BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

151 related articles for article (PubMed ID: 36364293)

  • 1. Substitutional Diversity-Oriented Synthesis and In Vitro Anticancer Activity of Framework-Integrated Estradiol-Benzisoxazole Chimeras.
    Kovács F; Adamecz DI; Nagy FI; Papp B; Kiricsi M; Frank É
    Molecules; 2022 Nov; 27(21):. PubMed ID: 36364293
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Efficient access to domain-integrated estradiol-flavone hybrids via the corresponding chalcones and their in vitro anticancer potential.
    Molnár B; Gopisetty MK; Nagy FI; Adamecz DI; Kása Z; Kiricsi M; Frank É
    Steroids; 2022 Nov; 187():109099. PubMed ID: 35970223
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Medicinal-Chemistry-Driven Approach to 2-Substituted Benzoxazole-Estradiol Chimeras: Synthesis, Anticancer Activity, and Early ADME Profile.
    Kovács F; Huliák I; Árva H; Kiricsi M; Erdős D; Kocsis M; Takács G; Balogh GT; Frank É
    ChemMedChem; 2023 Nov; 18(22):e202300352. PubMed ID: 37727903
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Multistep Synthesis and In Vitro Anticancer Evaluation of 2-Pyrazolyl-Estradiol Derivatives, Pyrazolocoumarin-Estradiol Hybrids and Analogous Compounds.
    Molnár B; Gopisetty MK; Adamecz DI; Kiricsi M; Frank É
    Molecules; 2020 Sep; 25(18):. PubMed ID: 32899643
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach.
    Preti D; Romagnoli R; Rondanin R; Cacciari B; Hamel E; Balzarini J; Liekens S; Schols D; Estévez-Sarmiento F; Quintana J; Estévez F
    J Enzyme Inhib Med Chem; 2018 Dec; 33(1):1225-1238. PubMed ID: 30141353
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Biological Activity, Apoptotic Induction and Cell Cycle Arrest of New Hydrazonoyl Halides Derivatives.
    Mohamed MF; Hassaneen HM; Elzayat EM; El-Hallouty SM; El-Manawaty M; Saleh FM; Mohamed Y; El-Zohiry D; Fahmy G; Abdelaal N; Hassanin N; Hossam N
    Anticancer Agents Med Chem; 2019; 19(9):1141-1149. PubMed ID: 30843494
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Development of new estradiol-cationic lipid hybrids: ten-carbon twin chain cationic lipid is a more suitable partner for estradiol to elicit better anticancer activity.
    Sudhakar G; Bathula SR; Banerjee R
    Eur J Med Chem; 2014 Oct; 86():653-63. PubMed ID: 25222876
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and Screening of Pro-apoptotic and Angio-inhibitory Activity of Novel Benzisoxazole Derivatives both In Vitro and In Vivo.
    Byrappa S; Rachaiah K; Kotian SY; Balaraju Y; Prabhuswamimath SC; Rai KML; Salimath BP
    Anticancer Agents Med Chem; 2019; 19(6):827-839. PubMed ID: 30648522
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Anti-Cancer Activity of Novel Dihydrotestosterone-Derived Ring A-Condensed Pyrazoles on Androgen Non-Responsive Prostate Cancer Cell Lines.
    Mótyán G; Gopisetty MK; Kiss-Faludy RE; Kulmány Á; Zupkó I; Frank É; Kiricsi M
    Int J Mol Sci; 2019 May; 20(9):. PubMed ID: 31052484
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Moxifloxacin-isatin Hybrids Tethered by 1,2,3-triazole and their Anticancer Activities.
    Yang M; Liu H; Zhang Y; Wang X; Xu Z
    Curr Top Med Chem; 2020; 20(16):1461-1467. PubMed ID: 31994464
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis, antitumor activity and structure-activity studies of novel pyridoxine-based bioisosteric analogs of estradiol.
    Pugachev MV; Pavelyev RS; Nguyen TNT; Gabbasova RR; Bulatov TM; Iksanova AG; Aljondi B; Bondar OV; Grishaev DY; Yamaleeva ZR; Kataeva ON; Nikishova TV; Balakin KV; Shtyrlin YG
    Bioorg Med Chem; 2021 Jan; 30():115957. PubMed ID: 33373820
    [TBL] [Abstract][Full Text] [Related]  

  • 12. New thieno[3,2-d]pyrimidine-based derivatives: Design, synthesis and biological evaluation as antiproliferative agents, EGFR and ARO inhibitors inducing apoptosis in breast cancer cells.
    Farghaly AM; AboulWafa OM; Baghdadi HH; Abd El Razik HA; Sedra SMY; Shamaa MM
    Bioorg Chem; 2021 Oct; 115():105208. PubMed ID: 34365057
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Hybrids of 4-hydroxy derivatives of goniothalamin and piplartine bearing a diester or a 1,2,3-triazole linker as antiproliferative agents.
    Grigolo TA; Braga CB; Ornelas C; Russowsky D; Ferreira-Silva GA; Ionta M; Pilli RA
    Bioorg Chem; 2021 Nov; 116():105292. PubMed ID: 34509797
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Straightforward synthesis of steroidal selenocyanates through oxidative umpolung selenocyanation of steroids and their antitumor activity.
    Huang Y; Peng Z; Wei M; Pang L; Cheng Y; Xiao JA; Gan C; Cui J
    J Steroid Biochem Mol Biol; 2023 Jan; 225():106203. PubMed ID: 36228841
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and Antitumor Evaluation of Novel Hybrids of Phenylsulfonylfuroxan and Estradiol Derivatives.
    Wan Q; Deng Y; Huang Y; Yu Z; Wang C; Wang K; Dong J; Chen Y
    ChemistryOpen; 2020 Feb; 9(2):176-182. PubMed ID: 32025462
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of novel 6-fluoro-3-(4-piperidinyl)-1,2-benzisoxazole derivatives as antiproliferative agents: a structure-activity relationship study.
    Benaka Prasad SB; Vinaya K; Ananda Kumar CS; Swarup S; Rangappa KS
    Invest New Drugs; 2009 Dec; 27(6):534-42. PubMed ID: 19066725
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties.
    Kiss A; Jójárt R; Mernyák E; Bartha S; Minorics R; Zupkó I; Schneider G
    Steroids; 2021 Dec; 176():108911. PubMed ID: 34499930
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and antiproliferative evaluation of some novel estradiol selenocyanates.
    Huang Y; Peng Z; Wei M; Gan C; Zhang Y; Chen S; Xiao J; Cui J
    Steroids; 2022 May; 181():108992. PubMed ID: 35202703
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design, synthesis, and biologic evaluation of novel chrysin derivatives as cytotoxic agents and caspase-3/7 activators.
    Al-Oudat BA; Alqudah MA; Audat SA; Al-Balas QA; El-Elimat T; Hassan MA; Frhat IN; Azaizeh MM
    Drug Des Devel Ther; 2019; 13():423-433. PubMed ID: 30774307
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and biological evaluation of 13α-estrone derivatives as potential antiproliferative agents.
    Szabó J; Pataki Z; Wölfling J; Schneider G; Bózsity N; Minorics R; Zupkó I; Mernyák E
    Steroids; 2016 Sep; 113():14-21. PubMed ID: 27263437
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.