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6. Next generation GLP-1/GIP/glucagon triple agonists normalize body weight in obese mice. Knerr PJ; Mowery SA; Douros JD; Premdjee B; Hjøllund KR; He Y; Kruse Hansen AM; Olsen AK; Perez-Tilve D; DiMarchi RD; Finan B Mol Metab; 2022 Sep; 63():101533. PubMed ID: 35809773 [TBL] [Abstract][Full Text] [Related]
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8. GLP-1 and GIP receptor signaling in beta cells - A review of receptor interactions and co-stimulation. Mayendraraj A; Rosenkilde MM; Gasbjerg LS Peptides; 2022 May; 151():170749. PubMed ID: 35065096 [TBL] [Abstract][Full Text] [Related]
9. Genetic and biased agonist-mediated reductions in β-arrestin recruitment prolong cAMP signaling at glucagon family receptors. Jones B; McGlone ER; Fang Z; Pickford P; Corrêa IR; Oishi A; Jockers R; Inoue A; Kumar S; Görlitz F; Dunsby C; French PMW; Rutter GA; Tan T; Tomas A; Bloom SR J Biol Chem; 2021; 296():100133. PubMed ID: 33268378 [TBL] [Abstract][Full Text] [Related]
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11. The GIP receptor displays higher basal activity than the GLP-1 receptor but does not recruit GRK2 or arrestin3 effectively. Al-Sabah S; Al-Fulaij M; Shaaban G; Ahmed HA; Mann RJ; Donnelly D; Bünemann M; Krasel C PLoS One; 2014; 9(9):e106890. PubMed ID: 25191754 [TBL] [Abstract][Full Text] [Related]
12. Tirzepatide modulates the regulation of adipocyte nutrient metabolism through long-acting activation of the GIP receptor. Regmi A; Aihara E; Christe ME; Varga G; Beyer TP; Ruan X; Beebe E; O'Farrell LS; Bellinger MA; Austin AK; Lin Y; Hu H; Konkol DL; Wojnicki S; Holland AK; Friedrich JL; Brown RA; Estelle AS; Badger HS; Gaidosh GS; Kooijman S; Rensen PCN; Coskun T; Thomas MK; Roell W Cell Metab; 2024 Jul; 36(7):1534-1549.e7. PubMed ID: 38878772 [TBL] [Abstract][Full Text] [Related]
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14. A Dual GLP-1/GIP Receptor Agonist Does Not Antagonize Glucagon at Its Receptor but May Act as a Biased Agonist at the GLP-1 Receptor. Al-Zamel N; Al-Sabah S; Luqmani Y; Adi L; Chacko S; Schneider TD; Krasel C Int J Mol Sci; 2019 Jul; 20(14):. PubMed ID: 31330984 [TBL] [Abstract][Full Text] [Related]
15. Human Epicardial Fat Expresses Glucagon-Like Peptide 1 and 2 Receptors Genes. Iacobellis G; Camarena V; Sant DW; Wang G Horm Metab Res; 2017 Aug; 49(8):625-630. PubMed ID: 28514806 [TBL] [Abstract][Full Text] [Related]
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17. A comparative transcriptomic analysis of glucagon-like peptide-1 receptor- and glucose-dependent insulinotropic polypeptide receptor-expressing cells in the hypothalamus. Smith C; Patterson-Cross R; Woodward O; Lewis J; Chiarugi D; Merkle F; Gribble F; Reimann F; Adriaenssens A Appetite; 2022 Jul; 174():106022. PubMed ID: 35430298 [TBL] [Abstract][Full Text] [Related]
18. The interplay of glucose-dependent insulinotropic polypeptide in adipose tissue. Kagdi S; Lyons SA; Beaudry JL J Endocrinol; 2024 Jun; 261(3):. PubMed ID: 38579777 [TBL] [Abstract][Full Text] [Related]
19. Targeting the GIPR for obesity: To agonize or antagonize? Potential mechanisms. Campbell JE Mol Metab; 2021 Apr; 46():101139. PubMed ID: 33290902 [TBL] [Abstract][Full Text] [Related]
20. Discovery of a potent GIPR peptide antagonist that is effective in rodent and human systems. Yang B; Gelfanov VM; El K; Chen A; Rohlfs R; DuBois B; Kruse Hansen AM; Perez-Tilve D; Knerr PJ; D'Alessio D; Campbell JE; Douros JD; Finan B Mol Metab; 2022 Dec; 66():101638. PubMed ID: 36400403 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]