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3. Mitochondrial Protease ClpP is a Target for the Anticancer Compounds ONC201 and Related Analogues. Graves PR; Aponte-Collazo LJ; Fennell EMJ; Graves AC; Hale AE; Dicheva N; Herring LE; Gilbert TSK; East MP; McDonald IM; Lockett MR; Ashamalla H; Moorman NJ; Karanewsky DS; Iwanowicz EJ; Holmuhamedov E; Graves LM ACS Chem Biol; 2019 May; 14(5):1020-1029. PubMed ID: 31021596 [TBL] [Abstract][Full Text] [Related]
4. ONC201/TIC10 plus TLY012 anti-cancer effects via apoptosis inhibitor downregulation, stimulation of integrated stress response and death receptor DR5 in gastric adenocarcinoma. Parker CS; Zhou L; Prabhu VV; Lee S; Miner TJ; Ross EA; El-Deiry WS Am J Cancer Res; 2023; 13(12):6290-6312. PubMed ID: 38187068 [TBL] [Abstract][Full Text] [Related]
5. ONC201 activates ER stress to inhibit the growth of triple-negative breast cancer cells. Yuan X; Kho D; Xu J; Gajan A; Wu K; Wu GS Oncotarget; 2017 Mar; 8(13):21626-21638. PubMed ID: 28423492 [TBL] [Abstract][Full Text] [Related]
8. ONC201 kills breast cancer cells Greer YE; Porat-Shliom N; Nagashima K; Stuelten C; Crooks D; Koparde VN; Gilbert SF; Islam C; Ubaldini A; Ji Y; Gattinoni L; Soheilian F; Wang X; Hafner M; Shetty J; Tran B; Jailwala P; Cam M; Lang M; Voeller D; Reinhold WC; Rajapakse V; Pommier Y; Weigert R; Linehan WM; Lipkowitz S Oncotarget; 2018 Apr; 9(26):18454-18479. PubMed ID: 29719618 [TBL] [Abstract][Full Text] [Related]
9. EZH2i EPZ-6438 and HDACi vorinostat synergize with ONC201/TIC10 to activate integrated stress response, DR5, reduce H3K27 methylation, ClpX and promote apoptosis of multiple tumor types including DIPG. Zhang Y; Zhou L; Safran H; Borsuk R; Lulla R; Tapinos N; Seyhan AA; El-Deiry WS Neoplasia; 2021 Aug; 23(8):792-810. PubMed ID: 34246076 [TBL] [Abstract][Full Text] [Related]
10. Single agent and synergistic combinatorial efficacy of first-in-class small molecule imipridone ONC201 in hematological malignancies. Prabhu VV; Talekar MK; Lulla AR; Kline CLB; Zhou L; Hall J; Van den Heuvel APJ; Dicker DT; Babar J; Grupp SA; Garnett MJ; McDermott U; Benes CH; Pu JJ; Claxton DF; Khan N; Oster W; Allen JE; El-Deiry WS Cell Cycle; 2018; 17(4):468-478. PubMed ID: 29157092 [TBL] [Abstract][Full Text] [Related]
11. Antitumorigenic effect of combination treatment with ONC201 and TRAIL in endometrial cancer Ray JE; Ralff MD; Jhaveri A; Zhou L; Dicker DT; Ross EA; El-Deiry WS Cancer Biol Ther; 2021 Dec; 22(10-12):554-563. PubMed ID: 34696710 [TBL] [Abstract][Full Text] [Related]
12. Combination of ONC201 and TLY012 induces selective, synergistic apoptosis in vitro and significantly delays PDAC xenograft growth in vivo. Jhaveri AV; Zhou L; Ralff MD; Lee YS; Navaraj A; Carneiro BA; Safran H; Prabhu VV; Ross EA; Lee S; El-Deiry WS Cancer Biol Ther; 2021 Dec; 22(10-12):607-618. PubMed ID: 34856854 [TBL] [Abstract][Full Text] [Related]
13. Dopamine pre-treatment impairs the anti-cancer effect of integrated stress response- and TRAIL pathway-inducing ONC201, ONC206 and ONC212 imipridones in pancreatic, colorectal cancer but not DMG cells. Zhang Y; Tapinos N; Lulla R; El-Deiry WS Am J Cancer Res; 2024; 14(5):2453-2464. PubMed ID: 38859853 [TBL] [Abstract][Full Text] [Related]
14. Anti-Tumor and Anti-Invasive Effects of ONC201 on Ovarian Cancer Cells and a Transgenic Mouse Model of Serous Ovarian Cancer. Fan Y; Wang J; Fang Z; Pierce SR; West L; Staley A; Tucker K; Yin Y; Sun W; Kong W; Prabhu V; Allen JE; Zhou C; Bae-Jump VL Front Oncol; 2022; 12():789450. PubMed ID: 35372029 [TBL] [Abstract][Full Text] [Related]
15. ONC201 induces the unfolded protein response (UPR) in high- and low-grade ovarian carcinoma cell lines and leads to cell death regardless of platinum sensitivity. Rumman M; Buck S; Polin L; Dzinic S; Boerner J; Winer IS Cancer Med; 2021 May; 10(10):3373-3387. PubMed ID: 33932119 [TBL] [Abstract][Full Text] [Related]
16. Preclinical evaluation of the imipridone family, analogs of clinical stage anti-cancer small molecule ONC201, reveals potent anti-cancer effects of ONC212. Wagner J; Kline CL; Ralff MD; Lev A; Lulla A; Zhou L; Olson GL; Nallaganchu BR; Benes CH; Allen JE; Prabhu VV; Stogniew M; Oster W; El-Deiry WS Cell Cycle; 2017 Oct; 16(19):1790-1799. PubMed ID: 28489985 [TBL] [Abstract][Full Text] [Related]
17. Small-Molecule ONC201/TIC10 Targets Chemotherapy-Resistant Colorectal Cancer Stem-like Cells in an Akt/Foxo3a/TRAIL-Dependent Manner. Prabhu VV; Allen JE; Dicker DT; El-Deiry WS Cancer Res; 2015 Apr; 75(7):1423-32. PubMed ID: 25712124 [TBL] [Abstract][Full Text] [Related]
18. ONC201 kills solid tumor cells by triggering an integrated stress response dependent on ATF4 activation by specific eIF2α kinases. Kline CL; Van den Heuvel AP; Allen JE; Prabhu VV; Dicker DT; El-Deiry WS Sci Signal; 2016 Feb; 9(415):ra18. PubMed ID: 26884600 [TBL] [Abstract][Full Text] [Related]
19. Caseinolytic protease P (CLPP) activated by ONC201 inhibits proliferation and promotes apoptosis in human epithelial ovarian cancer cells by inducing mitochondrial dysfunction. Kou X; Ding H; Li L; Chao H Ann Transl Med; 2021 Sep; 9(18):1463. PubMed ID: 34734015 [TBL] [Abstract][Full Text] [Related]
20. Potent preclinical sensitivity to imipridone-based combination therapies in oncohistone H3K27M-mutant diffuse intrinsic pontine glioma is associated with induction of the integrated stress response, TRAIL death receptor DR5, reduced ClpX and apoptosis. Borsuk R; Zhou L; Chang WI; Zhang Y; Sharma A; Prabhu VV; Tapinos N; Lulla RR; El-Deiry WS Am J Cancer Res; 2021; 11(9):4607-4623. PubMed ID: 34659909 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]