BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

191 related articles for article (PubMed ID: 4629015)

  • 1. Synthesis of some bis(2,4-diaminopyrimidines) and bis(2,4-diaminoquinazolines) as potential antimalarial agents.
    Hynes JB; Gratz RF; Ashton WT
    J Med Chem; 1972 Dec; 15(12):1332-3. PubMed ID: 4629015
    [No Abstract]   [Full Text] [Related]  

  • 2. 2,4-Diaminothieno(2,3-d)pyrimidines as antifolates and antimalarials. 1. Synthesis of 2,4-diamino-5,6,7,8-tetrahydrothianaphthena(2,3-d)pyrimidines and related compounds.
    Rosowsky A; Chaykovsky M; Chen KK; Lin M; Modest EJ
    J Med Chem; 1973 Mar; 16(3):185-8. PubMed ID: 4632693
    [No Abstract]   [Full Text] [Related]  

  • 3. Synthesis of 5-substituted quinazolines as potential antimalarial agents.
    Ashton WT; Hynes JB
    J Med Chem; 1973 Nov; 16(11):1233-7. PubMed ID: 4583883
    [No Abstract]   [Full Text] [Related]  

  • 4. Folate antagonists. 9. 2,4-Diamino-6-((aralkyl)alkylamino)quinazolines, a potent class of antimetabolites with prodigious antimalarial effects.
    Elslager EF; Bird OD; Clarke J; Perricone SC; Worth DF
    J Med Chem; 1972 Nov; 15(11):1138-46. PubMed ID: 4631920
    [No Abstract]   [Full Text] [Related]  

  • 5. 2,4-Diaminothieno(2,3-d)pyrimidines as antifolates and antimalarials. 2. Synthesis of 2,4-diaminopyrido(4',3':4,5)thieno(2,3-d)pyrimidines and 2,4-diamino-8H-thiopyrano(4',3':4,5)thieno(2,3-d)pyrimidines.
    Chaykovsky M; Lin M; Rosowsky A; Modest EJ
    J Med Chem; 1973 Mar; 16(3):188-91. PubMed ID: 4632694
    [No Abstract]   [Full Text] [Related]  

  • 6. 2,4-Diaminothieno(2,3-d)pyrimidines as antifolates and antimalarials. 3. Synthesis of 5,6-disubstituted derivatives and related tetracyclic analogs.
    Rosowsky A; Chen KK; Lin M
    J Med Chem; 1973 Mar; 16(3):191-4. PubMed ID: 4632695
    [No Abstract]   [Full Text] [Related]  

  • 7. Effect of trifluoromethoxy, chlorodifluoromethoxy, and trifluoromethyl on the antimalarial activity of 5-benzyl- and 5-phenyl-2,4-diaminopyrimidines.
    Stogryn EL
    J Med Chem; 1973 Dec; 16(12):1399-401. PubMed ID: 4587856
    [No Abstract]   [Full Text] [Related]  

  • 8. Synthesis and evaluation of 6-arylactamido-2,4-diaminoquinazolines and related compounds as folic acid antagonists.
    Hynes JB; Ashton WT
    J Med Chem; 1975 Mar; 18(3):263-5. PubMed ID: 1094114
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Folate antagonists. 12. Antimalarial and antibacterial effects of 2,4-diamino-6-[(aralkyl and alicyclid)thio-, sulfinyl-, and sulfonyl]quinazolines.
    Elslager EF; Davoll J; Jacob P; Johnson AM; Johnson J; Werbel LM
    J Med Chem; 1978 Jul; 21(7):639-43. PubMed ID: 97382
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Quinazolines. 12. 1,3-Diaminobenzo(f)quinazolines containing long-chain alkyl or chloro substituents on the central ring. Synthesis and biological evaluation as candidate antifolate and antimalarial agents.
    Rosowsky A; Huang PC; Papathanasopoulos N; Modest EJ
    J Med Chem; 1974 Nov; 17(11):1217-22. PubMed ID: 4606974
    [No Abstract]   [Full Text] [Related]  

  • 11. Synthesis of analogs of 6-arylthio-, 6-arylsulfinyl-, and 6-arylsulfonyl-2, 4-diaminoquinazolines as potential antimalarial agents.
    Hynes JB; Ashton WT; Merriman HG; Walker FC
    J Med Chem; 1974 Jul; 17(7):682-4. PubMed ID: 4600305
    [No Abstract]   [Full Text] [Related]  

  • 12. Folate antagonists. 4. Antimalarial and antimetabolite effects of 2,4-diamino-6-((benzyl)amino)pyrido(2,3-d)-pyrimidines.
    Davoll J; Clarke J; Elslager EF
    J Med Chem; 1972 Aug; 15(8):837-9. PubMed ID: 5044297
    [No Abstract]   [Full Text] [Related]  

  • 13. Inhibition of mammalian dihydrofolate reductase by selected 2,4-diaminiquinazolines and related compounds.
    Richter WE; McCormack JJ
    J Med Chem; 1974 Sep; 17(9):943-7. PubMed ID: 4213189
    [No Abstract]   [Full Text] [Related]  

  • 14. Folate antagonists. 3. 2,4-Diamino-6-(heterocyclic)quinazolines, a novel class of antimetabolites with potent antimalarial and antibacterial activity.
    Elslager EF; Clarke J; Werbel LM; Worth DF; Davoll J
    J Med Chem; 1972 Aug; 15(8):827-36. PubMed ID: 4625530
    [No Abstract]   [Full Text] [Related]  

  • 15. Quinazolines as inhibitors of dihydrofolate reductase. 3. Analogs of pteroic and isopteroic acids.
    Hynes JB; Buck JM; D'Souza L; Freisheim JH
    J Med Chem; 1975 Dec; 18(12):1191-4. PubMed ID: 811798
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Folate antagonists. 13. 2,4-Diamino-6-](alpha,alpha,alpha-trifluoro-m-tolyl)thio]quinazoline and related 2,4-diamino-6-[(phenyl- and naphthyl)thio]quinazolines, a unique class of antimetabolites with extraordinary antimalarial and antibacterial effects.
    Elslager EF; Jacob P; Johnson J; Werbel LM; Worth DF; Rane L
    J Med Chem; 1978 Oct; 21(10):1059-70. PubMed ID: 102792
    [TBL] [Abstract][Full Text] [Related]  

  • 17. [Studies on antimalarials. XV. Synthesis and antimalarial activities of some bis(2,4-diaminoquinazol-6-yl-substituted aminomethyl) aromatic derivatives].
    Zhou WC; Dai ZR; Ding YL; Zhang XP
    Yao Xue Xue Bao; 1985 Jul; 20(7):536-41. PubMed ID: 3913278
    [No Abstract]   [Full Text] [Related]  

  • 18. Pteridines. 2. New 6,7-disubstituted pteridines as potential antimalarial and antitumor agents.
    Rosowsky A; Chaykovsky M; Lin M; Modest EJ
    J Med Chem; 1973 Aug; 16(8):869-75. PubMed ID: 4200929
    [No Abstract]   [Full Text] [Related]  

  • 19. Synthesis of potential antimalarial agents. Preparation of some 6-amino-5,8-dimethoxyquinolines and the corresponding 6-amino-5,8-quinolinediones.
    Temple C; Rose JD; Montgomery JA
    J Med Chem; 1974 Jun; 17(6):615-9. PubMed ID: 4598023
    [No Abstract]   [Full Text] [Related]  

  • 20. Synthesis of 2,4-diamino-5-(4-arylthiophenyl)-and 5-(4-arylsulfonylphenyl)pyrimidines as antimalarials.
    Das BP; Boykin DW
    J Med Chem; 1974 Mar; 17(3):372-4. PubMed ID: 4590245
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 10.