BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

128 related articles for article (PubMed ID: 6142117)

  • 1. (Imidazolylphenyl)formamidines. A structurally novel class of potent histamine H2 receptor antagonists.
    Donetti A; Cereda E; Bellora E; Gallazzi A; Bazzano C; Vanoni P; Del Soldato P; Micheletti R; Pagani F; Giachetti A
    J Med Chem; 1984 Mar; 27(3):380-6. PubMed ID: 6142117
    [TBL] [Abstract][Full Text] [Related]  

  • 2. N-(fluoroethyl)(imidazolylphenyl)formamidines. The issue of the active species of mifentidine.
    Donetti A; Cereda E; Ezhaya A; Micheletti R
    J Med Chem; 1989 May; 32(5):957-61. PubMed ID: 2565401
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Pharmacology of mifentidine, a novel H2-receptor antagonist.
    Pagani F; Micheletti R; Brambilla A; Schiavone A; Montagna E; Ciprandi C; Giachetti A
    Arzneimittelforschung; 1985; 35(1A):451-5. PubMed ID: 2859036
    [TBL] [Abstract][Full Text] [Related]  

  • 4. A comparison of some of the pharmacological properties of etintidine, a new histamine H2-receptor antagonist, with those of cimetidine, ranitidine and tiotidine.
    Cavanagh RL; Usakewicz JJ; Buyniski JP
    J Pharmacol Exp Ther; 1983 Jan; 224(1):171-9. PubMed ID: 6129316
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Substituent effect on the stereochemistry of H2-receptor antagonists of the phenylformamidine series. A conformation-dependent mode of interaction with the H2 receptor.
    Donetti A; Bastiaans HM; Kramer K; Bietti G; Cereda E; Dubini E; Mondoni M; Bast A; Timmerman H
    J Med Chem; 1991 Jun; 34(6):1772-6. PubMed ID: 1676425
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Evaluation of novel compounds interacting with H2-histamine receptors: effect on histamine-sensitive adenylate cyclase activity in guinea-pig gastric mucosa.
    Micheletti R; Oliva D; Belfiore P; Giachetti A; Nicosia S
    Agents Actions; 1985 Jul; 16(5):291-4. PubMed ID: 2864816
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and assessment of formamidines as new histamine H2-receptor antagonists.
    Anglada L; Raga M; Márquez M; Sacristán A; Castelló JM; Ortiz JA
    Arzneimittelforschung; 1997 Apr; 47(4A):431-4. PubMed ID: 9205738
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Bioisosteric prototype design of biaryl imidazolyl and triazolyl competitive histamine H2-receptor antagonists.
    Lipinski CA; LaMattina JL; Oates PJ
    J Med Chem; 1986 Nov; 29(11):2154-63. PubMed ID: 2878075
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Histamine H2 receptor antagonists. 1. Synthesis of N-cyano and N-carbamoyl amidine derivatives and their biological activities.
    Yanagisawa I; Hirata Y; Ishii Y
    J Med Chem; 1984 Jul; 27(7):849-57. PubMed ID: 6145803
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Gastric antisecretory effect of FRG-8813, a new histamine H2 receptor antagonist, in rats and dogs.
    Shibata M; Yamaura T; Inaba N; Onodera S; Chida Y; Ohnishi H
    Eur J Pharmacol; 1993 Apr; 235(2-3):245-53. PubMed ID: 8099553
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Conformational requirements for histamine H2-receptor inhibitors: a structure-activity study of phenylene analogues related to cimetidine and tiotidine.
    Hoffman JM; Pietruszkiewicz AM; Habecker CN; Phillips BT; Bolhofer WA; Cragoe EJ; Torchiana ML; Lumma WC; Baldwin JJ
    J Med Chem; 1983 Feb; 26(2):140-4. PubMed ID: 6131129
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Pharmacological profile of mifentidine: a novel H2-receptor antagonist.
    Giachetti A; Pagani F; Micheletti R; Brambilla A; Cereda E; Donetti A
    Agents Actions; 1985 Apr; 16(3-4):173-5. PubMed ID: 2861730
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Studies on histamine H2 receptor antagonists. 2. Synthesis and pharmacological activities of N-sulfamoyl and N-sulfonyl amidine derivatives.
    Yanagisawa I; Hirata Y; Ishii Y
    J Med Chem; 1987 Oct; 30(10):1787-93. PubMed ID: 2888895
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Pseudosymmetry and bioisosterism in biaryl pyridyl competitive histamine H2-receptor antagonists.
    Lipinski CA; LaMattina JL; Hohnke LA
    J Med Chem; 1985 Nov; 28(11):1628-36. PubMed ID: 2866245
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Cyanoguanidine-thiourea equivalence in the development of the histamine H2-receptor antagonist, cimetidine.
    Durant GJ; Emmett JC; Ganellin CR; Miles PD; Parsons ME; Prain HD; White GR
    J Med Chem; 1977 Jul; 20(7):901-6. PubMed ID: 17751
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Pharmacological profile of etintidine, a new histamine H2-receptor antagonist.
    Scott CK; Katz LB; Shriver DA
    Arch Int Pharmacodyn Ther; 1986 May; 281(1):5-21. PubMed ID: 2875695
    [TBL] [Abstract][Full Text] [Related]  

  • 17. FR145715, a novel histamine H2 receptor antagonist, with specific anti-Helicobacter pylori activities.
    Ishikawa H; Ito H; Higaki M; Higaki M; Matsumoto Y; Kamimura T; Katsura Y; Tomishi T; Inoue Y; Takasugi H; Tomoi M; Krakowka S; Yoshida K
    Eur J Pharmacol; 1999 Aug; 378(3):299-310. PubMed ID: 10493106
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Comparison of cimetidine with new H2-antagonists in rabbit and guinea pig gastric cells.
    Batzri S; Harmon JW; Toles R
    Eur J Pharmacol; 1983 Oct; 94(1-2):1-8. PubMed ID: 6140169
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Characterization and development of cimetidine as a histamine H2-receptor antagonist.
    Brimblecombe RW; Duncan WA; Durant GJ; Emmett JC; Ganellin CR; Leslie GB; Parsons ME
    Gastroenterology; 1978 Feb; 74(2 Pt 2):339-47. PubMed ID: 23336
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Pharmacology of ORF 17578, a new histamine H2-receptor antagonist: comparison with cimetidine and ranitidine.
    Katz LB; Scott CK; Shriver DA
    J Pharmacol Exp Ther; 1986 May; 237(2):404-10. PubMed ID: 2871172
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.