BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

168 related articles for article (PubMed ID: 36322425)

  • 1. Ibuprofen: a weak inhibitor of carbonic anhydrase II.
    Combs J; Andring J; McKenna R
    Acta Crystallogr F Struct Biol Commun; 2022 Nov; 78(Pt 11):395-402. PubMed ID: 36322425
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Carbonic anhydrase II in complex with carboxylic acid-based inhibitors.
    Lomelino CL; McKenna R
    Acta Crystallogr F Struct Biol Commun; 2019 Mar; 75(Pt 3):166-170. PubMed ID: 30839290
    [TBL] [Abstract][Full Text] [Related]  

  • 3. 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: solution and X-ray crystallographic studies.
    Leitans J; Sprudza A; Tanc M; Vozny I; Zalubovskis R; Tars K; Supuran CT
    Bioorg Med Chem; 2013 Sep; 21(17):5130-8. PubMed ID: 23859774
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Insights into the effect of elaborating coumarin-based aryl enaminones with sulfonamide or carboxylic acid functionality on carbonic anhydrase inhibitory potency and selectivity.
    Ibrahim HS; Abdelrahman MA; Nocentini A; Bua S; Abdel-Aziz HA; Supuran CT; Abou-Seri SM; Eldehna WM
    Bioorg Chem; 2022 Sep; 126():105888. PubMed ID: 35661530
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.
    Di Fiore A; De Simone G; Menchise V; Pedone C; Casini A; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2005 Apr; 15(7):1937-42. PubMed ID: 15780637
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Carbonic anhydrase inhibitors: X-ray and molecular modeling study for the interaction of a fluorescent antitumor sulfonamide with isozyme II and IX.
    Alterio V; Vitale RM; Monti SM; Pedone C; Scozzafava A; Cecchi A; De Simone G; Supuran CT
    J Am Chem Soc; 2006 Jun; 128(25):8329-35. PubMed ID: 16787097
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as potent carbonic anhydrase inhibitors: synthesis, biological evaluation, and enzyme--ligand X-ray studies.
    Gitto R; Agnello S; Ferro S; De Luca L; Vullo D; Brynda J; Mader P; Supuran CT; Chimirri A
    J Med Chem; 2010 Mar; 53(6):2401-8. PubMed ID: 20170095
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Identification, crystallization, and first X-ray structure analyses of phenyl boronic acid-based inhibitors of human carbonic anhydrase-II.
    Rasheed S; Huda NU; Fisher SZ; Falke S; Gul S; Ahmad MS; Choudhary MI
    Int J Biol Macromol; 2024 May; 267(Pt 1):131268. PubMed ID: 38580011
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Structural study of interaction between brinzolamide and dorzolamide inhibition of human carbonic anhydrases.
    Pinard MA; Boone CD; Rife BD; Supuran CT; McKenna R
    Bioorg Med Chem; 2013 Nov; 21(22):7210-5. PubMed ID: 24090602
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Dissecting the inhibition mechanism of cytosolic versus transmembrane carbonic anhydrases by ESR.
    Ciani L; Cecchi A; Temperini C; Supuran CT; Ristori S
    J Phys Chem B; 2009 Oct; 113(42):13998-4005. PubMed ID: 19778001
    [TBL] [Abstract][Full Text] [Related]  

  • 11. A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases.
    Langella E; D'Ambrosio K; D'Ascenzio M; Carradori S; Monti SM; Supuran CT; De Simone G
    Chemistry; 2016 Jan; 22(1):97-100. PubMed ID: 26507456
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds.
    Abdel-Aziz AA; El-Azab AS; Ceruso M; Supuran CT
    Bioorg Med Chem Lett; 2014 Nov; 24(22):5185-9. PubMed ID: 25442309
    [TBL] [Abstract][Full Text] [Related]  

  • 13. New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: biological evaluation and molecular modelling studies.
    Carradori S; Mollica A; Ceruso M; D'Ascenzio M; De Monte C; Chimenti P; Sabia R; Akdemir A; Supuran CT
    Bioorg Med Chem; 2015 Jul; 23(13):2975-81. PubMed ID: 26007302
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Selenocarbamates As a Prodrug-Based Approach to Carbonic Anhydrase Inhibition.
    Angeli A; Ferraroni M; Capperucci A; Tanini D; Costantino G; Supuran CT
    ChemMedChem; 2022 Jun; 17(11):e202200085. PubMed ID: 35238480
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Design and synthesis of some new benzoylthioureido phenyl derivatives targeting carbonic anhydrase enzymes.
    Najm MAA; Mahmoud WR; Taher AT; Abbas SE; Awadallah FM; Allam HA; Vullo D; Supuran CT
    J Enzyme Inhib Med Chem; 2022 Dec; 37(1):2702-2709. PubMed ID: 36168122
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of different thio-scaffolds bearing sulfonamide with subnanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism.
    Angeli A; Tanini D; Capperucci A; Malevolti G; Turco F; Ferraroni M; Supuran CT
    Bioorg Chem; 2018 Dec; 81():642-648. PubMed ID: 30253337
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.
    Garaj V; Puccetti L; Fasolis G; Winum JY; Montero JL; Scozzafava A; Vullo D; Innocenti A; Supuran CT
    Bioorg Med Chem Lett; 2005 Jun; 15(12):3102-8. PubMed ID: 15905091
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazinyl- or 2-(cyanophenylmethylene)-1,3,4-thiadiazol-3(2H)-yl moieties.
    Alafeefy AM; Abdel-Aziz HA; Vullo D; Al-Tamimi AM; Awaad AS; Mohamed MA; Capasso C; Supuran CT
    J Enzyme Inhib Med Chem; 2015 Feb; 30(1):52-6. PubMed ID: 24666294
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structural study of the location of the phenyl tail of benzene sulfonamides and the effect on human carbonic anhydrase inhibition.
    Güzel-Akdemir O; Biswas S; Lastra K; McKenna R; Supuran CT
    Bioorg Med Chem; 2013 Nov; 21(21):6674-80. PubMed ID: 24012377
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors.
    Tanc M; Carta F; Bozdag M; Scozzafava A; Supuran CT
    Bioorg Med Chem; 2013 Aug; 21(15):4502-10. PubMed ID: 23769167
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.