3. PubMed ID: 2547129
[No Abstract] [Full Text] [Related]
7. 5-Piperazinyl-3-sulfonylindazoles as potent and selective 5-hydroxytryptamine-6 antagonists.
Liu KG; Robichaud AJ; Bernotas RC; Yan Y; Lo JR; Zhang MY; Hughes ZA; Huselton C; Zhang GM; Zhang JY; Kowal DM; Smith DL; Schechter LE; Comery TA
J Med Chem; 2010 Nov; 53(21):7639-46. PubMed ID: 20932009
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and biological activity of a series of aryl tropanyl esters and amides chemically related to 1H-indole-3-carboxylic acid endo 8-methyl-8-azabicyclo[3.2.1]oct-3-yl ester. Development of a 5-HT4 agonist endowed with potent antinociceptive activity.
Romanelli MN; Ghelardini C; Dei S; Matucci R; Mori F; Scapecchi S; Teodori E; Bartolini A; Galli A; Giotti A
Arzneimittelforschung; 1993 Aug; 43(8):913-8. PubMed ID: 8216452
[TBL] [Abstract][Full Text] [Related]
9. The antinociceptive effect induced by FR140423 is mediated through spinal 5-HT2A and 5-HT3 receptors.
Ochi T; Goto T
Eur J Pharmacol; 2000 Dec; 409(2):167-72. PubMed ID: 11104830
[TBL] [Abstract][Full Text] [Related]
10. Benzoxazines. II. Synthesis, conformational analysis, and structure--activity relationships of 3,4-dihydro-2H-1,4-benzoxazine-8-carboxamide derivatives as potent and long-acting serotonin-3 (5-HT3) receptor antagonists.
Kuroita T; Marubayashi N; Sano M; Kanzaki K; Inaba K; Kawakita T
Chem Pharm Bull (Tokyo); 1996 Nov; 44(11):2051-60. PubMed ID: 8945770
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and structure-activity relationships of potent and orally active 5-HT4 receptor antagonists: indazole and benzimidazolone derivatives.
Schaus JM; Thompson DC; Bloomquist WE; Susemichel AD; Calligaro DO; Cohen ML
J Med Chem; 1998 May; 41(11):1943-55. PubMed ID: 9599243
[TBL] [Abstract][Full Text] [Related]
12. New 2-piperazinylbenzimidazole derivatives as 5-HT3 antagonists. Synthesis and pharmacological evaluation.
Orjales A; Mosquera R; Labeaga L; Rodes R
J Med Chem; 1997 Feb; 40(4):586-93. PubMed ID: 9046349
[TBL] [Abstract][Full Text] [Related]
13. Antagonistic activities of N-3389, a newly synthesized diazabicyclo derivative, at 5-HT3 and 5-HT4 receptors.
Hagihara K; Hayakawa T; Arai T; Eguchi H; Mino S; Kawase S
Eur J Pharmacol; 1994 Dec; 271(1):159-66. PubMed ID: 7698198
[TBL] [Abstract][Full Text] [Related]
14. Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
Klein RL; Sanna E; McQuilkin SJ; Whiting PJ; Harris RA
Eur J Pharmacol; 1994 Jul; 268(2):237-46. PubMed ID: 7957645
[TBL] [Abstract][Full Text] [Related]
15. Specific [3H]LY278584 binding to 5-HT3 recognition sites in rat cerebral cortex.
Wong DT; Robertson DW; Reid LR
Eur J Pharmacol; 1989 Jul; 166(1):107-10. PubMed ID: 2806363
[TBL] [Abstract][Full Text] [Related]
16. Propulsion in guinea pig colon induced by 5-hydroxytryptamine (HT) via 5-HT4 and 5-HT3 receptors.
Jin JG; Foxx-Orenstein AE; Grider JR
J Pharmacol Exp Ther; 1999 Jan; 288(1):93-7. PubMed ID: 9862758
[TBL] [Abstract][Full Text] [Related]
17. Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT(6) antagonists.
Liu KG; Robichaud AJ; Greenfield AA; Lo JR; Grosanu C; Mattes JF; Cai Y; Zhang GM; Zhang JY; Kowal DM; Smith DL; Di L; Kerns EH; Schechter LE; Comery TA
Bioorg Med Chem; 2011 Jan; 19(1):650-62. PubMed ID: 21093272
[TBL] [Abstract][Full Text] [Related]
18. Glycinergic potentiation by some 5-HT(3) receptor antagonists: insight into selectivity.
Chesnoy-Marchais D; Lévi S; Acher F
Eur J Pharmacol; 2000 Aug; 402(3):205-13. PubMed ID: 10958886
[TBL] [Abstract][Full Text] [Related]
19. Effect of the amide fragment on 5-HT1A receptor activity of some analogs of MP 3022.
Paluchowska MH; Charakchieva-Minol S; Tatarczyńska E; Kłodzińska A
Pol J Pharmacol; 1999; 51(5):415-21. PubMed ID: 10817542
[TBL] [Abstract][Full Text] [Related]
20. Design and synthesis of 6-chloro-3,4-dihydro-4-methyl-2H-1,4-benzoxazine-8-carboxamide derivatives as potent serotonin-3 (5-HT3) receptor antagonists.
Kuroita T; Sakamori M; Kawakita T
Chem Pharm Bull (Tokyo); 1996 Apr; 44(4):756-64. PubMed ID: 8681408
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
