These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

239 related articles for article (PubMed ID: 36325394)

  • 1. Covalent drugs targeting histidine - an unexploited opportunity?
    Che J; Jones LH
    RSC Med Chem; 2022 Oct; 13(10):1121-1126. PubMed ID: 36325394
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Cereblon covalent modulation through structure-based design of histidine targeting chemical probes.
    Cruite JT; Dann GP; Che J; Donovan KA; Ferrao S; Ficarro SB; Fischer ES; Gray NS; Huerta F; Kong NR; Liu H; Marto JA; Metivier RJ; Nowak RP; Zerfas BL; Jones LH
    RSC Chem Biol; 2022 Aug; 3(9):1105-1110. PubMed ID: 36128501
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Covalent drug discovery using sulfur(VI) fluoride exchange warheads.
    Huang H; Jones LH
    Expert Opin Drug Discov; 2023 Jul; 18(7):725-735. PubMed ID: 37243622
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Covalent Stapling of the Cereblon Sensor Loop Histidine Using Sulfur-Heterocycle Exchange.
    Cruite JT; Nowak RP; Donovan KA; Ficarro SB; Huang H; Liu H; Liu Y; Marto JA; Metivier RJ; Fischer ES; Jones LH
    ACS Med Chem Lett; 2023 Nov; 14(11):1576-1581. PubMed ID: 37974938
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Sulfonyl fluorides as privileged warheads in chemical biology.
    Narayanan A; Jones LH
    Chem Sci; 2015 May; 6(5):2650-2659. PubMed ID: 28706662
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Rational targeting of active-site tyrosine residues using sulfonyl fluoride probes.
    Hett EC; Xu H; Geoghegan KF; Gopalsamy A; Kyne RE; Menard CA; Narayanan A; Parikh MD; Liu S; Roberts L; Robinson RP; Tones MA; Jones LH
    ACS Chem Biol; 2015 Apr; 10(4):1094-8. PubMed ID: 25571984
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1.
    Alboreggia G; Udompholkul P; Baggio C; Muzzarelli K; Assar Z; Pellecchia M
    J Med Chem; 2024 May; 67(10):8172-8185. PubMed ID: 38695666
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Development of sulfonyl fluoride chemical probes to advance the discovery of cereblon modulators.
    Liu Y; Nowak RP; Che J; Donovan KA; Huerta F; Liu H; Metivier RJ; Fischer ES; Jones LH
    RSC Med Chem; 2024 Feb; 15(2):607-611. PubMed ID: 38389883
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.
    Fadeyi OO; Hoth LR; Choi C; Feng X; Gopalsamy A; Hett EC; Kyne RE; Robinson RP; Jones LH
    ACS Chem Biol; 2017 Aug; 12(8):2015-2020. PubMed ID: 28718624
    [TBL] [Abstract][Full Text] [Related]  

  • 10. ABPP-CoDEL: Activity-Based Proteome Profiling-Guided Discovery of Tyrosine-Targeting Covalent Inhibitors from DNA-Encoded Libraries.
    Jiang L; Liu S; Jia X; Gong Q; Wen X; Lu W; Yang J; Wu X; Wang X; Suo Y; Li Y; Uesugi M; Qu ZB; Tan M; Lu X; Zhou L
    J Am Chem Soc; 2023 Nov; 145(46):25283-25292. PubMed ID: 37857329
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Covalent Inhibitors of Protein-Protein Interactions Targeting Lysine, Tyrosine, or Histidine Residues.
    Gambini L; Baggio C; Udompholkul P; Jossart J; Salem AF; Perry JJP; Pellecchia M
    J Med Chem; 2019 Jun; 62(11):5616-5627. PubMed ID: 31095386
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Arylfluorosulfate-Based Electrophiles for Covalent Protein Labeling: A New Addition to the Arsenal.
    Martín-Gago P; Olsen CA
    Angew Chem Int Ed Engl; 2019 Jan; 58(4):957-966. PubMed ID: 30024079
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Activation-Free Sulfonyl Fluoride Probes for Fragment Screening.
    Petri L; Ábrányi-Balogh P; Csorba N; Keeley A; Simon J; Ranđelović I; Tóvári J; Schlosser G; Szabó D; Drahos L; Keserű GM
    Molecules; 2023 Mar; 28(7):. PubMed ID: 37049805
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Characterising covalent warhead reactivity.
    Martin JS; MacKenzie CJ; Fletcher D; Gilbert IH
    Bioorg Med Chem; 2019 May; 27(10):2066-2074. PubMed ID: 30975501
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Imidazoles are Tunable Nucleofuges for Developing Tyrosine-Reactive Electrophiles.
    Justin Grams R; Yuan K; Founds MW; Ware ML; Pilar MG; Hsu KL
    Chembiochem; 2024 May; ():e202400382. PubMed ID: 38819848
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Advances in covalent kinase inhibitors.
    Abdeldayem A; Raouf YS; Constantinescu SN; Moriggl R; Gunning PT
    Chem Soc Rev; 2020 May; 49(9):2617-2687. PubMed ID: 32227030
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Lysine-Targeted Inhibitors and Chemoproteomic Probes.
    Cuesta A; Taunton J
    Annu Rev Biochem; 2019 Jun; 88():365-381. PubMed ID: 30633551
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Genetically Encoded Epoxide Warhead for Precise and Versatile Covalent Targeting of Proteins.
    Zhang J; Wang X; Huang Q; Ye J; Wang J
    J Am Chem Soc; 2024 Jun; 146(23):16173-16183. PubMed ID: 38819260
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Peptide-Based Covalent Inhibitors Bearing Mild Electrophiles to Target a Conserved His Residue of the Bacterial Sliding Clamp.
    Compain G; Monsarrat C; Blagojevic J; Brillet K; Dumas P; Hammann P; Kuhn L; Martiel I; Engilberge S; Oliéric V; Wolff P; Burnouf DY; Wagner J; Guichard G
    JACS Au; 2024 Feb; 4(2):432-440. PubMed ID: 38425897
    [TBL] [Abstract][Full Text] [Related]  

  • 20. The expanding repertoire of covalent warheads for drug discovery.
    Mehta NV; Degani MS
    Drug Discov Today; 2023 Dec; 28(12):103799. PubMed ID: 37839776
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 12.