These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

58 related articles for article (PubMed ID: 3775387)

  • 1. Human alpha- and gamma-thrombin inhibition by trypsin inhibitors supports predictions from molecular graphics experiments.
    Sugawara Y; Birktoft JJ; Berliner LJ
    Semin Thromb Hemost; 1986 Jul; 12(3):209-12. PubMed ID: 3775387
    [No Abstract]   [Full Text] [Related]  

  • 2. Inhibition of bovine beta-trypsin, human alpha-thrombin and porcine pancreatic beta-kallikrein-B by benzamidine and its bis-, tris- and tetra-derivatives: thermodynamic and molecular modeling study.
    Menegatti E; Ferroni R; Nastruzzi C; Bortolotti F; Scalia S; Amiconi G; Bolognesi M; Coletta M; Onesti S; Fruttero R
    Farmaco; 1991 Nov; 46(11):1297-310. PubMed ID: 1811616
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Enzyme binding selectivity prediction: alpha-thrombin vs trypsin inhibition.
    Mlinsek G; Novic M; Kotnik M; Solmajer T
    J Chem Inf Comput Sci; 2004; 44(5):1872-82. PubMed ID: 15446847
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Highly selective mechanism-based thrombin inhibitors: structures of thrombin and trypsin inhibited with rigid peptidyl aldehydes.
    Krishnan R; Zhang E; Hakansson K; Arni RK; Tulinsky A; Lim-Wilby MS; Levy OE; Semple JE; Brunck TK
    Biochemistry; 1998 Sep; 37(35):12094-103. PubMed ID: 9724521
    [TBL] [Abstract][Full Text] [Related]  

  • 5. N alpha-arylsulfonyl-omega-amidinophenyl-alpha-aminoalkyl-carboxylic acid amides as specific thrombin inhibitors.
    Stürzebecher J
    Folia Haematol Int Mag Klin Morphol Blutforsch; 1982; 109(1):83-8. PubMed ID: 6177613
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Molecular design and characterization of an alpha-thrombin inhibitor containing a novel P1 moiety.
    Malikayil JA; Burkhart JP; Schreuder HA; Broersma RJ; Tardif C; Kutcher LW; Mehdi S; Schatzman GL; Neises B; Peet NP
    Biochemistry; 1997 Feb; 36(5):1034-40. PubMed ID: 9033393
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, synthesis and molecular modelling of 1-amidinopiperidine thrombin inhibitors.
    Smolnikar I; Perdih A; Stegnar M; Prezelj A; Solmajer T; Urleb U; Obreza A
    Pharmazie; 2007 Apr; 62(4):243-54. PubMed ID: 17484277
    [TBL] [Abstract][Full Text] [Related]  

  • 8. [Synthetic inhibitors of serine proteinases. 12. The inhibition of trypsin, plasmin and thrombin by 3-[amidinophenyl]-1-phenyl-propanone-(1) with substituents in the aliphatic intermediate chain].
    Walsmann P; Griessmann R; Horn H; Markwardt F; Richter P; Stürzebecher J; Wagner G
    Pharmazie; 1976 Jun; 31(6):410-1. PubMed ID: 134380
    [No Abstract]   [Full Text] [Related]  

  • 9. [Inhibition of thrombin, plasmin and trypsin effect by alkyl- and alkoxybenzamidine].
    Markwardt F; Walsmann P; Landmann H
    Pharmazie; 1970 Sep; 25(9):551-4. PubMed ID: 4249689
    [No Abstract]   [Full Text] [Related]  

  • 10. [The modification of the effect of trypsin on blood coagulation by natural and synthetic trypsin and thrombin inhibitors].
    Landman H; Markwardt F; Perlewitz J
    Thromb Diath Haemorrh; 1969 Dec; 22(3):552-68. PubMed ID: 5382290
    [No Abstract]   [Full Text] [Related]  

  • 11. In-depth study of tripeptide-based alpha-ketoheterocycles as inhibitors of thrombin. Effective utilization of the S1' subsite and its implications to structure-based drug design.
    Costanzo MJ; Almond HR; Hecker LR; Schott MR; Yabut SC; Zhang HC; Andrade-Gordon P; Corcoran TW; Giardino EC; Kauffman JA; Lewis JM; de Garavilla L; Haertlein BJ; Maryanoff BE
    J Med Chem; 2005 Mar; 48(6):1984-2008. PubMed ID: 15771442
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Selectivity of neutral/weakly basic P1 group inhibitors of thrombin and trypsin by a molecular dynamics study.
    Wu EL; Han K; Zhang JZ
    Chemistry; 2008; 14(28):8704-14. PubMed ID: 18680136
    [TBL] [Abstract][Full Text] [Related]  

  • 13. [Synthetic inhibitors of serine proteinases. Part 26: Inhibition of trypsin, plasmin and thrombin by amides of N alpha-arylsulfonylated 2-amino-4-(4-amidino-phenyl) butyric acid and 2-amino-5-amidinophenyl valeric acids (author's transl)].
    Stürzebecher J; Markwardt F; Vieweg H; Wagner G; Walsmann P
    Pharmazie; 1982 Apr; 37(4):281-3. PubMed ID: 6212947
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Alpha-1-antitrypsin. 3. Inhibition of trypsin, thrombin, plasmin and leucoproteinases.
    Tan BH; Gans H
    Pharm Weekbl; 1969 Jun; 104(26):717-25. PubMed ID: 4239740
    [No Abstract]   [Full Text] [Related]  

  • 15. Molecular modeling and 3D-QSAR studies on the interaction mechanism of tripeptidyl thrombin inhibitors with human alpha-thrombin.
    Jiang H; Chen K; Tang Y; Chen J; Li Q; Wang Q; Ji R
    J Med Chem; 1997 Sep; 40(19):3085-90. PubMed ID: 9301672
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Quantitative structure-activity relationships and molecular graphics in ligand receptor interactions: amidine inhibition of trypsin.
    Recanatini M; Klein T; Yang CZ; McClarin J; Langridge R; Hansch C
    Mol Pharmacol; 1986 Apr; 29(4):436-46. PubMed ID: 3702862
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Human alpha-thrombin inhibition by the active site titrant N alpha-(N,N-dimethylcarbamoyl)-alpha-azalysine p-nitrophenyl ester: a comparative kinetic and X-ray crystallographic study.
    Nardini M; Pesce A; Rizzi M; Casale E; Ferraccioli R; Balliano G; Milla P; Ascenzi P; Bolognesi M
    J Mol Biol; 1996 May; 258(5):851-9. PubMed ID: 8637015
    [TBL] [Abstract][Full Text] [Related]  

  • 18. [Synthetic inhibitors of serine proteinases. Part 25: Inhibition of trypsin, plasmin and thrombin by amides of N alpha-substituted amidinophenylalanines and 3-amidinophenyl-3-aminopropionic acids (author's transl)].
    Stürzebecher J; Horn H; Markwardt F; Wagner G; Walsmann P
    Pharmazie; 1981 Sep; 36(9):639-41. PubMed ID: 6458047
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Novel potent and selective thrombin inhibitors based on a central 1,4-benzoxazin-3(4H)-one scaffold.
    Ilas J; Tomasić T; Kikelj D
    J Med Chem; 2008 May; 51(9):2863-7. PubMed ID: 18412326
    [TBL] [Abstract][Full Text] [Related]  

  • 20. [Synthetic inhibitors of serine proteinases. Part 24: Inhibition of trypsin, plasmin and thrombin by cyclic amides of N alpha-arylsulfonylamidinophenyl-glycines (author's transl)].
    Stürzebecher J; Markwardt F; Voigt B; Wagner G; Walsmann P
    Pharmazie; 1981; 36(7):501-2. PubMed ID: 6456466
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 3.