171 related articles for article (PubMed ID: 38576720)
1. Cell penetration of oxadiazole-containing macrocycles.
Huh S; Batistatou N; Wang J; Saunders GJ; Kritzer JA; Yudin AK
RSC Chem Biol; 2024 Apr; 5(4):328-334. PubMed ID: 38576720
[TBL] [Abstract][Full Text] [Related]
2. Oxadiazole grafts in peptide macrocycles.
Frost JR; Scully CC; Yudin AK
Nat Chem; 2016 Dec; 8(12):1105-1111. PubMed ID: 27874866
[TBL] [Abstract][Full Text] [Related]
3. Beyond Rule-of-five: Permeability Assessment of Semipeptidic Macrocycles.
L'Exact M; Comeau C; Bourhis A; Boisvert O; Fröhlich U; Létourneau D; Marsault É; Lavigne P; Grandbois M; Boudreault PL
Biochim Biophys Acta Biomembr; 2023 Oct; 1865(7):184196. PubMed ID: 37400050
[TBL] [Abstract][Full Text] [Related]
4. Label-free quantification of passive membrane permeability of cyclic peptides across lipid bilayers: penetration speed of cyclosporin A across lipid bilayers.
Ono T; Tabata KV; Goto Y; Saito Y; Suga H; Noji H; Morimoto J; Sando S
Chem Sci; 2023 Jan; 14(2):345-349. PubMed ID: 36687349
[TBL] [Abstract][Full Text] [Related]
5. Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure.
Fouché M; Schäfer M; Berghausen J; Desrayaud S; Blatter M; Piéchon P; Dix I; Martin Garcia A; Roth HJ
ChemMedChem; 2016 May; 11(10):1048-59. PubMed ID: 27154275
[TBL] [Abstract][Full Text] [Related]
6. Cell Penetration Profiling Using the Chloroalkane Penetration Assay.
Peraro L; Deprey KL; Moser MK; Zou Z; Ball HL; Levine B; Kritzer JA
J Am Chem Soc; 2018 Sep; 140(36):11360-11369. PubMed ID: 30118219
[TBL] [Abstract][Full Text] [Related]
7. Highly Conformationally Restricted Cyclopropane Tethers with Three-Dimensional Structural Diversity Drastically Enhance the Cell Permeability of Cyclic Peptides.
Matsui K; Kido Y; Watari R; Kashima Y; Yoshida Y; Shuto S
Chemistry; 2017 Mar; 23(13):3034-3041. PubMed ID: 27878880
[TBL] [Abstract][Full Text] [Related]
8. Property-Driven Development of Passively Permeable Macrocyclic Scaffolds Using Heterocycles.
Saunders GJ; Yudin AK
Angew Chem Int Ed Engl; 2022 Aug; 61(33):e202206866. PubMed ID: 35687524
[TBL] [Abstract][Full Text] [Related]
9. Understanding Cell Penetration of Cyclic Peptides.
Dougherty PG; Sahni A; Pei D
Chem Rev; 2019 Sep; 119(17):10241-10287. PubMed ID: 31083977
[TBL] [Abstract][Full Text] [Related]
10. Lessons for Oral Bioavailability: How Conformationally Flexible Cyclic Peptides Enter and Cross Lipid Membranes.
Linker SM; Schellhaas C; Kamenik AS; Veldhuizen MM; Waibl F; Roth HJ; Fouché M; Rodde S; Riniker S
J Med Chem; 2023 Feb; 66(4):2773-2788. PubMed ID: 36762908
[TBL] [Abstract][Full Text] [Related]
11. Achieving enhanced cell penetration of short conformationally constrained peptides through amphiphilicity tuning.
Tian Y; Zeng X; Li J; Jiang Y; Zhao H; Wang D; Huang X; Li Z
Chem Sci; 2017 Nov; 8(11):7576-7581. PubMed ID: 29568420
[TBL] [Abstract][Full Text] [Related]
12. The penetrating properties of the tumor homing peptide LyP-1 in model lipid membranes.
Ciobanasu C; Dragomir I; Apetrei A
J Pept Sci; 2019 Mar; 25(3):e3145. PubMed ID: 30588706
[TBL] [Abstract][Full Text] [Related]
13. Development of Endocyclic Control Elements for Peptide Macrocycles.
Appavoo SD; Kaji T; Frost JR; Scully CCG; Yudin AK
J Am Chem Soc; 2018 Jul; 140(28):8763-8770. PubMed ID: 29920073
[TBL] [Abstract][Full Text] [Related]
14. Insights on Structure-Passive Permeability Relationship in Pyrrole and Furan-Containing Macrocycles.
Ly HM; Desgagné M; Nguyen DT; Comeau C; Froehlich U; Marsault É; Boudreault PL
J Med Chem; 2024 Mar; 67(5):3711-3726. PubMed ID: 38417040
[TBL] [Abstract][Full Text] [Related]
15. Quantitative measurement of cytosolic penetration using the chloroalkane penetration assay.
Deprey K; Kritzer JA
Methods Enzymol; 2020; 641():277-309. PubMed ID: 32713526
[TBL] [Abstract][Full Text] [Related]
16. Optimization of Cyclic Peptide Property Using Chromatographic Capacity Factor on Permeability of Passive Cell Membrane and Human Induced Pluripotent Stem Cell-Derived Intestinal Membrane.
Watanabe A; Uehara S; Akazawa T; Fujiu M
J Pharm Sci; 2022 Jul; 111(7):1879-1886. PubMed ID: 35385719
[TBL] [Abstract][Full Text] [Related]
17. Structure-Permeability Relationship of Semipeptidic Macrocycles-Understanding and Optimizing Passive Permeability and Efflux Ratio.
Le Roux A; Blaise É; Boudreault PL; Comeau C; Doucet A; Giarrusso M; Collin MP; Neubauer T; Kölling F; Göller AH; Seep L; Tshitenge DT; Wittwer M; Kullmann M; Hillisch A; Mittendorf J; Marsault E
J Med Chem; 2020 Jul; 63(13):6774-6783. PubMed ID: 32453569
[TBL] [Abstract][Full Text] [Related]
18. Heterocycles: Versatile control elements in bioactive macrocycles.
Soor HS; Appavoo SD; Yudin AK
Bioorg Med Chem; 2018 Jun; 26(10):2774-2779. PubMed ID: 29735427
[TBL] [Abstract][Full Text] [Related]
19. Enantiomeric cyclic peptides with different Caco-2 permeability suggest carrier-mediated transport.
Marelli UK; Bezençon J; Puig E; Ernst B; Kessler H
Chemistry; 2015 May; 21(22):8023-7. PubMed ID: 25917866
[TBL] [Abstract][Full Text] [Related]
20. Parallel Screening Using the Chloroalkane Penetration Assay Reveals Structure-Penetration Relationships.
Mientkiewicz KM; Peraro L; Kritzer JA
ACS Chem Biol; 2021 Jul; 16(7):1184-1190. PubMed ID: 34224243
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
