These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
9. The drug-specific properties of hypoxia-inducible factor-prolyl hydroxylase inhibitors in mice reveal a significant contribution of the kidney compared to the liver to erythropoietin induction. Nakai T; Saigusa D; Kato K; Fukuuchi T; Koshiba S; Yamamoto M; Suzuki N Life Sci; 2024 Jun; 346():122641. PubMed ID: 38614299 [TBL] [Abstract][Full Text] [Related]
10. Discovery of DS-1093a: An oral hypoxia-inducible factor prolyl hydroxylase inhibitor for the treatment of renal anemia. Tanaka N; Fukuda T; Takano R; Sasaki K; Tsuji T; Goto R; Kuribayashi T; Yamaguchi K; Niitsu Y; Ishii K; Hashimoto M; Takahashi S; Obayashi H Bioorg Med Chem Lett; 2024 Oct; 111():129891. PubMed ID: 39019240 [TBL] [Abstract][Full Text] [Related]
11. Discovery of novel 2-[(4-hydroxy-6-oxo-2,3-dihydro-1H-pyridine-5-carbonyl)amino]acetic acid derivatives as HIF prolyl hydroxylase inhibitors for treatment of renal anemia. Hamada M; Takayama T; Shibata T; Hiratate A; Takahashi M; Yashiro M; Takayama N; Okumura-Kitajima L; Koretsune H; Kajiyama H; Naruse T; Kato S; Takano H; Kakinuma H Bioorg Med Chem Lett; 2018 Jun; 28(10):1725-1730. PubMed ID: 29681433 [TBL] [Abstract][Full Text] [Related]
12. Photoactivatable Prolyl Hydroxylase 2 Inhibitors for Stabilizing the Hypoxia-Inducible Factor with Light. Li Z; Su K; Jiang Z; Yu Y; You Q; Zhang X J Med Chem; 2019 Aug; 62(16):7583-7588. PubMed ID: 31244107 [TBL] [Abstract][Full Text] [Related]
13. A small-molecule inhibitor of hypoxia-inducible factor prolyl hydroxylase improves obesity, nephropathy and cardiomyopathy in obese ZSF1 rats. Signore PE; Guo G; Wei Z; Zhang W; Lin A; Del Balzo U PLoS One; 2021; 16(8):e0255022. PubMed ID: 34339435 [TBL] [Abstract][Full Text] [Related]
14. The selective prolyl hydroxylase inhibitor IOX5 stabilizes HIF-1α and compromises development and progression of acute myeloid leukemia. Lawson H; Holt-Martyn JP; Dembitz V; Kabayama Y; Wang LM; Bellani A; Atwal S; Saffoon N; Durko J; van de Lagemaat LN; De Pace AL; Tumber A; Corner T; Salah E; Arndt C; Brewitz L; Bowen M; Dubusse L; George D; Allen L; Guitart AV; Fung TK; So CWE; Schwaller J; Gallipoli P; O'Carroll D; Schofield CJ; Kranc KR Nat Cancer; 2024 Jun; 5(6):916-937. PubMed ID: 38637657 [TBL] [Abstract][Full Text] [Related]
15. Click Chemistry-Based Discovery of [3-Hydroxy-5-(1 H-1,2,3-triazol-4-yl)picolinoyl]glycines as Orally Active Hypoxia-Inducing Factor Prolyl Hydroxylase Inhibitors with Favorable Safety Profiles for the Treatment of Anemia. Wu Y; Jiang Z; Li Z; Gu J; You Q; Zhang X J Med Chem; 2018 Jun; 61(12):5332-5349. PubMed ID: 29856623 [TBL] [Abstract][Full Text] [Related]
16. HIF stabilizers in the management of renal anemia: from bench to bedside to pediatrics. Kular D; Macdougall IC Pediatr Nephrol; 2019 Mar; 34(3):365-378. PubMed ID: 29569190 [TBL] [Abstract][Full Text] [Related]
17. Molecular mechanisms of action and therapeutic uses of pharmacological inhibitors of HIF-prolyl 4-hydroxylases for treatment of ischemic diseases. Selvaraju V; Parinandi NL; Adluri RS; Goldman JW; Hussain N; Sanchez JA; Maulik N Antioxid Redox Signal; 2014 Jun; 20(16):2631-65. PubMed ID: 23992027 [TBL] [Abstract][Full Text] [Related]
18. Protein Hydroxylation by Hypoxia-Inducible Factor (HIF) Hydroxylases: Unique or Ubiquitous? Strowitzki MJ; Cummins EP; Taylor CT Cells; 2019 Apr; 8(5):. PubMed ID: 31035491 [TBL] [Abstract][Full Text] [Related]
20. Effects of hypoxia-inducible factor prolyl hydroxylase inhibitors on iron regulation in non-dialysis-dependent chronic kidney disease patients with anemia: A systematic review and meta-analysis. Li J; Xie QH; You L; Xu NX; Hao CM Pharmacol Res; 2021 Jan; 163():105256. PubMed ID: 33086081 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]